General Information of the Compound
Compound ID
CP0372613
Compound Name
8-((2-chloro-4-methylphenyl)(2-chlorophenyl)methyl)-3-(pyrimidin-4-yl)-8-azabicyclo[3.2.1]octan-3-ol
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Structure
Formula
C25H25Cl2N3O
Molecular Weight
454.401
Canonical SMILES
Cc1ccc(C(N2C3CCC2CC(O)(C3)c2ccncn2)c2ccccc2Cl)c(Cl)c1
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InChI
InChI=1S/C25H25Cl2N3O/c1-16-6-9-20(22(27)12-16)24(19-4-2-3-5-21(19)26)30-17-7-8-18(30)14-25(31,13-17)23-10-11-28-15-29-23/h2-6,9-12,15,17-18,24,31H,7-8,13-14H2,1H3
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InChIKey
JKCGUKCHGQOSKC-UHFFFAOYSA-N
Physicochemical Property
logP
5.69582
Rotatable Bonds
4
Heavy Atom Count
31
Polar Areas
49.25
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
4
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44574586
ChEMBL ID
CHEMBL512411
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 535 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 5.2 nM
   TI
   LI
   LO
   TS