General Information of the Compound
Compound ID
CP0357660
Compound Name
6-[1-(cyclopropylmethyl)pyrazol-4-yl]-N-[5-[(3R)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl]pyridine-2-carboxamide
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Structure
Formula
C26H29F3N6O2
Molecular Weight
514.552
Canonical SMILES
CC(C)(O)[C@@H]1CCN(C1)c1cnc(c(NC(=O)c2cccc(n2)-c2cnn(CC3CC3)c2)c1)C(F)(F)F
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InChI
InChI=1S/C26H29F3N6O2/c1-25(2,37)18-8-9-34(15-18)19-10-22(23(30-12-19)26(27,28)29)33-24(36)21-5-3-4-20(32-21)17-11-31-35(14-17)13-16-6-7-16/h3-5,10-12,14,16,18,37H,6-9,13,15H2,1-2H3,(H,33,36)/t18-/m1/s1
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InChIKey
JKIDUHXOZVXHEI-GOSISDBHSA-N
Physicochemical Property
logP
4.6184
Rotatable Bonds
7
Heavy Atom Count
37
Polar Areas
96.17
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 165129719
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01378, Leucine-rich repeat serine/threonine-protein kinase 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000004 SH-SY5Y Homo sapiens (Human)  1
1
IC50 = 0.4 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 8.6 nM