General Information of the Compound
Compound ID
CP0311844
Compound Name
US11078186, Example 119
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Structure
Formula
C29H28F7N3O3
Molecular Weight
599.547
Canonical SMILES
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C(=O)CC#N)c1ccc(F)cc1
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InChI
InChI=1S/C29H28F7N3O3/c1-26(20-6-8-22(30)9-7-20)17-39(25(41)19-11-14-38(15-12-19)24(40)10-13-37)16-23(26)18-2-4-21(5-3-18)27(42,28(31,32)33)29(34,35)36/h2-9,19,23,42H,10-12,14-17H2,1H3/t23-,26+/m0/s1
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InChIKey
JACZDQDBHYAEIU-JYFHCDHNSA-N
Physicochemical Property
logP
5.17388
Rotatable Bonds
5
Heavy Atom Count
42
Polar Areas
84.64
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
4
Complexity
42

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 153313942
ChEMBL ID
CHEMBL4756133
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02658, Nuclear receptor ROR-alpha
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS
Protein ID: PT03033, Nuclear receptor ROR-beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS
Protein ID: PT02663, Nuclear receptor ROR-gamma
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
EC50 = 505 nM
   TI
   LI
   LO
   TS
Protein ID: PT01555, Oxysterols receptor LXR-alpha
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000044 CV-1 Chlorocebus aethiops (Green monkey)  1
1
EC50 = 739 nM
   TI
   LI
   LO
   TS
Protein ID: PT01887, Oxysterols receptor LXR-beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000044 CV-1 Chlorocebus aethiops (Green monkey)  1
1
EC50 = 1130 nM
   TI
   LI
   LO
   TS