General Information of the Compound
Compound ID
CP0281750
Compound Name
1-[[(1R)-1-cyclopropyl-2,2,2-trifluoroethyl]amino]-7-[6-(1,1-dioxo-1,4-thiazinan-4-yl)pyridazin-3-yl]-5H-pyrido[4,3-b]indole-4-carboxamide
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Structure
Formula
C25H24F3N7O3S
Molecular Weight
559.574
Canonical SMILES
NC(=O)c1cnc(N[C@H](C2CC2)C(F)(F)F)c2c3ccc(cc3[nH]c12)-c1ccc(nn1)N1CCS(=O)(=O)CC1
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InChI
InChI=1S/C25H24F3N7O3S/c26-25(27,28)22(13-1-2-13)32-24-20-15-4-3-14(11-18(15)31-21(20)16(12-30-24)23(29)36)17-5-6-19(34-33-17)35-7-9-39(37,38)10-8-35/h3-6,11-13,22,31H,1-2,7-10H2,(H2,29,36)(H,30,32)/t22-/m1/s1
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InChIKey
UJGMROGDTTZZAX-JOCHJYFZSA-N
Physicochemical Property
logP
3.2596
Rotatable Bonds
6
Heavy Atom Count
39
Polar Areas
146.96
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
8
Complexity
39

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 42636019
SID: 81075067
ChEMBL ID
CHEMBL1835152
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01214, Tyrosine-protein kinase JAK2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000082 HEL Homo sapiens (Human)  1
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 2 nM