General Information of the Compound
Compound ID
CP0141066
Compound Name
3-[(1S)-1-(1-cyclopropyl-6-fluorobenzimidazol-2-yl)-2-[1-(2-methylpropanoyl)piperidin-4-yl]ethyl]-1-[4-(4-fluorophenoxy)phenyl]imidazolidine-2,4-dione
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Formula
C36H37F2N5O4
Molecular Weight
641.719
Canonical SMILES
CC(C)C(=O)N1CCC(C[C@H](N2C(=O)CN(C2=O)c2ccc(Oc3ccc(F)cc3)cc2)c2nc3ccc(F)cc3n2C2CC2)CC1
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InChI
InChI=1S/C36H37F2N5O4/c1-22(2)35(45)40-17-15-23(16-18-40)19-32(34-39-30-14-5-25(38)20-31(30)42(34)27-6-7-27)43-33(44)21-41(36(43)46)26-8-12-29(13-9-26)47-28-10-3-24(37)4-11-28/h3-5,8-14,20,22-23,27,32H,6-7,15-19,21H2,1-2H3/t32-/m0/s1
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InChIKey
WSJZBXXQVPZXIT-YTTGMZPUSA-N
Physicochemical Property
logP
7.2363
Rotatable Bonds
9
Heavy Atom Count
47
Polar Areas
87.98
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
6
Complexity
47

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4783205
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01286, Bile acid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000148 Huh-7 Homo sapiens (Human)  1
1
IC50 = 0.05 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 32.9 nM