General Information of the Compound
Compound ID
CP0132360
Compound Name
2-methyl-N-[2-[3-[[2-(prop-2-enoylamino)acetyl]amino]anilino]pyrimidin-5-yl]-5-[[3-(trifluoromethyl)benzoyl]amino]benzamide
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Synonyms
1431727-04-6
BDBM50020476
GTPL8145
PLS-123
PMID24915291C38
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Structure
Formula
C31H26F3N7O4
Molecular Weight
617.588
Canonical SMILES
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1C(=O)Nc1cnc(Nc2cccc(NC(=O)CNC(=O)C=C)c2)nc1
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InChI
InChI=1S/C31H26F3N7O4/c1-3-26(42)35-17-27(43)38-21-8-5-9-22(13-21)41-30-36-15-24(16-37-30)40-29(45)25-14-23(11-10-18(25)2)39-28(44)19-6-4-7-20(12-19)31(32,33)34/h3-16H,1,17H2,2H3,(H,35,42)(H,38,43)(H,39,44)(H,40,45)(H,36,37,41)
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InChIKey
SMOPKEHQPPXRSH-UHFFFAOYSA-N
Physicochemical Property
logP
5.29272
Rotatable Bonds
10
Heavy Atom Count
45
Polar Areas
154.21
Hydrogen Bond Donor Count
5
Hydrogen Bond Acceptor Count
7
Complexity
45

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 71556703
SID: 163556749
ChEMBL ID
CHEMBL3290148
Clinical Information about the Compound
Drug 1 ( PMID24915291C38 )
Drug Name PMID24915291C38
Target(s)
Tyrosine-protein kinase Tec (PSCTK4)
Inhibitor
Tyrosine-protein kinase BTK (ATK)
Inhibitor
B lymphocyte kinase (BLK)
Inhibitor
Erbb4 tyrosine kinase receptor (Erbb-4)
Inhibitor
Tyrosine-protein kinase BMX (BMX)
Inhibitor
Tyrosine-protein kinase TXK (TXK)
Inhibitor
ERBB2 messenger RNA (HER2 mRNA)
Inhibitor
Epidermal growth factor receptor (EGFR)
Inhibitor