General Information of the Compound
Compound ID
CP0127130
Compound Name
5-[[(5S)-5-methyl-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yl]oxy]-N-[3-(trifluoromethyl)phenyl]indole-1-carboxamide
    Show/Hide
Structure
Formula
C23H18F3N5O2
Molecular Weight
453.424
Canonical SMILES
C[C@@H]1NCc2ncnc(Oc3ccc4n(ccc4c3)C(=O)Nc3cccc(c3)C(F)(F)F)c12
    Show/Hide
InChI
InChI=1S/C23H18F3N5O2/c1-13-20-18(11-27-13)28-12-29-21(20)33-17-5-6-19-14(9-17)7-8-31(19)22(32)30-16-4-2-3-15(10-16)23(24,25)26/h2-10,12-13,27H,11H2,1H3,(H,30,32)/t13-/m0/s1
    Show/Hide
InChIKey
IOYGLPLYVXPZNZ-ZDUSSCGKSA-N
Physicochemical Property
logP
5.4868
Rotatable Bonds
3
Heavy Atom Count
33
Polar Areas
81.07
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 127040317
ChEMBL ID
CHEMBL3747182
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
IC50 = 118 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 16 nM