General Information of the Compound
Compound ID
CP0070344
Compound Name
1-cyclopropyl-3-[2-[(2S)-3-(5-fluorospiro[3H-1-benzofuran-2,4'-piperidine]-1'-yl)-2-hydroxypropoxy]-4-methoxyphenyl]urea
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Structure
Formula
C26H32FN3O5
Molecular Weight
485.556
Canonical SMILES
COc1ccc(NC(=O)NC2CC2)c(OC[C@@H](O)CN2CCC3(Cc4cc(F)ccc4O3)CC2)c1
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InChI
InChI=1S/C26H32FN3O5/c1-33-21-5-6-22(29-25(32)28-19-3-4-19)24(13-21)34-16-20(31)15-30-10-8-26(9-11-30)14-17-12-18(27)2-7-23(17)35-26/h2,5-7,12-13,19-20,31H,3-4,8-11,14-16H2,1H3,(H2,28,29,32)/t20-/m0/s1
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InChIKey
FEODIUOQCJLGCM-FQEVSTJZSA-N
Physicochemical Property
logP
3.3276
Rotatable Bonds
8
Heavy Atom Count
35
Polar Areas
92.29
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
6
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 72945511
ChEMBL ID
CHEMBL3099946
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01070, C-C chemokine receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 2.2 nM
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