General Information of the Compound
Compound ID
CP0069691
Compound Name
CHEBI:15640
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Synonyms
[3H]folinic acid
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Structure
Formula
C20H23N7O7
Molecular Weight
473.446
Canonical SMILES
Nc1nc(=O)c2N(C=O)C(CNc3ccc(cc3)C(=O)N[C@@H](CCC(O)=O)C(O)=O)CNc2[nH]1
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InChI
InChI=1S/C20H23N7O7/c21-20-25-16-15(18(32)26-20)27(9-28)12(8-23-16)7-22-11-3-1-10(2-4-11)17(31)24-13(19(33)34)5-6-14(29)30/h1-4,9,12-13,22H,5-8H2,(H,24,31)(H,29,30)(H,33,34)(H4,21,23,25,26,32)/t12?,13-/m0/s1
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InChIKey
VVIAGPKUTFNRDU-ABLWVSNPSA-N
CAS
1958/5/9
Physicochemical Property
logP
-0.7311
Rotatable Bonds
10
Heavy Atom Count
34
Polar Areas
219.84
Hydrogen Bond Donor Count
7
Hydrogen Bond Acceptor Count
9
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 135403648
SID: 15332102
ChEMBL ID
CHEMBL1679
DrugBank ID
DB00650
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01651, Dihydrofolate reductase
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000108 CCRF-CEM Homo sapiens (Human)  1
1
Ki = 2370 nM
   TI
   LI
   LO
   TS
Protein ID: PT06163, Solute carrier organic anion transporter family member 1A3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000031 MDCK Canis lupus familiaris (Dog)  1
1
Ki = 8200 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( [3H]folinic acid )
Drug Name [3H]folinic acid
Target(s)
Proton-coupled folate transporter (SLC46A1)
Modulator