General Information of the Compound
Compound ID
CP0052205
Compound Name
5,5',5''-[1,3,6-naphthalenetriyltris(sulfonylimino)]tris[1,3-benzenesulfonate analogue
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Synonyms
Antrypol
Belganyl
Farma
Farma 939
Fourneau
Germanin
Germanin (TN)
Moranyl
Naganil
Naganin
Naganine
Naganol
Naganol 6 Na
Naphuride
SGCTO-001
SURAMIN SODIUM
SVR
Sodium suramin
Suramin
Suramine
Suramine sodium
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Structure
Formula
C51H40N6O23S6
Molecular Weight
1297.302
Canonical SMILES
Cc1ccc(cc1NC(=O)c1cccc(NC(=O)Nc2cccc(c2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(c3cc(cc(c23)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O)c1)C(=O)Nc1ccc(c2cc(cc(c12)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O
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InChI
InChI=1S/C51H40N6O23S6/c1-25-9-11-29(49(60)54-37-13-15-41(83(69,70)71)35-21-33(81(63,64)65)23-43(45(35)37)85(75,76)77)19-39(25)56-47(58)27-5-3-7-31(17-27)52-51(62)53-32-8-4-6-28(18-32)48(59)57-40-20-30(12-10-26(40)2)50(61)55-38-14-16-42(84(72,73)74)36-22-34(82(66,67)68)24-44(46(36)38)86(78,79)80/h3-24H,1-2H3,(H,54,60)(H,55,61)(H,56,58)(H,57,59)(H2,52,53,62)(H,63,64,65)(H,66,67,68)(H,69,70,71)(H,72,73,74)(H,75,76,77)(H,78,79,80)
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InChIKey
FIAFUQMPZJWCLV-UHFFFAOYSA-N
CAS
145-63-1
Physicochemical Property
logP
6.74324
Rotatable Bonds
16
Heavy Atom Count
86
Polar Areas
483.75
Hydrogen Bond Donor Count
12
Hydrogen Bond Acceptor Count
17
Complexity
86

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 4261196
SID: 14792752
ChEMBL ID
CHEMBL265502
DrugBank ID
DB04786
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03558, P2Y purinoceptor 11
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000094 1321N1 Homo sapiens (Human)  2
1
Ki = 112.2 nM
   TI
   LI
   LO
   TS
2
Ki = 302 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( Suramin )
Drug Name Suramin
Company Bayer Pharmaceuticals Corporation
Indication
African trypanosomiasis
Phase 1
Target(s)
Follicle-stimulating hormone receptor (FSHR)
Antagonist
Heparanase (HPSE)
Inhibitor
Drug 2 ( Suramin )
Drug Name Suramin
Company Bayer Pharmaceuticals Corporation
Indication
African trypanosomiasis
Phase 1
Coronavirus Disease 2019 (COVID-19)
Investigative