General Information of the Compound
Compound ID
CP0041669
Compound Name
(R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimethyl-4-(2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl)-1H-pyrrol-2-yl)methylene)indolin-2-one
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Synonyms
(2R)-1-[[5-[(Z)-[5-[[(2,6-DICHLOROPHENYL)METHYL]SULFONYL]-1,2-DIHYDRO-2-OXO-3H-INDOL-3-YLIDENE]METHYL]-2,4-DIMETHYL-1H-PYRROL-3-YL]CARBONYL]-2-(1-PYRROLIDINYLMETHYL)PYRROLIDINE
(R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimethyl-4-(2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl)-1H-pyrrol-2-yl)methylene)indolin-2-one
0VXU5T5R3J
477575-56-7
CHEBI:90197
CHEMBL450786
PHA 665752
PHA-665752
PHA-665752 hydrate
PHA665752
TCMDC-125885
UNII-0VXU5T5R3J
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Structure
Formula
C32H34Cl2N4O4S
Molecular Weight
641.621
Canonical SMILES
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1
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InChI
InChI=1S/C32H34Cl2N4O4S/c1-19-29(35-20(2)30(19)32(40)38-14-6-7-21(38)17-37-12-3-4-13-37)16-24-23-15-22(10-11-28(23)36-31(24)39)43(41,42)18-25-26(33)8-5-9-27(25)34/h5,8-11,15-16,21,35H,3-4,6-7,12-14,17-18H2,1-2H3,(H,36,39)/b24-16-/t21-/m1/s1
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InChIKey
OYONTEXKYJZFHA-SSHUPFPWSA-N
Physicochemical Property
logP
6.10534
Rotatable Bonds
7
Heavy Atom Count
43
Polar Areas
102.58
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
5
Complexity
43

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 10461815
SID: 15483678
ChEMBL ID
CHEMBL450786
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01201, Hepatocyte growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549 Homo sapiens (Human)  1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CL000282 GTL-16 Homo sapiens (Human)  1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 38 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 42 nM
2 IC50 = 9 nM
3 IC50 = 38 nM
4 Kd = 0.27 nM
5 Kd = 0.64 nM
6 Kd = 0.83 nM
Clinical Information about the Compound
Drug 1 ( PHA-665752 )
Drug Name PHA-665752
Company Pfizer Inc
Indication
Solid tumour/cancer
Investigative
Target(s)
Proto-oncogene c-Met (MET)
Inhibitor