General Information of the Compound
Compound ID
CP0014495
Compound Name
4-[2-[6-(4-methylpiperazine-1-carbonyl)naphthalen-2-yl]ethylamino]quinazoline-6-carbonitrile
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Synonyms
PMID26161698-Compound-47
Quinazoline derivative 9
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Structure
Formula
C27H26N6O
Molecular Weight
450.546
Canonical SMILES
CN1CCN(CC1)C(=O)c1ccc2cc(CCNc3ncnc4ccc(cc34)C#N)ccc2c1
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InChI
InChI=1S/C27H26N6O/c1-32-10-12-33(13-11-32)27(34)23-6-5-21-14-19(2-4-22(21)16-23)8-9-29-26-24-15-20(17-28)3-7-25(24)30-18-31-26/h2-7,14-16,18H,8-13H2,1H3,(H,29,30,31)
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InChIKey
VNADJTWHOAMTLY-UHFFFAOYSA-N
CAS
1449228-40-3
Physicochemical Property
logP
3.69688
Rotatable Bonds
5
Heavy Atom Count
34
Polar Areas
85.15
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 71661259
ChEMBL ID
CHEMBL4076837
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00926, Cyclin-dependent kinase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000156 HT-1080 Homo sapiens (Human)  1
1
EC50 = 530 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( Quinazoline derivative 9 )
Drug Name Quinazoline derivative 9
Company SENEX BIOTECHNOLOGY INC
Indication
Breast cancer
Phase 1
Target(s)
MEK kinase kinase 2 (MAP4K2)
Inhibitor
SPS1/STE20-related protein kinase YSK4 (YSK4)
Inhibitor