| Compound ID |
Compound Name |
Compound Formula |
|
CP0545265
|
N-[4-[[2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]-2-methoxyphenyl]-1-(3-fluoropropyl)azetidin-3-amine
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|
C30H28F4N4O2S
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
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CP0551988
|
2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-3-[4-[1-(3-fluoropropyl)azetidin-3-yl]oxy-3-methoxyphenoxy]-6H-thieno[2,3-e]indazole
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|
C30H27F4N3O3S
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
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CP0573007
|
N-[4-[[2-[4-fluoro-2-(2-fluoropropan-2-yl)phenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]-2-methoxyphenyl]-1-(3-fluoropropyl)azetidin-3-amine
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|
C31H31F3N4O2S
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
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CP0569178
|
2-[4-fluoro-2-(2-fluoropropan-2-yl)phenyl]-3-[4-[1-(3-fluoropropyl)azetidin-3-yl]oxy-3-methoxyphenoxy]-6H-thieno[2,3-e]indazole
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|
C31H30F3N3O3S
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
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CP0569393
|
3-[4-[1-(3-fluoropropyl)azetidin-3-yl]oxy-3-methoxyphenoxy]-2-[4-fluoro-2-(2,2,2-trifluoroethyl)phenyl]-6H-thieno[2,3-e]indazole
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|
C30H26F5N3O3S
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0043589
|
(13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pentane-1-sulfinyl)-nonyl]-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthrene-3,17-diol
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|
C32H47F5O3S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0568297
|
2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-3-[3-fluoro-4-[1-(3-fluoropropyl)azetidin-3-yl]oxyphenoxy]-6H-thieno[2,3-e]indazole
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|
C29H24F5N3O2S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0576564
|
N-[4-[[2-[4-fluoro-2-(2-fluoropropan-2-yl)phenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]phenyl]-1-(3-fluoropropyl)azetidin-3-amine
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|
C30H29F3N4OS
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0543544
|
N-[4-[[2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]-2-fluorophenyl]-1-(3-fluoropropyl)azetidin-3-amine
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|
C29H25F5N4OS
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0568767
|
1-(3-fluoropropyl)-N-[4-[[2-[4-fluoro-2-(2,2,2-trifluoroethyl)phenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]-2-methoxyphenyl]azetidin-3-amine
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|
C30H27F5N4O2S
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0568223
|
2-[4-fluoro-2-(2-fluoropropan-2-yl)phenyl]-3-[3-fluoro-4-[1-(3-fluoropropyl)azetidin-3-yl]oxyphenoxy]-6H-thieno[2,3-e]indazole
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|
C30H27F4N3O2S
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0571259
|
1-(3-fluoropropyl)-N-[4-[[2-[4-fluoro-2-(2,2,2-trifluoroethyl)phenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]phenyl]azetidin-3-amine
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|
C29H25F5N4OS
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
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CP0551915
|
2-[2-(1,1-difluoroethyl)-4,5-difluorophenyl]-3-[4-[1-(3-fluoropropyl)azetidin-3-yl]oxy-3-methoxyphenoxy]-6H-thieno[2,3-e]indazole
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|
C30H26F5N3O3S
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0571814
|
3-[3-fluoro-4-[1-(3-fluoropropyl)azetidin-3-yl]oxyphenoxy]-2-[4-fluoro-2-(2,2,2-trifluoroethyl)phenyl]-6H-thieno[2,3-e]indazole
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|
C29H23F6N3O2S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0546742
|
N-[4-[[2-[2-(1,1-difluoroethyl)-4,5-difluorophenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]-2-methoxyphenyl]-1-(3-fluoropropyl)azetidin-3-amine
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|
C30H27F5N4O2S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0571248
|
2-[2-(1,1-difluoroethyl)-4,5-difluorophenyl]-3-[4-[1-(3-fluoropropyl)azetidin-3-yl]oxyphenoxy]-6H-thieno[2,3-e]indazole
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|
C29H24F5N3O2S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
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CP0569727
|
N-[4-[[2-[2-(1,1-difluoroethyl)-4,5-difluorophenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]phenyl]-1-(3-fluoropropyl)azetidin-3-amine
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|
C29H25F5N4OS
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
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CP0545402
|
2-[2-(1,1-difluoroethyl)-4,5-difluorophenyl]-3-[3-fluoro-4-[1-(3-fluoropropyl)azetidin-3-yl]oxyphenoxy]-6H-thieno[2,3-e]indazole
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|
C29H23F6N3O2S
|
1
|
| 1 |
IC50 = 5.3 nM
|
|
|
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CP0543545
|
(E)-3-[4-[[2-[3-(1,1-difluoroethyl)-4-fluorophenyl]-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]prop-2-enoic acid
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|
C25H17F3O4S
|
1
|
| 1 |
IC50 = 6.5 nM
|
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