| Compound ID |
Compound Name |
Compound Formula |
|
CP0478532
|
4-[4-(3-hydroxypropoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C30H34O4
|
1
|
| 1 |
EC50 = 0.22 nM
|
|
|
|
CP0394515
|
4-[4-(4-hydroxybutoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C31H36O4
|
1
|
| 1 |
EC50 = 0.92 nM
|
|
|
|
CP0511782
|
4-[4-(2-hydroxyethyl)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C29H32O3
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0414095
|
4-[3-[3-tert-butyl-4-(diethylamino)phenyl]-4-(3-hydroxypropoxy)phenyl]benzoic acid
Show/Hide
|
C30H37NO4
|
1
|
| 1 |
EC50 = 1.9 nM
|
|
|
|
CP0414087
|
4-[4-methoxy-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C28H30O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0409710
|
4-[3-(3-tert-butyl-4-pyrrolidin-1-ylphenyl)-4-(3-hydroxypropoxy)phenyl]benzoic acid
Show/Hide
|
C30H35NO4
|
1
|
| 1 |
EC50 = 2.1 nM
|
|
|
|
CP0076073
|
6-(3-(1-Adamantyl)-4-methoxyphenyl)-2-naphthoic acid
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|
C28H28O3
|
1
|
| 1 |
EC50 = 3.1 nM
|
|
|
|
CP0405756
|
4-[3-[3-tert-butyl-4-(diethylamino)phenyl]-4-(2-hydroxyethoxy)phenyl]benzoic acid
Show/Hide
|
C29H35NO4
|
1
|
| 1 |
EC50 = 3.6 nM
|
|
|
|
CP0414094
|
4-[4-(hydroxymethyl)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C28H30O3
|
1
|
| 1 |
EC50 = 4.4 nM
|
|
|
|
CP0409711
|
4-[3-[3-tert-butyl-4-(diethylamino)phenyl]-4-(4-hydroxybutoxy)phenyl]benzoic acid
Show/Hide
|
C31H39NO4
|
1
|
| 1 |
EC50 = 4.7 nM
|
|
|
|
CP0542889
|
4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C31H36O5
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0542914
|
4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]-2-methylbenzoic acid
Show/Hide
|
C32H38O5
|
1
|
| 1 |
EC50 = 7.4 nM
|
|
|
|
CP0414091
|
CD-5789
Show/Hide
|
C29H33NO4
|
1
|
| 1 |
EC50 = 7.7 nM
|
|
|
|
CP0414093
|
4-[4-[3-(cyclopropylamino)propoxy]-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C33H39NO3
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0425258
|
4-[3-(3-tert-butyl-4-pyrrolidin-1-ylphenyl)-4-(4-hydroxybutoxy)phenyl]benzoic acid
Show/Hide
|
C31H37NO4
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0394517
|
6-[2-(4,4-dimethyl-2,3-dihydrothiochromen-6-yl)ethynyl]pyridine-2-carboxylic acid
Show/Hide
|
C19H17NO2S
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0569823
|
2-chloro-4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C31H35ClO5
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0387569
|
4-[3-[4-(diethylamino)-3-ethylphenyl]-4-(3-hydroxypropoxy)phenyl]benzoic acid
Show/Hide
|
C28H33NO4
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0414097
|
4-[4-hydroxy-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C27H28O3
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0151451
|
CD666
Show/Hide
|
C24H28O3
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0394516
|
3-methoxy-4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C32H38O6
|
1
|
| 1 |
EC50 = 47 nM
|
|
|
|
CP0047520
|
6-(3-Adamantan-1-yl-4-hydroxy-phenyl)-naphthalene-2-carboxylic acid
Show/Hide
|
C27H26O3
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0414096
|
US9963439, BMS961
Show/Hide
|
C23H26FNO4
|
1
|
| 1 |
EC50 = 51 nM
|
|
|
|
CP0447781
|
4-[4-(4-hydroxybutoxy)-3-[4-pyrrolidin-1-yl-3-(trifluoromethyl)phenyl]phenyl]benzoic acid
Show/Hide
|
C28H28F3NO4
|
1
|
| 1 |
EC50 = 53 nM
|
|
|
|
CP0414088
|
4-[3-chloro-4-(2-methoxyethoxymethoxy)-5-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C31H35ClO5
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0476675
|
4-[3-[3-tert-butyl-4-(4-hydroxybutylamino)phenyl]-4-(2-hydroxyethoxy)phenyl]benzoic acid
Show/Hide
|
C29H35NO5
|
1
|
| 1 |
EC50 = 67 nM
|
|
|
|
CP0577998
|
6-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]pyridine-3-carboxylic acid
Show/Hide
|
C30H35NO5
|
1
|
| 1 |
EC50 = 85 nM
|
|
|
|
CP0414089
|
4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]-3-methylbenzoic acid
Show/Hide
|
C32H38O5
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0575892
|
2-methoxy-4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C32H38O6
|
1
|
| 1 |
EC50 = 168 nM
|
|
|
|
CP0543343
|
3-fluoro-4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C31H35FO5
|
1
|
| 1 |
EC50 = 279 nM
|
|
|
|
CP0476105
|
4-[3-[4-(diethylamino)phenyl]-4-(3-hydroxypropoxy)phenyl]benzoic acid
Show/Hide
|
C26H29NO4
|
1
|
| 1 |
EC50 = 353 nM
|
|
|
|
CP0569822
|
3-chloro-4-[4-(2-methoxyethoxymethoxy)-3-(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)phenyl]benzoic acid
Show/Hide
|
C31H35ClO5
|
1
|
| 1 |
EC50 = 422 nM
|
|
|
|
CP0387570
|
4-[3-[3-tert-butyl-4-(2-oxopyrrolidin-1-yl)phenyl]-4-(2-hydroxyethoxy)phenyl]benzoic acid
Show/Hide
|
C29H31NO5
|
1
|
| 1 |
EC50 = 918 nM
|
|
|
|
CP0414098
|
4-[3-(3-tert-butyl-4-pyrrolidin-1-ylphenyl)-4-(carboxymethoxy)phenyl]benzoic acid
Show/Hide
|
C29H31NO5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0446009
|
4-[3-(2,6-dichlorophenoxy)-4-fluoroindazol-1-yl]benzoic acid
Show/Hide
|
C20H11Cl2FN2O3
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0545410
|
4-[3-(2,6-dichlorophenoxy)-4-methylindazol-1-yl]benzoic acid
Show/Hide
|
C21H14Cl2N2O3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0326782
|
4-[1-(2,6-dichlorobenzoyl)indazol-3-yl]benzoic acid
Show/Hide
|
C21H12Cl2N2O3
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0446010
|
4-[5-cyano-3-(2,6-dichlorophenoxy)indazol-1-yl]benzoic acid
Show/Hide
|
C21H11Cl2N3O3
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0504410
|
4-[3-(2,6-dichlorophenoxy)indazol-1-yl]benzoic acid
Show/Hide
|
C20H12Cl2N2O3
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0517633
|
6-[3-(2,6-dichlorophenoxy)indazol-1-yl]pyridine-3-carboxylic acid
Show/Hide
|
C19H11Cl2N3O3
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0516068
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-(methylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C22H15Cl2N3O3S
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0451919
|
4-[5-(dimethylcarbamoyl)-3-phenylsulfanylindazol-1-yl]benzoic acid
Show/Hide
|
C23H19N3O3S
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0508491
|
4-[3-(2,6-dichlorophenoxy)pyrazolo[3,4-b]pyridin-1-yl]benzoic acid
Show/Hide
|
C19H11Cl2N3O3
|
1
|
| 1 |
IC50 = 3800 nM
|
|
|
|
CP0451776
|
4-[5-(azetidine-1-carbonyl)-3-(2,6-dichlorophenyl)sulfanylindazol-1-yl]benzoic acid
Show/Hide
|
C24H17Cl2N3O3S
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0446008
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-(morpholine-4-carbonyl)indazol-1-yl]benzoic acid
Show/Hide
|
C25H19Cl2N3O4S
|
1
|
| 1 |
IC50 = 4200 nM
|
|
|
|
CP0432212
|
4-[3-(2,6-dichlorophenyl)sulfanylindazol-1-yl]benzoic acid
Show/Hide
|
C20H12Cl2N2O2S
|
1
|
| 1 |
IC50 = 4400 nM
|
|
|
|
CP0451926
|
4-[3-(2,6-dichlorophenoxy)-5-methylsulfonylindazol-1-yl]benzoic acid
Show/Hide
|
C21H14Cl2N2O5S
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0447694
|
4-[3-(2,6-dichlorophenyl)sulfinylindazol-1-yl]benzoic acid
Show/Hide
|
C20H12Cl2N2O3S
|
1
|
| 1 |
IC50 = 5600 nM
|
|
|
|
CP0562932
|
3-(2,6-dichlorophenoxy)-1H-indazole
Show/Hide
|
C13H8Cl2N2O
|
1
|
| 1 |
IC50 = 5700 nM
|
|
|
|
CP0388520
|
4-[3-(2,6-dichlorophenoxy)indazol-1-yl]-3-methylbenzoic acid
Show/Hide
|
C21H14Cl2N2O3
|
1
|
| 1 |
IC50 = 6200 nM
|
|
|
|
CP0505232
|
4-[3-[(2,6-dichlorophenyl)methyl]indazol-1-yl]benzoic acid
Show/Hide
|
C21H14Cl2N2O2
|
1
|
| 1 |
IC50 = 6800 nM
|
|
|
|
CP0518039
|
4-[3-(2,6-dichlorophenoxy)pyrazolo[4,3-b]pyridin-1-yl]benzoic acid
Show/Hide
|
C19H11Cl2N3O3
|
1
|
| 1 |
IC50 = 6800 nM
|
|
|
|
CP0452052
|
4-[3-[2-chloro-6-(trifluoromethyl)phenoxy]-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C24H17ClF3N3O4
|
1
|
| 1 |
IC50 = 7200 nM
|
|
|
|
CP0451777
|
4-[3-(2,6-dichlorophenoxy)-7-fluoroindazol-1-yl]benzoic acid
Show/Hide
|
C20H11Cl2FN2O3
|
1
|
| 1 |
IC50 = 7600 nM
|
|
|
|
CP0534631
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-(4-methylpiperazine-1-carbonyl)indazol-1-yl]benzoic acid
Show/Hide
|
C26H22Cl2N4O3S
|
1
|
| 1 |
IC50 = 7700 nM
|
|
|
|
CP0545409
|
4-[3-(2,6-dichlorophenyl)sulfonylindazol-1-yl]benzoic acid
Show/Hide
|
C20H12Cl2N2O4S
|
1
|
| 1 |
IC50 = 8400 nM
|
|
|
|
CP0551474
|
4-[3-(3,5-diethyl-1-methylpyrazol-4-yl)oxyindazol-1-yl]benzoic acid
Show/Hide
|
C22H22N4O3
|
1
|
| 1 |
IC50 = 9100 nM
|
|
|
|
CP0053566
|
N-[5-(2-chlorobenzoyl)-4-(3-chlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
Show/Hide
|
C26H20Cl2N2O4S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0350381
|
2-[2-[(S)-(3,5-dimethyl-1,2-oxazol-4-yl)-hydroxymethyl]-1-benzofuran-5-yl]-N-[(S)-(2,4-dimethylphenyl)-phenylmethyl]acetamide
Show/Hide
|
C31H30N2O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0388523
|
5-[3-(2,6-dichlorophenoxy)indazol-1-yl]pyridine-2-carboxylic acid
Show/Hide
|
C19H11Cl2N3O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0445999
|
4-[3-(2,6-dichlorophenoxy)-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0446001
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0446005
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-[ethyl(methyl)carbamoyl]indazol-1-yl]benzoic acid
Show/Hide
|
C24H19Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0446006
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-(pyrrolidine-1-carbonyl)indazol-1-yl]benzoic acid
Show/Hide
|
C25H19Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0447695
|
4-[1-(2,6-dichlorobenzoyl)-6-(dimethylcarbamoyl)indazol-3-yl]benzoic acid
Show/Hide
|
C24H17Cl2N3O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0447696
|
4-[3-(2-chloro-6-methylphenoxy)-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C24H20ClN3O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0451751
|
4-[3-(2,6-dichlorophenyl)sulfonyl-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0451752
|
4-[5-(dimethylcarbamoyl)-3-(2-methylphenyl)sulfanylindazol-1-yl]benzoic acid
Show/Hide
|
C24H21N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0451753
|
4-[3-(2,4-dichlorophenyl)sulfanyl-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0451778
|
4-[3-(2,6-dichlorophenoxy)indazol-1-yl]-3,5-difluorobenzoic acid
Show/Hide
|
C20H10Cl2F2N2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0451781
|
4-[3-(2,6-dichlorophenoxy)indazol-1-yl]cyclohexane-1-carboxylic acid
Show/Hide
|
C20H18Cl2N2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0451920
|
4-[3-(2,6-dichlorophenoxy)-6-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0451923
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-(3,3-difluoroazetidine-1-carbonyl)indazol-1-yl]benzoic acid
Show/Hide
|
C24H15Cl2F2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0455016
|
4-[3-(2,6-dichlorophenyl)sulfinyl-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0455017
|
4-[3-(2,6-dichloroanilino)-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H18Cl2N4O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0466958
|
4-[3-(2,6-dichlorophenoxy)-7-methylindazol-1-yl]benzoic acid
Show/Hide
|
C21H14Cl2N2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0504412
|
4-[3-(2,6-dichlorophenoxy)indazol-1-yl]-3-fluorobenzoic acid
Show/Hide
|
C20H11Cl2FN2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0516069
|
4-[3-(2,6-dichloroanilino)indazol-1-yl]benzoic acid
Show/Hide
|
C20H13Cl2N3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0516070
|
4-[3-(2-chloro-6-fluorophenyl)sulfanyl-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17ClFN3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0516071
|
4-[3-(2,5-dichlorophenyl)sulfanyl-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0516072
|
4-[3-(2,6-dichlorophenoxy)indazol-1-yl]cyclohexane-1-carboxylic acid
Show/Hide
|
C20H18Cl2N2O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0529159
|
4-[3-(2,3-dichlorophenyl)sulfanyl-5-(dimethylcarbamoyl)indazol-1-yl]benzoic acid
Show/Hide
|
C23H17Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0532760
|
4-[5-(dimethylcarbamoyl)-3-(2,6-dimethylphenyl)sulfanylindazol-1-yl]benzoic acid
Show/Hide
|
C25H23N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0532761
|
4-[5-(dimethylcarbamoyl)-3-(2,4,6-trimethylphenyl)sulfanylindazol-1-yl]benzoic acid
Show/Hide
|
C26H25N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
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CP0532762
|
4-[3-(2,6-dichlorophenyl)sulfanyl-5-[2-hydroxyethyl(methyl)carbamoyl]indazol-1-yl]benzoic acid
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|
C24H19Cl2N3O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0539695
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4-[5-[benzyl(methyl)carbamoyl]-3-(2,6-dichlorophenyl)sulfanylindazol-1-yl]benzoic acid
Show/Hide
|
C29H21Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0405429
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N-(4-ethylphenyl)-N-(2-methylpropyl)-3-(methylsulfonimidoyl)-4-(oxan-4-ylmethoxy)benzenesulfonamide
Show/Hide
|
C25H36N2O5S2
|
1
|
| 1 |
IC50 > 10000 nM
|
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