Compound ID |
Compound Name |
Compound Formula |
CP0424056
|
1,3-dimethyl-5-(7-methyl-2-piperidin-4-ylindazol-5-yl)pyridin-2-one
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|
C20H24N4O
|
1
|
1 |
IC50 = 250 nM
|
|
|
CP0531875
|
5-[2-(4-cyclobutylpiperazin-1-yl)quinazolin-6-yl]-1-methylpyridin-2-one
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|
C22H25N5O
|
1
|
1 |
IC50 = 1400 nM
|
|
|
CP0409312
|
1-methyl-5-(7-methyl-2-piperidin-4-ylindazol-5-yl)pyridin-2-one
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|
C19H22N4O
|
1
|
1 |
IC50 = 1600 nM
|
|
|
CP0424053
|
1-methyl-5-[8-methyl-2-(4-propan-2-ylpiperazin-1-yl)quinazolin-6-yl]pyridin-2-one
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|
C22H27N5O
|
1
|
1 |
IC50 = 5900 nM
|
|
|
CP0525568
|
1,6-dimethyl-5-(7-methyl-2-piperidin-4-ylindazol-5-yl)pyridin-2-one
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|
C20H24N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0528718
|
5-methoxy-6-pyridin-4-yl-1H-indole
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|
C14H12N2O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0409314
|
1,4-dimethyl-5-(7-methyl-2-piperidin-4-ylindazol-5-yl)pyridin-2-one
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|
C20H24N4O
|
1
|
1 |
IC50 > 4200 nM
|
|
|
CP0424067
|
8-[2-[(3S,4S)-3-fluoropiperidin-4-yl]-7-(trifluoromethyl)indazol-5-yl]-2,3-dihydro-1H-indolizin-5-one
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|
C21H20F4N4O
|
1
|
1 |
IC50 > 6500 nM
|
|
|
CP0941521
|
5-cyclopropyl-6-(2,6-dimethylpyridin-4-yl)-N-((3R,4R)-3-fluoropiperidin-4-yl)-1H-indazol-3-amine
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|
C22H26FN5
|
1
|
1 |
IC50 > 8000 nM
|
|
|