Brief Information of the Cell Line and Protein
Cell Line ID: CL000749 , HUVEC-C
Synonyms
HUV-EC-C
HUVEC
Category Finite cell line
Organism
Homo sapiens (Human)
Protein ID: PT04124 , Proteinase-activated receptor 2
Gene Name F2RL1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P55085
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000749  Protein ID: PT04124
 
Compound ID Compound Name Compound Formula
CP0528563
2-[(2S,5R,8S,11S)-5-benzyl-8-[[1-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[(2S)-2-cyclohexyl-2-[[(2S)-3-cyclohexyl-2-(1,2-oxazole-5-carbonylamino)propanoyl]amino]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]methyl]-11-[3-(diaminomethylideneamino)propyl]-3,6,12,15-tetraoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid;2,2,2-trifluoroacetic acid
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C75H114F9N15O26
 1
1
EC50 = 90 nM
   TI
   LI
   LO
   TS
CP0557269
2-[(2S,5R,8S,11S)-5-benzyl-8-[[1-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[(2S)-2-cyclohexyl-2-[[(2S)-3-cyclohexyl-2-(1,2-oxazole-5-carbonylamino)propanoyl]amino]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]methyl]-11-[3-(diaminomethylideneamino)propyl]-3,6,12,15-tetraoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid;2,2,2-trifluoroacetic acid
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C71H112F3N15O22
 1
1
EC50 = 1000 nM
   TI
   LI
   LO
   TS