| Compound ID |
Compound Name |
Compound Formula |
|
CP0421620
|
3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-methyl-3-(((R)-4-methyl-1,1-dioxido-3,4-dihydro-2H-benzo[b][1,4,5]oxathiazepin-2-yl)methyl)phenyl)propanoic acid
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|
C28H30N4O6S
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0421621
|
3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-methyl-3-((4-methyl-1,1-dioxido-3,4-dihydro-2H-benzo[b][1,4,5]oxathiazepin-2-yl)methyl)phenyl)propanoic acid
Show/Hide
|
C28H30N4O6S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0574553
|
5-[(1S,2S)-2-(1-methyltriazol-4-yl)cyclopropyl]-1-[3-[3-[(2R)-2-propylpiperidine-1-carbonyl]phenyl]phenyl]pyrazole-4-carboxylic acid
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|
C31H34N6O3
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0421630
|
BDBM304749
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|
C28H30N4O6S
|
1
|
| 1 |
EC50 = 83 nM
|
|
|
|
CP0573654
|
5-[2-(1-methyltriazol-4-yl)cyclopropyl]-1-[3-[3-(2-propylpiperidine-1-carbonyl)phenyl]phenyl]pyrazole-4-carboxylic acid
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|
C31H34N6O3
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0421619
|
3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-methyl-3-((5-methyl-1,1-dioxido-4,5-dihydrobenzo[f][1,2,5]thiadiazepin-2(3H)-yl)methyl)phenyl)propanoic acid
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|
C28H31N5O5S
|
1
|
| 1 |
EC50 = 570 nM
|
|
|
|
CP0421628
|
3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-methyl-3-(((S)-4-methyl-1,1-dioxido-3,4-dihydro-2H-benzo[b][1,4,5]oxathiazepin-2-yl)methyl)phenyl)propanoic acid
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|
C28H30N4O6S
|
1
|
| 1 |
EC50 = 760 nM
|
|
|
|
CP0471989
|
3-(7-methoxy-1-methyl-1H-1,2,3-benzotriazol-5-yl)-3-{4-methyl-3-[(N-methylbenzenesulfonamido)methyl]phenyl}propanoic acid
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|
C26H28N4O5S
|
1
|
| 1 |
EC50 = 850 nM
|
|
|
|
CP0577668
|
5-cyclopropyl-1-[3-[3-(dimethylcarbamoyl)-2-fluorophenyl]phenyl]pyrazole-4-carboxylic acid
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|
C22H20FN3O3
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0530245
|
3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-methyl-3-((3-methyl-1,1-dioxido-3,4-dihydro-2H-benzo[b][1,4,5]oxathiazepin-2-yl)methyl)phenyl)propanoic acid
Show/Hide
|
C28H30N4O6S
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0573651
|
5-cyclopropyl-1-[3-[3-(dimethylcarbamoyl)phenyl]phenyl]pyrazole-4-carboxylic acid
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|
C22H21N3O3
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0530244
|
3-(3-((1,1-dioxido-3,4-dihydro-2H-benzo[b][1,4,5]oxathiazepin-2-yl)methyl)-4-methylphenyl)-3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)propanoic acid
Show/Hide
|
C27H28N4O6S
|
1
|
| 1 |
EC50 = 1600 nM
|
|
|
|
CP0577661
|
5-cyclopropyl-1-[3-[(1R,3S)-3-(dimethylcarbamoyl)cyclohexyl]phenyl]pyrazole-4-carboxylic acid
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|
C22H27N3O3
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0580065
|
5-cyclopropyl-1-[3-[3-[cyclopropylmethyl(methyl)carbamoyl]-2-fluorophenyl]phenyl]pyrazole-4-carboxylic acid
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|
C25H24FN3O3
|
1
|
| 1 |
EC50 = 2200 nM
|
|
|
|
CP0571260
|
5-cyclopropyl-1-[3-[2-fluoro-3-(piperidine-1-carbonyl)phenyl]phenyl]pyrazole-4-carboxylic acid
Show/Hide
|
C25H24FN3O3
|
1
|
| 1 |
EC50 = 2300 nM
|
|
|
|
CP0543319
|
5-cyclopropyl-1-[3-[2-fluoro-3-(3-propylmorpholine-4-carbonyl)phenyl]phenyl]pyrazole-4-carboxylic acid
Show/Hide
|
C27H28FN3O4
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
|
CP0574551
|
5-cyclopropyl-1-[3-[(1R,3S)-3-(piperidine-1-carbonyl)cyclohexyl]phenyl]pyrazole-4-carboxylic acid
Show/Hide
|
C25H31N3O3
|
1
|
| 1 |
EC50 = 2700 nM
|
|
|
|
CP0577662
|
1-[3-[3-(2-propylpiperidine-1-carbonyl)phenyl]phenyl]-5-(2-pyridazin-3-ylcyclopropyl)pyrazole-4-carboxylic acid
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|
C32H33N5O3
|
1
|
| 1 |
EC50 = 2800 nM
|
|
|
|
CP0533586
|
3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(3-((4-methyl-1,1-dioxido-3,4-dihydro-2H-benzo[b][1,4,5]oxathiazepin-2-yl)methyl)phenyl)propanoic acid
Show/Hide
|
C27H28N4O6S
|
1
|
| 1 |
EC50 = 2900 nM
|
|
|
|
CP0577110
|
1-[3-[3-(2-propylpiperidine-1-carbonyl)phenyl]phenyl]-5-(2-pyridin-3-ylcyclopropyl)pyrazole-4-carboxylic acid
Show/Hide
|
C33H34N4O3
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
|
CP0471987
|
3-[3-[[benzenesulfonyl(methyl)amino]methyl]-4-methylphenyl]-3-(1-methylbenzotriazol-5-yl)propanoic acid
Show/Hide
|
C25H26N4O4S
|
1
|
| 1 |
EC50 = 3400 nM
|
|
|
|
CP0545153
|
5-cyclopropyl-1-[3-[2-fluoro-3-[(2R)-2-propylpiperidine-1-carbonyl]phenyl]phenyl]pyrazole-4-carboxylic acid
Show/Hide
|
C28H30FN3O3
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0577660
|
1-[3-[3-[bis(cyclopropylmethyl)carbamoyl]-2-fluorophenyl]phenyl]-5-cyclopropylpyrazole-4-carboxylic acid
Show/Hide
|
C28H28FN3O3
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0579640
|
5-cyclopropyl-1-[3-[2-fluoro-3-[(2S)-2-propylpiperidine-1-carbonyl]phenyl]phenyl]pyrazole-4-carboxylic acid
Show/Hide
|
C28H30FN3O3
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0579200
|
1-[3-[3-(7-azaspiro[4.5]decane-7-carbonyl)-2-fluorophenyl]phenyl]-5-cyclopropylpyrazole-4-carboxylic acid
Show/Hide
|
C29H30FN3O3
|
1
|
| 1 |
EC50 = 3700 nM
|
|
|
|
CP0551755
|
1-[3-[3-(2-propylpiperidine-1-carbonyl)phenyl]phenyl]-5-(2-pyridin-2-ylcyclopropyl)pyrazole-4-carboxylic acid
Show/Hide
|
C33H34N4O3
|
1
|
| 1 |
EC50 = 3800 nM
|
|
|
|
CP0579086
|
5-cyclopropyl-1-[3-[3-(2-propylpiperidine-1-carbonyl)cyclohexyl]phenyl]pyrazole-4-carboxylic acid
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|
C28H37N3O3
|
1
|
| 1 |
EC50 = 4100 nM
|
|
|
|
CP0579201
|
1-[3-[(1R,3S)-3-[(2R)-2-butylpyrrolidine-1-carbonyl]cyclohexyl]phenyl]-5-cyclopropylpyrazole-4-carboxylic acid
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
EC50 = 4300 nM
|
|
|
|
CP0573653
|
1-[3-[3-(2-butylpyrrolidine-1-carbonyl)cyclohexyl]phenyl]-5-cyclopropylpyrazole-4-carboxylic acid
Show/Hide
|
C28H37N3O3
|
1
|
| 1 |
EC50 = 4400 nM
|
|
|
|
CP0574552
|
5-[(1R,2R)-2-(1-methyltriazol-4-yl)cyclopropyl]-1-[3-[3-[(2R)-2-propylpiperidine-1-carbonyl]phenyl]phenyl]pyrazole-4-carboxylic acid
Show/Hide
|
C31H34N6O3
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
