Brief Information of the Cell Line and Protein
Cell Line ID: CL000524 , HEK293-FT
Synonyms
HEK-293FT
HEK 293FT
HEK-293-FT
HEK293FT
293-FT
293FT
FT-293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_6911
Protein ID: PT01839 , Vasopressin V1a receptor
Gene Name AVPR1A
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P37288
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000524  Protein ID: PT01839
 
Compound ID Compound Name Compound Formula
CP0117986
(2S)-1-[(4R,7S,10S,13S,16S,19R)-19-amino-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13-[(2S)-butan-2-yl]-16-[(4-hydroxyphenyl)methyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]-N-[(2S)-1-[(2-amino-2-oxoethyl)amino]-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamide
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C43H66N12O12S2
 1
1
EC50 = 260 nM
   TI
   LI
   LO
   TS
CP0405331
(2S)-2-(dimethylcarbamothioyl)-N-[[2-methyl-4-(1-methyl-4,10-dihydropyrazolo[4,3-c][1,5]benzodiazepine-5-carbonyl)phenyl]methyl]pyrrolidine-1-carboxamide
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C28H33N7O2S
 2
1
IC50 = 2200 nM
   TI
   LI
   LO
   TS
2
IC50 = 5900 nM
   TI
   LI
   LO
   TS