| Compound ID |
Compound Name |
Compound Formula |
|
CP0142382
|
[2-methyl-3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidin-7-yl]urea
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|
C21H23F3N6O2
|
2
|
| 1 |
EC50 = 12589.25 nM
|
|
|
| 2 |
EC50 > 31622.78 nM
|
|
|
|
CP0153348
|
2-methyl-3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidin-7-amine
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|
C20H22F3N5O
|
2
|
| 1 |
EC50 = 12589.25 nM
|
|
|
| 2 |
EC50 > 31622.78 nM
|
|
|
|
CP0142386
|
2-methyl-3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-morpholin-4-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C20H21F3N4O2
|
2
|
| 1 |
EC50 > 15848.93 nM
|
|
|
| 2 |
EC50 = 15848.93 nM
|
|
|
|
CP0153352
|
3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-morpholin-4-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C19H19F3N4O2
|
2
|
| 1 |
EC50 = 15848.93 nM
|
|
|
| 2 |
EC50 > 31622.78 nM
|
|
|
|
CP0085474
|
2-methyl-3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-(oxan-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C21H22F3N3O2
|
2
|
| 1 |
EC50 = 25118.86 nM
|
|
|
| 2 |
EC50 > 31622.78 nM
|
|
|
|
CP0067451
|
3-[(2,3-dichlorophenyl)methyl]-5-morpholin-4-yl-2-(trifluoromethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C18H15Cl2F3N4O2
|
1
|
| 1 |
EC50 > 31622.78 nM
|
|
|
|
CP0085471
|
2-methyl-3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-7-carboxylic acid
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|
C21H21F3N4O3
|
1
|
| 1 |
EC50 > 31622.78 nM
|
|
|
|
CP0142384
|
2-amino-3-[(2,3-dichlorophenyl)methyl]-5-(oxan-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C18H18Cl2N4O2
|
1
|
| 1 |
EC50 > 31622.78 nM
|
|
|
|
CP0153351
|
2-methyl-5-morpholin-4-yl-3-(naphthalen-1-ylmethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C22H22N4O2
|
2
|
| 1 |
EC50 > 31622.78 nM
|
|
|
| 2 |
EC50 = 31622.78 nM
|
|
|
|
CP0193724
|
3-[(2,3-dichlorophenyl)methyl]-2-ethyl-5-pyridin-4-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C20H16Cl2N4O
|
1
|
| 1 |
EC50 > 31622.78 nM
|
|
|
|
CP0207212
|
2-methyl-3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-7-carboxamide
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|
C21H22F3N5O2
|
1
|
| 1 |
EC50 > 31622.78 nM
|
|
|
|
CP0085472
|
3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-5-pyridin-4-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C20H15F3N4O
|
1
|
| 1 |
EC50 > 31622.78 nM
|
|
|
|
CP0153354
|
3-[(2,3-dichlorophenyl)methyl]-2-methoxy-5-pyridin-4-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
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|
C19H14Cl2N4O2
|
1
|
| 1 |
EC50 > 31622.78 nM
|
|
|
|
CP0093020
|
2-methyl-5-(2-methylmorpholin-4-yl)-3-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
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|
C20H22F3N5O2
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0077449
|
2-methyl-1-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-7-morpholin-4-ylimidazo[1,2-a]pyrimidin-5-one
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|
C20H21F3N4O2
|
1
|
| 1 |
IC50 > 29000 nM
|
|
|
