Brief Information of the Cell Line and Protein
Cell Line ID: CL000392 , Y1
Synonyms
Y-1
Y 1
Clone Y-1
Clone Y1
GM05384
Category Cancer cell line
Organism
Mus musculus (Mouse)
Cellosaurus ID
CVCL_0585
Protein ID: PT02992 , Adrenocorticotropic hormone receptor
Gene Name MC2R
Organism Mus musculus, Mouse
Protein Classification Membrane receptor
Uniprot ID Q64326
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000392  Protein ID: PT02992
 
Compound ID Compound Name Compound Formula
CP0045108
(4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S)-6-amino-1-[(2S)-2-{[(1S)-1-carbamoyl-2-methylpropyl]carbamoyl}pyrrolidin-1-yl]-1-oxohexan-2-yl]carbamoyl}methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoyl}-4-carbamimidamidobutyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(1H-imidazol-5-yl)ethyl]carbamoyl}-4-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-acetamido-3-hydroxypropanamido]-3-(4-hydroxyphenyl)propanamido]-3-hydroxypropanamido]-4-(methylsulfanyl)butanamido]butanoic acid
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C77H109N21O19S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0149367
(R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid [(R)-1-(4-chloro-benzyl)-2-(4-cyclohexyl-4-[1,2,4]triazol-1-ylmethyl-piperidin-1-yl)-2-oxo-ethyl]-amide
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C33H41ClN6O2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0269557
(R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(2-[1,2,4]triazol-1-ylmethyl-phenyl)-piperazin-1-yl]-ethyl}-amide
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C32H34ClN7O2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0393281
(R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid {(R)-1-(4-chloro-benzyl)-2-oxo-2-[4-(2-[1,2,4]triazol-4-ylmethyl-phenyl)-piperazin-1-yl]-ethyl}-amide
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C32H34ClN7O2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS