Brief Information of the Cell Line and Protein
Cell Line ID: CL000386 , Flp-In-CHO
Synonyms
Flp-In CHO
CHO Flp-In
CHO-Flp-In
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_U424
Protein ID: PT03121 , Free fatty acid receptor 4
Gene Name FFAR4
Organism Mus musculus, Mouse
Protein Classification Membrane receptor
Uniprot ID Q7TMA4
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000386  Protein ID: PT03121
 
Compound ID Compound Name Compound Formula
CP0408827
(1S,2S)-2-[4-[4-fluoro-3-methoxy-1-(4-methylphenyl)indazol-6-yl]phenyl]cyclopropane-1-carboxylic acid
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C25H21FN2O3
 1
1
EC50 = 17 nM
   TI
   LI
   LO
   TS
CP0109820
(1S,2S)-2-[4-(3-methoxy-1-pyridin-2-ylindazol-6-yl)phenyl]cyclopropane-1-carboxylic acid
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C23H19N3O3
 1
1
EC50 = 410 nM
   TI
   LI
   LO
   TS
CP0408828
(1S,2S)-2-[4-[3-methyl-1-(4-methylphenyl)indazol-6-yl]phenyl]cyclopropane-1-carboxylic acid
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C25H22N2O2
 1
1
EC50 = 510 nM
   TI
   LI
   LO
   TS
CP0430074
(1S,2S)-2-[4-[4-fluoro-3-methyl-1-(4-methylphenyl)indazol-6-yl]phenyl]cyclopropane-1-carboxylic acid
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C25H21FN2O2
 1
1
EC50 = 540 nM
   TI
   LI
   LO
   TS
CP0446633
(1S,2S)-2-[4-(4-fluoro-3-methoxy-1-pyridin-2-ylindazol-6-yl)phenyl]cyclopropane-1-carboxylic acid
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C23H18FN3O3
 1
1
EC50 = 620 nM
   TI
   LI
   LO
   TS
CP0408826
(1S,2S)-2-[4-[3-methyl-1-(4-methylphenyl)pyrazolo[4,3-c]pyridin-6-yl]phenyl]cyclopropane-1-carboxylic acid
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C24H21N3O2
 1
1
EC50 = 640 nM
   TI
   LI
   LO
   TS
CP0396394
(1S,2S)-2-[3-fluoro-4-[3-methyl-1-(5-methylpyridin-2-yl)pyrazolo[4,3-c]pyridin-6-yl]phenyl]cyclopropane-1-carboxylic acid
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C23H19FN4O2
 1
1
EC50 = 1000 nM
   TI
   LI
   LO
   TS