| Compound ID |
Compound Name |
Compound Formula |
|
CP0476603
|
N-(4-bromophenyl)-2-[5-[(2,3-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]hexanamide
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|
C26H30BrN3O4
|
2
|
| 1 |
EC50 = 6.457 nM
|
|
|
| 2 |
EC50 = 245.47 nM
|
|
|
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CP0259831
|
1-(4-chlorophenyl)-3-[1-methyl-3-oxo-2-phenyl-5-(propan-2-yl)-2,3-dihydro-1H-pyrazol-4-yl]urea
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|
C20H21ClN4O2
|
2
|
| 1 |
EC50 = 32.36 nM
|
|
|
| 2 |
EC50 = 51.29 nM
|
|
|
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CP0423004
|
N-(4-chlorophenyl)-2-[5-[(2,3-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]hexanamide
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|
C26H30ClN3O4
|
2
|
| 1 |
EC50 = 54.95 nM
|
|
|
| 2 |
EC50 = 93.33 nM
|
|
|
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CP0422998
|
N-(4-chlorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]hexanamide
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|
C25H28ClN3O3
|
2
|
| 1 |
EC50 = 125.89 nM
|
|
|
| 2 |
EC50 = 5248.07 nM
|
|
|
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CP0422991
|
N-(4-chlorophenyl)-2-[5-[(2,3-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
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|
C23H24ClN3O4
|
2
|
| 1 |
EC50 = 144.54 nM
|
|
|
| 2 |
EC50 = 154.88 nM
|
|
|
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CP0423003
|
N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]hexanamide
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|
C25H28BrN3O3
|
2
|
| 1 |
EC50 = 147.91 nM
|
|
|
| 2 |
EC50 = 11481.54 nM
|
|
|
|
CP0422996
|
N-(4-chlorophenyl)-2-[5-[(2,3-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C22H22ClN3O4
|
2
|
| 1 |
EC50 = 169.82 nM
|
|
|
| 2 |
EC50 = 223.87 nM
|
|
|
|
CP0518541
|
N-(4-bromophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]hexanamide
Show/Hide
|
C25H28BrN3O3
|
2
|
| 1 |
EC50 = 331.13 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0444595
|
N-(4-bromophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22BrN3O3
|
2
|
| 1 |
EC50 = 851.14 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0520509
|
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C21H20ClN3O3
|
2
|
| 1 |
EC50 = 1230.27 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0471757
|
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22ClN3O3
|
2
|
| 1 |
EC50 = 1380.38 nM
|
|
|
| 2 |
EC50 = 17378.01 nM
|
|
|
|
CP0473681
|
N-(4-bromophenyl)-2-[5-[(2-fluorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
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|
C21H19BrFN3O2
|
2
|
| 1 |
EC50 = 1778.28 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0459090
|
N-(4-bromophenyl)-2-[5-[(4-fluorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C21H19BrFN3O2
|
2
|
| 1 |
EC50 = 1819.7 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0519029
|
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]butanamide
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|
C23H24ClN3O3
|
2
|
| 1 |
EC50 = 1862.09 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0391343
|
N-(4-bromophenyl)-2-[5-[(3-fluorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
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|
C21H19BrFN3O2
|
2
|
| 1 |
EC50 = 2089.3 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0389680
|
N-(4-chlorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C21H20ClN3O3
|
2
|
| 1 |
EC50 = 2238.72 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0423001
|
N-(4-bromophenyl)-2-[5-[(4-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22BrN3O3
|
2
|
| 1 |
EC50 = 2630.27 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
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CP0518558
|
N-(4-chlorophenyl)-2-[5-[(2,6-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C22H22ClN3O4
|
2
|
| 1 |
EC50 = 2630.27 nM
|
|
|
| 2 |
EC50 = 2818.38 nM
|
|
|
|
CP0422993
|
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]-3-methylbutanamide
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|
C24H26ClN3O3
|
2
|
| 1 |
EC50 = 2818.38 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0476610
|
N-(4-chlorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22ClN3O3
|
2
|
| 1 |
EC50 = 3388.44 nM
|
|
|
| 2 |
EC50 = 25118.86 nM
|
|
|
|
CP0493747
|
N-(4-ethylphenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C23H25N3O3
|
2
|
| 1 |
EC50 = 5011.87 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0422995
|
N-(4-chloro-2-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H19ClFN3O3
|
2
|
| 1 |
EC50 = 5623.41 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0407523
|
N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H20BrN3O3
|
2
|
| 1 |
EC50 = 6025.6 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0459089
|
N-(4-chlorophenyl)-2-[5-[(2,5-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C22H22ClN3O4
|
2
|
| 1 |
EC50 = 6309.57 nM
|
|
|
| 2 |
EC50 = 10000 nM
|
|
|
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CP0422992
|
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]pentanamide
Show/Hide
|
C24H26ClN3O3
|
2
|
| 1 |
EC50 = 6309.57 nM
|
|
|
| 2 |
EC50 = 9772.37 nM
|
|
|
|
CP0391357
|
N-(3-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22FN3O3
|
2
|
| 1 |
EC50 = 7585.78 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0391339
|
N-(4-methoxyphenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C22H23N3O4
|
2
|
| 1 |
EC50 = 7943.28 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0476609
|
N-(4-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22FN3O3
|
2
|
| 1 |
EC50 = 8511.38 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0391344
|
N-(4-bromo-2-nitrophenyl)-2-[5-[(4-fluorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C20H16BrFN4O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0391354
|
N-(4-cyanophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C22H20N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0422994
|
2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]-N-[4-(trifluoromethoxy)phenyl]acetamide
Show/Hide
|
C22H20F3N3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0422997
|
N-(4-chlorophenyl)-2-cyclopropyl-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C24H24ClN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0422999
|
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-6-oxo-3-(trifluoromethyl)pyridazin-1-yl]acetamide
Show/Hide
|
C21H17ClF3N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0423000
|
N-(2-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22FN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0423005
|
N-(3-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H20ClN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0423006
|
N-(2-chlorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22ClN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0423008
|
N-(4-chloro-2,6-difluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H18ClF2N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
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CP0459087
|
N-(2,4-dichlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H19Cl2N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0459088
|
N-(3-chlorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
Show/Hide
|
C22H22ClN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0459092
|
N-(4-chloro-2,6-difluorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H18ClF2N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0459094
|
N-(2,4-difluoro-6-nitrophenyl)-2-[5-[(4-fluorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C20H15F3N4O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0473683
|
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-6-oxo-3-(trifluoromethyl)pyridazin-1-yl]hexanamide
Show/Hide
|
C25H25ClF3N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0476606
|
N-(4-chloro-2-fluorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H19ClFN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0489685
|
N-(3-cyanophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C22H20N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0519030
|
N-(2-cyanophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C22H20N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
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CP0552490
|
N-(2-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C21H20ClN3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
