Brief Information of the Cell Line and Protein
Cell Line ID: CL000386 , Flp-In-CHO
Synonyms
Flp-In CHO
CHO Flp-In
CHO-Flp-In
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_U424
Protein ID: PT01179 , Beta-1 adrenergic receptor
Gene Name ADRB1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P08588
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000386  Protein ID: PT01179
 
Compound ID Compound Name Compound Formula
CP0137322
1H-indol-2-yl-[4-[2-(4-methoxyphenoxy)ethyl]piperazin-1-yl]methanone
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C22H25N3O3
 1
1
Ki = 77 nM
   TI
   LI
   LO
   TS
CP0391154
(3aS,9bS)-7,9-dimethoxy-3a-methyl-2,3,4,9b-tetrahydro-1H-chromeno[3,4-b]pyrrole
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C14H19NO3
 1
1
Ki = 1000 nM
   TI
   LI
   LO
   TS
CP0066194
N-[2-(1,3-benzodioxol-5-yl)ethyl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenylpropan-1-amine
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C28H33NO4
 1
1
Ki = 1885 nM
   TI
   LI
   LO
   TS
CP0248166
benzyl 5-[4-(2-methylprop-2-enyl)piperazin-1-yl]-1,3-dihydroisoindole-2-carboxylate
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C24H29N3O2
 1
1
Ki = 1894 nM
   TI
   LI
   LO
   TS
CP0387083
(3aS,9bS)-3a-methyl-5-phenyl-2,3,4,9b-tetrahydro-1H-pyrrolo[2,3-c]quinoline
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C18H20N2
 1
1
Ki = 3162.28 nM
   TI
   LI
   LO
   TS
CP0064183
4-[3-methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy]furo[3,2-c]pyridine
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C21H16N4O2
 1
1
Ki = 7600 nM
   TI
   LI
   LO
   TS
CP0244206
7-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]thieno[2,3-c]pyridine
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C21H12F3N3OS
 1
1
Ki = 8500 nM
   TI
   LI
   LO
   TS
CP0369306
4-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
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C21H12F3N3O2
 1
1
Ki = 8500 nM
   TI
   LI
   LO
   TS
CP0064188
4-[4-(6-methylimidazo[1,2-a]pyrazin-5-yl)-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
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C21H13F3N4O2
 1
1
Ki = 9600 nM
   TI
   LI
   LO
   TS
CP0002071
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N-prop-2-enylprop-2-en-1-amine
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C17H22N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0391120
(1S,2R)-1-ethyl-7-methoxy-2-methyl-3,4-dihydro-1H-naphthalen-2-amine
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C14H21NO
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0391121
(3S,4S)-4-ethyl-3,6-dimethyl-2,4-dihydrochromen-3-amine
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C13H19NO
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0411059
(3S,4S)-4-ethyl-3-methyl-1-phenyl-2,4-dihydroquinolin-3-amine
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C18H22N2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS