| Compound ID |
Compound Name |
Compound Formula |
|
CP0151699
|
(S)-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4H,4aH,5H,6H,7H,8H-cyclohexa[f]indazol-5-yl](1-benzothiophen-3-yl)methanol
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|
C27H25FN2OS
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0047174
|
(1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-hydroxyacetyl)-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-3,6-dien-5-one
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|
C21H28O5
|
1
|
| 1 |
EC50 = 3.4 nM
|
|
|
|
CP0424208
|
(S)-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4H,4aH,5H,6H,7H-cyclopenta[f]indazol-5-yl](1-benzothiophen-3-yl)methanol
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|
C26H23FN2OS
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0424336
|
(R)-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4H,4aH,5H,6H,7H-cyclopenta[f]indazol-5-yl](1-benzofuran-3-yl)methanol
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|
C26H23FN2O2
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
|
CP0434459
|
(R)-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4H,4aH,5H,6H,7H-cyclopenta[f]indazol-5-yl](naphthalen-1-yl)methanol
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|
C28H25FN2O
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0461955
|
(S)-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4H,4aH,5H,6H,7H-cyclopenta[f]indazol-5-yl](1-benzofuran-3-yl)methanol
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|
C26H23FN2O2
|
1
|
| 1 |
EC50 = 92 nM
|
|
|
|
CP0464253
|
(S)-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4H,4aH,5H,6H,7H-cyclopenta[f]indazol-5-yl](naphthalen-1-yl)methanol
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|
C28H25FN2O
|
1
|
| 1 |
EC50 = 94 nM
|
|
|
|
CP0059549
|
(R)-[(4aR,5S)-1-(4-fluorophenyl)-4a-methyl-1H,4H,4aH,5H,6H,7H,8H-cyclohexa[f]indazol-5-yl](1-benzothiophen-2-yl)methanol
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|
C27H25FN2OS
|
1
|
| 1 |
EC50 = 1209 nM
|
|
|