| Compound ID |
Compound Name |
Compound Formula |
|
CP0211420
|
1-[[3-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]-7-methylpurin-6-one
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|
C17H15ClN6O2
|
5
|
| 1 |
EC50 > 40000 nM
|
|
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| 2 |
IC50 = 10 nM
|
|
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| 3 |
IC50 = 19 nM
|
|
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| 4 |
IC50 = 20 nM
|
|
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| 5 |
IC50 = 71 nM
|
|
|
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CP0391125
|
3-[[5-[(E)-2-(4-chlorophenyl)prop-1-enyl]-1,2,4-oxadiazol-3-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
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|
C19H14ClN5O2
|
3
|
| 1 |
EC50 > 40000 nM
|
|
|
| 2 |
IC50 = 53 nM
|
|
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| 3 |
IC50 = 105 nM
|
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|
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CP0391126
|
1-[[3-[(E)-2-(4-chlorophenyl)prop-1-enyl]-1,2,4-oxadiazol-5-yl]methyl]-7-methylpurin-6-one
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|
C18H15ClN6O2
|
3
|
| 1 |
EC50 > 40000 nM
|
|
|
| 2 |
IC50 = 55 nM
|
|
|
| 3 |
IC50 = 75 nM
|
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|
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CP0392459
|
3-[[3-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
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|
C18H14ClN5O2
|
3
|
| 1 |
EC50 > 40000 nM
|
|
|
| 2 |
IC50 = 21 nM
|
|
|
| 3 |
IC50 = 120 nM
|
|
|
|
CP0392463
|
3-[[3-[2-(4-chlorophenyl)-2-hydroxyethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
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|
C18H14ClN5O3
|
3
|
| 1 |
EC50 > 40000 nM
|
|
|
| 2 |
IC50 = 75 nM
|
|
|
| 3 |
IC50 = 204 nM
|
|
|
|
CP0425054
|
3-[[5-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-3-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
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|
C18H14ClN5O2
|
3
|
| 1 |
EC50 > 40000 nM
|
|
|
| 2 |
IC50 = 89 nM
|
|
|
| 3 |
IC50 = 411 nM
|
|
|
|
CP0385690
|
N-[2-[4-(difluoromethoxy)phenyl]ethyl]-2-(8-methyl-4-oxoquinazolin-3-yl)acetamide
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|
C20H19F2N3O3
|
4
|
| 1 |
EC50 > 47000 nM
|
|
|
| 2 |
IC50 = 142 nM
|
|
|
| 3 |
IC50 = 2620 nM
|
|
|
| 4 |
IC50 > 25000 nM
|
|
|
|
CP0392455
|
6-[[3-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]-1-methylpyrazolo[4,3-d]pyrimidin-7-one
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|
C17H15ClN6O2
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0509261
|
3-[[3-[2-(4-chlorophenyl)-2-fluoroethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
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|
C18H13ClFN5O2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0404298
|
3-[[3-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]-5-methylpyrido[2,3-d]pyrimidin-4-one
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|
C19H16ClN5O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0462431
|
N-[2-(4-chlorophenyl)ethyl]-2-(8-cyano-4-oxoquinazolin-3-yl)acetamide
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|
C19H15ClN4O2
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0395902
|
6-methyl-5-[2-(trifluoromethyl)phenyl]-1H-indazole
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|
C15H11F3N2
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0447265
|
6-methoxy-5-[2-(trifluoromethyl)phenyl]-1H-indazole
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|
C15H11F3N2O
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0469481
|
3-[[5-[2-(4-chlorophenyl)propyl]-1,2,4-oxadiazol-3-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
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|
C19H16ClN5O2
|
1
|
| 1 |
IC50 = 105 nM
|
|
|
|
CP0425043
|
N-[2-(4-chlorophenyl)ethyl]-2-(5-methyl-4-oxoquinazolin-3-yl)acetamide
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|
C19H18ClN3O2
|
1
|
| 1 |
IC50 = 112 nM
|
|
|
|
CP0469584
|
3-[[3-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrimido[4,5-d]pyrimidin-4-one
Show/Hide
|
C17H13ClN6O2
|
1
|
| 1 |
IC50 = 113 nM
|
|
|
|
CP0472931
|
1-[[5-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-3-yl]methyl]-7-methylpurin-6-one
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|
C17H15ClN6O2
|
1
|
| 1 |
IC50 = 136 nM
|
|
|
|
CP0440771
|
6-chloro-5-[2-(trifluoromethyl)phenyl]-1H-indazole
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|
C14H8ClF3N2
|
1
|
| 1 |
IC50 = 169 nM
|
|
|
|
CP0401633
|
6-[[3-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrimido[4,5-c]pyridazin-5-one
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|
C17H13ClN6O2
|
1
|
| 1 |
IC50 = 176 nM
|
|
|
|
CP0447248
|
6-(cyclopropylmethoxy)-5-[2-(trifluoromethyl)phenyl]-1H-indazole
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|
C18H15F3N2O
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0401643
|
1-[[5-[(E)-2-(4-chlorophenyl)prop-1-enyl]-1,2,4-oxadiazol-3-yl]methyl]-7-methylpurin-6-one
Show/Hide
|
C18H15ClN6O2
|
1
|
| 1 |
IC50 = 274 nM
|
|
|
|
CP0401632
|
N-[2-(4-chlorophenyl)ethyl]-2-(6-methyl-4-oxoquinazolin-3-yl)acetamide
Show/Hide
|
C19H18ClN3O2
|
1
|
| 1 |
IC50 = 287 nM
|
|
|
|
CP0392454
|
N-[2-(4-chlorophenyl)ethyl]-2-[4-oxo-8-(trifluoromethyl)quinazolin-3-yl]acetamide
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|
C19H15ClF3N3O2
|
1
|
| 1 |
IC50 = 306 nM
|
|
|
|
CP0425044
|
3-[[3-[2-(4-chlorophenyl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]pteridin-4-one
Show/Hide
|
C17H13ClN6O2
|
1
|
| 1 |
IC50 = 314 nM
|
|
|
|
CP0487896
|
N-[2-(4-chlorophenyl)ethyl]-2-(8-methyl-4-oxoquinazolin-3-yl)acetamide
Show/Hide
|
C19H18ClN3O2
|
1
|
| 1 |
IC50 = 358 nM
|
|
|
|
CP0440768
|
5-[2-(trifluoromethyl)phenyl]-1H-indazole
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|
C14H9F3N2
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0395903
|
6-(trifluoromethoxy)-5-[2-(trifluoromethyl)phenyl]-1H-indazole
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|
C15H8F6N2O
|
1
|
| 1 |
IC50 = 627 nM
|
|
|
|
CP0472932
|
3-[[5-[(E)-2-(4-chlorophenyl)ethenyl]-1,2,4-oxadiazol-3-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
Show/Hide
|
C18H12ClN5O2
|
1
|
| 1 |
IC50 = 652 nM
|
|
|
|
CP0498112
|
N-[2-(4-chlorophenyl)ethyl]-2-(8-fluoro-4-oxoquinazolin-3-yl)acetamide
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|
C18H15ClFN3O2
|
1
|
| 1 |
IC50 = 791 nM
|
|
|
|
CP0404296
|
N-[2-(4-chlorophenyl)ethyl]-2-(4-oxopyrido[3,4-d]pyrimidin-3-yl)acetamide
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|
C17H15ClN4O2
|
1
|
| 1 |
IC50 = 1080 nM
|
|
|
|
CP0462428
|
N-[2-(4-chlorophenyl)ethyl]-2-(4-oxopyrido[2,3-d]pyrimidin-3-yl)acetamide
Show/Hide
|
C17H15ClN4O2
|
1
|
| 1 |
IC50 = 1170 nM
|
|
|
|
CP0401621
|
N-[2-(4-methoxyphenyl)ethyl]-2-(8-methyl-4-oxoquinazolin-3-yl)acetamide
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|
C20H21N3O3
|
1
|
| 1 |
IC50 = 1370 nM
|
|
|
|
CP0467962
|
3-[[3-[2-(6-chloropyridin-3-yl)ethyl]-1,2,4-oxadiazol-5-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
Show/Hide
|
C17H13ClN6O2
|
1
|
| 1 |
IC50 = 1380 nM
|
|
|
|
CP0404297
|
3-[[5-[2-(4-chlorophenyl)ethyl]-1,3,4-oxadiazol-2-yl]methyl]pyrido[2,3-d]pyrimidin-4-one
Show/Hide
|
C18H14ClN5O2
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0499832
|
N-[2-(4-chlorophenyl)ethyl]-2-(8-methoxy-4-oxoquinazolin-3-yl)acetamide
Show/Hide
|
C19H18ClN3O3
|
1
|
| 1 |
IC50 = 2150 nM
|
|
|
|
CP0401638
|
N-[2-(3-methoxyphenyl)ethyl]-2-(8-methyl-4-oxoquinazolin-3-yl)acetamide
Show/Hide
|
C20H21N3O3
|
1
|
| 1 |
IC50 > 16700 nM
|
|
|
|
CP0401640
|
N-[2-(2-methoxyphenyl)ethyl]-2-(8-methyl-4-oxoquinazolin-3-yl)acetamide
Show/Hide
|
C20H21N3O3
|
1
|
| 1 |
IC50 > 16700 nM
|
|
|
|
CP0401641
|
N-[2-(4-chlorophenyl)ethyl]-2-(7-methyl-4-oxoquinazolin-3-yl)acetamide
Show/Hide
|
C19H18ClN3O2
|
1
|
| 1 |
IC50 > 16700 nM
|
|
|
