Compound ID |
Compound Name |
Compound Formula |
CP0013607
|
2-methoxyacetic acid [(1S,2S)-2-[2-[3-(1H-benzimidazol-2-yl)propyl-methyl-amino]ethyl]-6-fluoro-1-isopropyl-tetralin-2-yl] ester;hydrate;hydrochloride
Show/Hide
|
C29H38FN3O3
|
1
|
1 |
IC50 = 1100 nM
|
|
|
CP0923188
|
2-[1-[2-[4-fluoro-2-(2-methoxyethoxy)phenyl]ethyl]piperidin-4-yl]-N-[(1R)-1-(4-fluorophenyl)-2-methylpropyl]acetamide
Show/Hide
|
C28H38F2N2O3
|
1
|
1 |
IC50 = 1900 nM
|
|
|
CP0873392
|
2-[1-[2-[3-fluoro-2-(2-methoxyethoxy)phenyl]ethyl]piperidin-4-yl]-N-[(1R)-1-(4-fluorophenyl)-2-methylpropyl]acetamide
Show/Hide
|
C28H38F2N2O3
|
1
|
1 |
IC50 = 2100 nM
|
|
|
CP0873393
|
2-[1-[2-[5-fluoro-2-(2-methoxyethoxy)phenyl]ethyl]piperidin-4-yl]-N-[(1R)-1-(4-fluorophenyl)-2-methylpropyl]acetamide
Show/Hide
|
C28H38F2N2O3
|
1
|
1 |
IC50 = 3100 nM
|
|
|
CP0941579
|
2-[1-[2-[2-fluoro-6-(2-methoxyethoxy)phenyl]ethyl]piperidin-4-yl]-N-[(1R)-1-(4-fluorophenyl)-2-methylpropyl]acetamide
Show/Hide
|
C28H38F2N2O3
|
1
|
1 |
IC50 = 3100 nM
|
|
|
CP0926518
|
N-[2-(4-fluorophenyl)-3-methylbutyl]-1-(2-phenylethyl)piperidine-4-carboxamide
Show/Hide
|
C25H33FN2O
|
1
|
1 |
IC50 = 3900 nM
|
|
|
CP0468566
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-(2-phenylethyl)piperidine-4-carboxamide
Show/Hide
|
C26H35FN2O
|
1
|
1 |
IC50 = 4400 nM
|
|
|
CP0865043
|
1-[(1R)-1-(4-fluorophenyl)-2-methylpropyl]-3-[1-(2-phenylethyl)piperidin-4-yl]urea
Show/Hide
|
C24H32FN3O
|
1
|
1 |
IC50 = 5000 nM
|
|
|
CP0952239
|
N-[(1R)-1-(4-fluorophenyl)-2-methylpropyl]-2-[1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl]acetamide
Show/Hide
|
C26H35FN2O2
|
1
|
1 |
IC50 = 6800 nM
|
|
|
CP0900988
|
N-[(1R)-1-(4-fluorophenyl)-2-methylpropyl]-2-[1-(2-phenylethyl)piperidin-4-yl]acetamide
Show/Hide
|
C25H33FN2O
|
1
|
1 |
IC50 = 10000 nM
|
|
|