Brief Information of the Cell Line and Protein
Cell Line ID: CL000218 , BT-474
Synonyms
Bt-474
BT474
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0179
Protein ID: PT03525 , Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Gene Name PIK3CA
Organism Mus musculus, Mouse
Protein Classification Enzyme
Uniprot ID P42337
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000218  Protein ID: PT03525
 
Compound ID Compound Name Compound Formula
CP0561456
US9156831, 10
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C22H31N9O4
 1
1
IC50 = 85 nM
   TI
   LI
   LO
   TS
CP0143273
US9156831, 3
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C22H31N9O3
 1
1
IC50 = 90 nM
   TI
   LI
   LO
   TS
CP0503594
US9156831, 11
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C22H31N9O4
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0117467
US9156831, 9
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C22H29N9O4
 1
1
IC50 = 330 nM
   TI
   LI
   LO
   TS
CP0093702
US9156831, 1
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C21H29N9O3
 1
1
IC50 = 360 nM
   TI
   LI
   LO
   TS
CP0093703
US9156831, 7
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C22H31N9O3
 1
1
IC50 = 420 nM
   TI
   LI
   LO
   TS
CP0173540
US9156831, 6
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C22H31N9O3
 1
1
IC50 = 530 nM
   TI
   LI
   LO
   TS
CP0283502
US9156831, 8
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C21H27N9O4
 1
1
IC50 = 590 nM
   TI
   LI
   LO
   TS