Compound ID |
Compound Name |
Compound Formula |
CP0190970
|
N-[(2S)-3-(1-methylcyclohexyl)-1-[[(4S,7R)-7-methyl-3-oxo-1-pyridin-2-ylsulfonylazepan-4-yl]amino]-1-oxopropan-2-yl]morpholine-4-carboxamide
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|
C27H41N5O6S
|
1
|
1 |
IC50 = 570 nM
|
|
|
CP0060769
|
5-(2-MORPHOLIN-4-YLETHOXY)BENZOFURAN-2-CARBOXYLIC ACID ((S)-3-METHYL-1-{(S)-3-OXO-1-[2-(3-PYRIDIN-2-YLPHENYL)ACETYL]AZEPAN-4-YLCARBAMOYL}BUTYL)AMIDE
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|
C40H47N5O7
|
1
|
1 |
IC50 = 940 nM
|
|
|
CP0197279
|
N-[(2S)-3-(1-methylcyclohexyl)-1-[[(4S,7R)-7-methyl-3-oxo-1-pyridin-2-ylsulfonylazepan-4-yl]amino]-1-oxopropan-2-yl]furan-2-carboxamide
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|
C27H36N4O6S
|
1
|
1 |
IC50 = 1400 nM
|
|
|
CP0197278
|
N-[(2S)-3-cyclohexyl-1-[[(4S,7R)-7-methyl-3-oxo-1-pyridin-2-ylsulfonylazepan-4-yl]amino]-1-oxopropan-2-yl]furan-2-carboxamide
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|
C26H34N4O6S
|
1
|
1 |
IC50 = 1780 nM
|
|
|
CP0281337
|
N-[(2S)-3-(1-methylcyclohexyl)-1-[[(4S,7R)-7-methyl-3-oxo-1-(pyridine-2-carbonyl)azepan-4-yl]amino]-1-oxopropan-2-yl]furan-2-carboxamide
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|
C28H36N4O5
|
1
|
1 |
IC50 = 3880 nM
|
|
|
CP0233764
|
N-[(2S)-4,4-dimethyl-1-[[(4S,7R)-7-methyl-3-oxo-1-pyridin-2-ylsulfonylazepan-4-yl]amino]-1-oxopentan-2-yl]furan-2-carboxamide
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|
C24H32N4O6S
|
1
|
1 |
IC50 = 4800 nM
|
|
|