| Compound ID |
Compound Name |
Compound Formula |
|
CP0426232
|
N-[(2S)-1-[[(2S)-3-(1H-indol-3-yl)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-3-methyl-1H-indene-2-carboxamide
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|
C37H38N4O5
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0086566
|
(2S)-2-[[2-(azepan-1-yl)acetyl]amino]-4-methyl-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pentanamide
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|
C35H48N4O5
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0213895
|
Kzr-616
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|
C30H42N4O8
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0062987
|
(2S)-3-(4-methoxyphenyl)-N-[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
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|
C31H40N4O7
|
1
|
| 1 |
IC50 = 98 nM
|
|
|
|
CP0151829
|
(2S)-N-[(2S)-3-(cyclopenten-1-yl)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
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|
C30H42N4O7
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0421117
|
N-[(2R)-1-[[(2S)-3-(4-methoxyphenyl)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]cyclohexanecarboxamide
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|
C32H41N3O6
|
1
|
| 1 |
IC50 = 141 nM
|
|
|
|
CP0403175
|
CHEMBL4454809
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|
C32H41N3O7
|
1
|
| 1 |
IC50 = 262 nM
|
|
|
|
CP0086565
|
CHEMBL4441524
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|
C31H43N3O7
|
1
|
| 1 |
IC50 = 374 nM
|
|
|
|
CP0477259
|
N-[(2R)-1-[[(2S)-1-[[(2S)-3-cyclobutyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-3-(4-methoxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-4-hydroxycyclohexane-1-carboxamide
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|
C30H43N3O7
|
1
|
| 1 |
IC50 = 556 nM
|
|
|
|
CP0847941
|
N-((R)-1-((S)-3-(1H-indol-3-yl)-1-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C37H38N4O5
|
1
|
| 1 |
IC50 = 573 nM
|
|
|
|
CP0859992
|
N-((R)-1-((S)-3-(4-methoxyphenyl)-1-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C36H39N3O6
|
1
|
| 1 |
IC50 = 764 nM
|
|
|
|
CP0098995
|
(2S)-2-[[2-(azepan-1-yl)acetyl]amino]-4-methyl-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-4-(4-methylphenyl)-1-oxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pentanamide
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|
C37H52N4O5
|
1
|
| 1 |
IC50 = 1920 nM
|
|
|
