| Compound ID |
Compound Name |
Compound Formula |
|
CP0056256
|
(3S)-1-[(1S,2R,4R)-4-[methyl(propan-2-yl)amino]-2-propylcyclohexyl]-3-[[6-(trifluoromethyl)quinazolin-4-yl]amino]pyrrolidin-2-one
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|
C26H36F3N5O
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0123082
|
(3S)-1-[(1S,2R,4R)-2-ethyl-4-[methyl(propan-2-yl)amino]cyclohexyl]-3-[[6-(trifluoromethyl)quinazolin-4-yl]amino]pyrrolidin-2-one
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|
C25H34F3N5O
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0095074
|
2-(ethylcarbamoylamino)-N-[(3S)-1-[(1S,2R,4R)-4-[methyl(propan-2-yl)amino]-2-propylcyclohexyl]-2-oxopyrrolidin-3-yl]-5-(trifluoromethyl)benzamide
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|
C28H42F3N5O3
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0363491
|
(3S)-1-[(1S,2S,4R)-4-[methyl(propan-2-yl)amino]-2-propan-2-ylcyclohexyl]-3-[[6-(trifluoromethyl)quinazolin-4-yl]amino]pyrrolidin-2-one
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|
C26H36F3N5O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0133134
|
(3S)-1-[(1S,2R,4R)-2-(methoxymethyl)-4-[methyl(propan-2-yl)amino]cyclohexyl]-3-[[6-(trifluoromethyl)quinazolin-4-yl]amino]pyrrolidin-2-one
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|
C25H34F3N5O2
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0123078
|
(3S)-3-[(6-chloroquinazolin-4-yl)amino]-1-[(1S,2R,4R)-4-[methyl(propan-2-yl)amino]-2-propylcyclohexyl]pyrrolidin-2-one
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|
C25H36ClN5O
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0123080
|
N-[2-[[(2S,3S)-3-hydroxy-1-(2-methylpropylamino)hexan-2-yl]amino]-2-oxoethyl]-2-(propan-2-ylcarbamoylamino)-5-(trifluoromethyl)benzamide
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|
C24H38F3N5O4
|
1
|
| 1 |
IC50 = 137 nM
|
|
|
|
CP0169732
|
(3S)-1-[(1S,2R,4R)-4-[methyl(propan-2-yl)amino]-2-(methylsulfonylmethyl)cyclohexyl]-3-[[6-(trifluoromethyl)quinazolin-4-yl]amino]pyrrolidin-2-one
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|
C25H34F3N5O3S
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0177648
|
N-[(1R,2S,5R)-5-[methyl(propan-2-yl)amino]-2-[(3S)-2-oxo-3-[[6-(trifluoromethyl)quinazolin-4-yl]amino]pyrrolidin-1-yl]cyclohexyl]methanesulfonamide
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|
C24H33F3N6O3S
|
1
|
| 1 |
IC50 = 287 nM
|
|
|
|
CP0066059
|
N-[2-[[(2S,3S)-1-(2,2-dimethylpropylamino)-3-hydroxyhexan-2-yl]amino]-2-oxoethyl]-2-(propan-2-ylcarbamoylamino)-5-(trifluoromethyl)benzamide
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|
C25H40F3N5O4
|
1
|
| 1 |
IC50 = 321 nM
|
|
|
|
CP0154997
|
N-[(1R,2S,5R)-5-[methyl(propan-2-yl)amino]-2-[(3S)-2-oxo-3-[[6-(trifluoromethyl)quinazolin-4-yl]amino]pyrrolidin-1-yl]cyclohexyl]acetamide
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|
C25H33F3N6O2
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0098462
|
N-[2-[[(2S,3S)-1-(cyclopropylmethylamino)-3-hydroxyhexan-2-yl]amino]-2-oxoethyl]-2-(propan-2-ylcarbamoylamino)-5-(trifluoromethyl)benzamide
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|
C24H36F3N5O4
|
1
|
| 1 |
IC50 = 1242 nM
|
|
|
|
CP0364171
|
N-[(3S)-1-[(1S,2R,4R)-2-[methyl(methylsulfonyl)amino]-4-[methyl(propan-2-yl)amino]cyclohexyl]-2-oxopyrrolidin-3-yl]-3-(trifluoromethyl)benzamide
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|
C24H35F3N4O4S
|
1
|
| 1 |
IC50 = 1570 nM
|
|
|
|
CP0059670
|
N-[(3S)-1-[(1S,2R,4R)-4-[methyl(propan-2-yl)amino]-2-(methylsulfonylmethyl)cyclohexyl]-2-oxopyrrolidin-3-yl]-3-(trifluoromethyl)benzamide
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|
C24H34F3N3O4S
|
1
|
| 1 |
IC50 = 1636 nM
|
|
|
|
CP0365951
|
N-[(3S)-1-[(1S,2R,4R)-2-(methanesulfonamido)-4-[methyl(propan-2-yl)amino]cyclohexyl]-2-oxopyrrolidin-3-yl]-3-(trifluoromethyl)benzamide
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|
C23H33F3N4O4S
|
1
|
| 1 |
IC50 = 3469 nM
|
|
|
|
CP0087964
|
N-[(2R)-1-[4-(4-chlorophenyl)piperidin-1-yl]-3-methyl-1-oxobutan-2-yl]benzamide
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|
C23H27ClN2O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
