| Compound ID |
Compound Name |
Compound Formula |
|
CP0084819
|
(R)-5-Propylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one
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|
C13H17N3O
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0036921
|
3-HYDROXYTYRAMINE HYDROCHLORIDE
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|
C8H11NO2
|
3
|
| 1 |
EC50 = 7.7 nM
|
|
|
| 2 |
EC50 = 65 nM
|
|
|
| 3 |
Ki = 422 nM
|
|
|
|
CP0006107
|
CAS_85760-74-3
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|
C13H21N3
|
3
|
| 1 |
EC50 = 8.2 nM
|
|
|
| 2 |
EC50 = 19 nM
|
|
|
| 3 |
Ki = 1185 nM
|
|
|
|
CP0401191
|
(10R)-3-propyl-10-(propylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
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|
C16H23N3O
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0393847
|
(10R)-10-(dipropylamino)-3-propyl-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
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|
C19H29N3O
|
1
|
| 1 |
EC50 = 13.7 nM
|
|
|
|
CP0409654
|
(10R)-10-[methyl(propyl)amino]-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
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|
C14H19N3O
|
1
|
| 1 |
EC50 = 18.1 nM
|
|
|
|
CP0398933
|
N-[4-[methyl-[(10R)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]amino]butyl]-1-benzofuran-2-carboxamide
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|
C24H26N4O3
|
1
|
| 1 |
EC50 = 19.5 nM
|
|
|
|
CP0240206
|
N-[4-[methyl-[(10R)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]amino]butyl]-1H-indole-2-carboxamide
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|
C24H27N5O2
|
1
|
| 1 |
EC50 = 27.7 nM
|
|
|
|
CP0381243
|
3-[2-(Phenethyl-propyl-amino)-ethyl]-phenol; hydrobromide
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|
C19H25NO
|
2
|
| 1 |
EC50 = 39 nM
|
|
|
| 2 |
Ki = 64.4 nM
|
|
|
|
CP0178363
|
(R)-5-Methylamino-5,6-dihydro-1H,4H-imidazo[4,5,1-ij]quinolin-2-one
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|
C11H13N3O
|
1
|
| 1 |
EC50 = 64.7 nM
|
|
|
|
CP0398936
|
(10R)-3-butyl-10-(methylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
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|
C15H21N3O
|
1
|
| 1 |
EC50 = 83 nM
|
|
|
|
CP0455926
|
N-[4-[methyl-[(10R)-2-oxo-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-10-yl]amino]butyl]-9H-fluorene-2-carboxamide
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|
C29H30N4O2
|
1
|
| 1 |
EC50 = 102 nM
|
|
|
|
CP0190768
|
3-[2-[cyclopropylmethyl(2-phenylethyl)amino]ethyl]phenol
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|
C20H25NO
|
2
|
| 1 |
EC50 = 181 nM
|
|
|
| 2 |
Ki = 118 nM
|
|
|
|
CP0398934
|
(10R)-10-(methylamino)-3-propyl-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
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|
C14H19N3O
|
1
|
| 1 |
EC50 = 549 nM
|
|
|
|
CP0401190
|
(10R)-10-amino-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one
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|
C10H11N3O
|
1
|
| 1 |
EC50 = 684 nM
|
|
|
|
CP0354873
|
3-[2-[cyclobutylmethyl(2-phenylethyl)amino]ethyl]phenol
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|
C21H27NO
|
3
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 1647 nM
|
|
|
| 3 |
Ki = 450 nM
|
|
|
|
CP0381244
|
3-[2-[hexyl(2-phenylethyl)amino]ethyl]phenol
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|
C22H31NO
|
3
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 1252 nM
|
|
|
| 3 |
Ki = 831 nM
|
|
|
|
CP0042262
|
N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sulfamoylbenzamide
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|
C15H23N3O4S
|
1
|
| 1 |
IC50 = 10.28 nM
|
|
|
|
CP0294038
|
N-[3-fluoro-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1-benzothiophene-2-carboxamide
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|
C24H28FN3O2S
|
1
|
| 1 |
IC50 = 421 nM
|
|
|
|
CP0273713
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]-3-fluorobutyl]-5-methoxy-1-benzofuran-2-carboxamide
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|
C24H26Cl2FN3O3
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0381245
|
3-[2-[butyl(2-phenylethyl)amino]ethyl]phenol
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|
C20H27NO
|
1
|
| 1 |
Ki = 1233 nM
|
|
|
|
CP0396539
|
3-[2-[pentyl(2-phenylethyl)amino]ethyl]phenol
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|
C21H29NO
|
1
|
| 1 |
Ki = 1420 nM
|
|
|
