| Compound ID |
Compound Name |
Compound Formula |
|
CP0414627
|
6,9-difluoro-8-methyl-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
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|
C14H10F2O2S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0549216
|
4,5-dihydrobenzo[g][1]benzothiole-2-carboxamide
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|
C13H11NOS
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0512395
|
2-[7-cyclopropyl-6-(trifluoromethyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylacetic acid
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|
C12H9F3N2O2S2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0406186
|
6-chloro-8-fluoro-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
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|
C13H8ClFO2S
|
2
|
| 1 |
EC50 = 12 nM
|
|
|
| 2 |
EC50 = 25 nM
|
|
|
|
CP0407494
|
4,5-dihydrothieno[3,2-d][1]benzoxepine-2-carboxamide
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|
C13H11NO2S
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0534345
|
5,5-dimethyl-4H-benzo[g][1]benzothiole-2-carboxamide
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|
C15H15NOS
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0495741
|
5-methyl-4,5-dihydrobenzo[g][1]benzothiole-2-carboxamide
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|
C14H13NOS
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0406188
|
3-thiatricyclo[8.4.0.02,6]tetradeca-1(14),2(6),4,10,12-pentaene-4-carboxamide
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|
C14H13NOS
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0511152
|
6,8-difluoro-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
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|
C12H6F2O2S2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0511153
|
6,7,8-trifluoro-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
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|
C12H5F3O2S2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0401678
|
6,7-dichloro-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
Show/Hide
|
C13H8Cl2O2S
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0344327
|
2-(6-chloro-7-cyclopropylthieno[3,2-d]pyrimidin-4-yl)sulfanylacetic acid
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|
C11H9ClN2O2S2
|
2
|
| 1 |
EC50 = 21 nM
|
|
|
| 2 |
EC50 = 23 nM
|
|
|
|
CP0420081
|
6-fluoro-8-methyl-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
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|
C14H11FO2S
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0511169
|
6-chloro-7-methoxy-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
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|
C14H11ClO3S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0462761
|
6,8-dichloro-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
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|
C13H8Cl2O2S
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0414628
|
6-fluoro-8-methyl-4H-thieno[3,2-c]chromene-2-carboxylic acid
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|
C13H9FO3S
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0511151
|
6-chloro-8-fluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
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|
C12H6ClFO3S
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0534346
|
6-chloro-8-methyl-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
Show/Hide
|
C14H11ClO2S
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0472651
|
4-methyl-4,5-dihydrobenzo[g][1]benzothiole-2-carboxamide
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|
C14H13NOS
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0420082
|
6,7-dichloro-4H-thieno[3,2-c]chromene-2-carboxylic acid
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|
C12H6Cl2O3S
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
|
CP0459964
|
7-chloro-8-fluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
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|
C12H6ClFO3S
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0511165
|
8-chloro-6-fluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
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|
C12H6ClFO3S
|
1
|
| 1 |
EC50 = 59 nM
|
|
|
|
CP0462760
|
6,7-difluoro-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
Show/Hide
|
C13H8F2O2S
|
1
|
| 1 |
EC50 = 61 nM
|
|
|
|
CP0406187
|
6-cyano-7-methyl-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
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|
C15H11NO2S
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0414629
|
7,8,9-trifluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
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|
C12H5F3O3S
|
1
|
| 1 |
EC50 = 67 nM
|
|
|
|
CP0468104
|
6-cyano-7-fluoro-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
Show/Hide
|
C14H8FNO2S
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0472947
|
6-chloro-7-fluoro-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
Show/Hide
|
C13H8ClFO2S
|
1
|
| 1 |
EC50 = 72 nM
|
|
|
|
CP0455455
|
6-cyano-8-fluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
Show/Hide
|
C13H6FNO3S
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0406185
|
6,9-difluoro-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
Show/Hide
|
C12H6F2O2S2
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0420084
|
6-cyano-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
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|
C14H9NO2S
|
1
|
| 1 |
EC50 = 82 nM
|
|
|
|
CP0414589
|
6-cyano-7-methoxy-4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
Show/Hide
|
C15H11NO3S
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0385487
|
2-(5-chloro-6-propylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C11H11ClN2O2S2
|
1
|
| 1 |
EC50 = 88 nM
|
|
|
|
CP0385489
|
2-(5-chloro-6-methylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C9H7ClN2O2S2
|
2
|
| 1 |
EC50 = 107 nM
|
|
|
| 2 |
EC50 = 157 nM
|
|
|
|
CP0512394
|
2-(7-cyclopropyl-6-methylthieno[3,2-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C12H12N2O2S2
|
1
|
| 1 |
EC50 = 115 nM
|
|
|
|
CP0420083
|
6-chloro-7-fluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
Show/Hide
|
C12H6ClFO3S
|
1
|
| 1 |
EC50 = 126 nM
|
|
|
|
CP0406184
|
5,5-dioxo-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
Show/Hide
|
C12H8O4S2
|
1
|
| 1 |
EC50 = 139 nM
|
|
|
|
CP0455149
|
2-(6-bromo-5-methylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C9H7BrN2O2S2
|
1
|
| 1 |
EC50 = 144 nM
|
|
|
|
CP0447120
|
6-fluoro-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
Show/Hide
|
C12H7FO2S2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0434373
|
N-[[4-[2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetyl]-1H-pyrrol-2-yl]methyl]cyclopropanesulfonamide
Show/Hide
|
C18H20N4O3S3
|
1
|
| 1 |
EC50 = 168 nM
|
|
|
|
CP0511164
|
6,8-dichloro-4H-thieno[3,2-c]chromene-2-carboxylic acid
Show/Hide
|
C12H6Cl2O3S
|
1
|
| 1 |
EC50 = 173 nM
|
|
|
|
CP0549215
|
6-fluoro-5,5-dioxo-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
Show/Hide
|
C12H7FO4S2
|
1
|
| 1 |
EC50 = 183 nM
|
|
|
|
CP0553202
|
8-fluoro-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
Show/Hide
|
C12H7FO2S2
|
1
|
| 1 |
EC50 = 186 nM
|
|
|
|
CP0385488
|
2-(5-bromo-6-methylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C9H7BrN2O2S2
|
1
|
| 1 |
EC50 = 208 nM
|
|
|
|
CP0555688
|
N-[[5-[2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetyl]furan-2-yl]methyl]-2-methylpropanamide
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|
C19H21N3O3S2
|
1
|
| 1 |
EC50 = 211 nM
|
|
|
|
CP0558261
|
N-[[5-[2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetyl]furan-2-yl]methyl]cyclopropanecarboxamide
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|
C19H19N3O3S2
|
1
|
| 1 |
EC50 = 249 nM
|
|
|
|
CP0550461
|
2-(5-chloro-6-cyclopropylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C11H9ClN2O2S2
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0545030
|
8-chloro-4H-thieno[3,2-c]chromene-2-carboxylic acid
Show/Hide
|
C12H7ClO3S
|
1
|
| 1 |
EC50 = 253 nM
|
|
|
|
CP0385485
|
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanyl-1-[5-(pyrrolidine-1-carbonyl)-1H-pyrrol-3-yl]ethanone
Show/Hide
|
C19H20N4O2S2
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0385490
|
2-(5-chloro-6-ethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C10H9ClN2O2S2
|
1
|
| 1 |
EC50 = 393 nM
|
|
|
|
CP0459445
|
N-cyano-2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetamide
Show/Hide
|
C11H10N4OS2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0561078
|
2-(6-bromo-7-methylthieno[3,2-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C9H7BrN2O2S2
|
1
|
| 1 |
EC50 = 417 nM
|
|
|
|
CP0434382
|
2-(6-chloro-7-methylthieno[3,2-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C9H7ClN2O2S2
|
1
|
| 1 |
EC50 = 435 nM
|
|
|
|
CP0385483
|
methyl 2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetate
Show/Hide
|
C11H12N2O2S2
|
1
|
| 1 |
EC50 = 445 nM
|
|
|
|
CP0553200
|
4H-thieno[3,2-c]thiochromene-2-carboxylic acid
Show/Hide
|
C12H8O2S2
|
1
|
| 1 |
EC50 = 461 nM
|
|
|
|
CP0516469
|
2-(5-chloro-6-propan-2-ylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C11H11ClN2O2S2
|
1
|
| 1 |
EC50 = 477 nM
|
|
|
|
CP0434371
|
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanyl-N-hydroxyacetamide
Show/Hide
|
C10H11N3O2S2
|
1
|
| 1 |
EC50 = 556 nM
|
|
|
|
CP0421067
|
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C10H10N2O2S2
|
1
|
| 1 |
EC50 = 570 nM
|
|
|
|
CP0447145
|
8-fluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
Show/Hide
|
C12H7FO3S
|
1
|
| 1 |
EC50 = 662 nM
|
|
|
|
CP0390443
|
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanyl-N-methylacetamide
Show/Hide
|
C11H13N3OS2
|
1
|
| 1 |
EC50 = 789 nM
|
|
|
|
CP0385486
|
2-(6-ethyl-5-methylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C11H12N2O2S2
|
1
|
| 1 |
EC50 = 835 nM
|
|
|
|
CP0390445
|
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetamide
Show/Hide
|
C10H11N3OS2
|
1
|
| 1 |
EC50 = 857 nM
|
|
|
|
CP0452379
|
2-(6,7-dimethylthieno[3,2-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C10H10N2O2S2
|
1
|
| 1 |
EC50 = 881 nM
|
|
|
|
CP0459446
|
2-(6-chloro-5-methylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C9H7ClN2O2S2
|
1
|
| 1 |
EC50 = 885 nM
|
|
|
|
CP0407493
|
4,5-dihydrobenzo[g][1]benzothiole-2-carboxylic acid
Show/Hide
|
C13H10O2S
|
1
|
| 1 |
EC50 = 1060 nM
|
|
|
|
CP0385484
|
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanyl-N-methylsulfonylacetamide
Show/Hide
|
C11H13N3O3S3
|
1
|
| 1 |
EC50 = 1462 nM
|
|
|
|
CP0459963
|
9-fluoro-4H-thieno[3,2-c]chromene-2-carboxylic acid
Show/Hide
|
C12H7FO3S
|
1
|
| 1 |
EC50 = 1878 nM
|
|
|
|
CP0520427
|
2-(7-chloro-6-methylthieno[3,2-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C9H7ClN2O2S2
|
1
|
| 1 |
EC50 = 1965 nM
|
|
|
|
CP0406183
|
5-oxo-4H-thieno[3,2-c]thiochromene-2-carboxylic acid
Show/Hide
|
C12H8O3S2
|
1
|
| 1 |
EC50 = 2309 nM
|
|
|
|
CP0167846
|
4H-thieno[3,2-c]chromene-2-carboxylic acid
Show/Hide
|
C12H8O3S
|
1
|
| 1 |
EC50 = 3875 nM
|
|
|
|
CP0452378
|
2-(5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetic acid
Show/Hide
|
C11H12N2O2S2
|
1
|
| 1 |
EC50 = 21928 nM
|
|
|
