| Compound ID |
Compound Name |
Compound Formula |
|
CP0192820
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid ((S)-1-benzyl-2-butylcarbamoyl-2-oxo-ethyl)-amide
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|
C27H33N3O7S
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
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CP0048127
|
(3S) 2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
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|
C22H24N2O6S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0342893
|
2-Methyl-1,1-dioxo-1,2,6,7-tetrahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
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|
C21H20N2O6S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0148043
|
6,7-Dichloro-2-methyl-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
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|
C19H18Cl2N2O4S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0172119
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid {(S)-1-benzyl-2-oxo-2-[2-(5-pyridin-2-yl-thiophene-2-sulfonylamino)-ethylcarbamoyl]-ethyl}-amide
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|
C34H35N5O9S3
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0177716
|
2-Methyl-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
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|
C19H20N2O4S
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0168893
|
2-Methyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid (5-benzenesulfonylamino-1-formyl-pentyl)-amide
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|
C24H29N3O8S2
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0185518
|
6,7-Dimethoxy-2-methyl-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
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|
C21H24N2O6S
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0362027
|
2-Methyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide(3R,3S diastereomeric mixture)
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|
C21H22N2O6S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0290024
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid {(S)-1-benzyl-2-[2-(4-fluoro-benzenesulfonylamino)-ethylcarbamoyl]-2-oxo-ethyl}-amide
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|
C31H33FN4O9S2
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0207897
|
2-Ethyl-1,1-dioxo-1,2,6,7-tetrahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid ((S)-1-benzyl-2-oxo-ethyl)-amide
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|
C22H22N2O6S
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0063942
|
6-Chloro-2-methyl-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
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|
C19H19ClN2O4S
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0133619
|
6,7-Dimethoxy-1,1-dioxo-3,4-dihydro-1H-1lambda*6*-benzo[c][1,2]oxathiine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide(3R,3S diastereomeric mixture)
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|
C20H21NO7S
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0370357
|
6-Fluoro-2-methyl-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide(3R,3S diastereomeric mixture)
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|
C19H19FN2O4S
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0288520
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid {(S)-1-benzyl-2-[3-(4-fluoro-benzenesulfonylamino)-propylcarbamoyl]-2-oxo-ethyl}-amide
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|
C32H35FN4O9S2
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0184142
|
2-Isopropyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide(3R,3S diastereomeric mixture)
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|
C23H26N2O6S
|
1
|
| 1 |
IC50 = 2600 nM
|
|
|
|
CP0193881
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid [(S)-2-(3-benzenesulfonylamino-propylcarbamoyl)-1-benzyl-2-oxo-ethyl]-amide
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|
C32H36N4O9S2
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0084259
|
6,7-Dichloro-2-methyl-1,1-dioxo-1,2-dihydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
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|
C19H16Cl2N2O4S
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0048650
|
4-Methoxy-2-methyl-1,1-dioxo-1,2-dihydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
Show/Hide
|
C20H20N2O5S
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0272619
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid {(S)-1-benzyl-2-[3-(4-nitro-benzenesulfonylamino)-propylcarbamoyl]-2-oxo-ethyl}-amide
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|
C32H35N5O11S2
|
1
|
| 1 |
IC50 = 3600 nM
|
|
|
|
CP0147827
|
2-Methyl-6-morpholin-4-yl-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[e][1,2]thiazine-3-carboxylic acid (1-benzyl-2-oxo-ethyl)-amide
Show/Hide
|
C23H27N3O5S
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
|
CP0208488
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid {(S)-1-benzyl-2-[2-(4-nitro-benzenesulfonylamino)-ethylcarbamoyl]-2-oxo-ethyl}-amide
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|
C31H33N5O11S2
|
1
|
| 1 |
IC50 = 4200 nM
|
|
|
|
CP0272483
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid [(S)-2-(2-benzenesulfonylamino-ethylcarbamoyl)-1-benzyl-2-oxo-ethyl]-amide
Show/Hide
|
C31H34N4O9S2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0113102
|
2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-1lambda*6*-thia-2-aza-anthracene-3-carboxylic acid (1-formyl-3-methyl-butyl)-amide
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|
C19H26N2O6S
|
1
|
| 1 |
IC50 > 3000 nM
|
|
|
