Brief Information of the Cell Line and Protein
Cell Line ID: CL000091 , MV4-11
Synonyms
MV-4-11
MV-4:11
MV4:11
MV 4;11
MV4;11
MV411
MV(4;11)
MV4II
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0064
Protein ID: PT02805 , CREB-binding protein
Gene Name CREBBP
Organism Homo sapiens, Human
Protein Classification Epigenetic regulator
Uniprot ID Q92793
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000091  Protein ID: PT02805
 
Compound ID Compound Name Compound Formula
CP0072530
3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-N-methyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamide
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C27H33F2N7O2
 1
1
EC50 = 6.6 nM
   TI
   LI
   LO
   TS
CP0127942
1-[3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone
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C27H32F2N6O2
 1
1
EC50 = 14 nM
   TI
   LI
   LO
   TS
CP0086089
1-[3-[2-fluoro-4-(1-methylpyrazol-4-yl)anilino]-1-[(3S)-oxolan-3-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone
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C22H25FN6O2
 1
1
EC50 = 910 nM
   TI
   LI
   LO
   TS