| Compound ID |
Compound Name |
Compound Formula |
|
CP0574846
|
N-[(1-methylindol-5-yl)methyl]-3-[[4-(trifluoromethoxy)phenoxy]methyl]azetidine-1-carboxamide
Show/Hide
|
C22H22F3N3O3
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0561785
|
N-[(1-methylindol-5-yl)methyl]-4-(4-methylphenoxy)benzamide
Show/Hide
|
C24H22N2O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0561788
|
N-[(1-methylindol-5-yl)methyl]-3-[(4-methylphenoxy)methyl]azetidine-1-carboxamide
Show/Hide
|
C22H25N3O2
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0547756
|
3-[(4-chlorophenoxy)methyl]-N-[(1-methylindol-5-yl)methyl]azetidine-1-carboxamide
Show/Hide
|
C21H22ClN3O2
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
|
CP0531394
|
3-[(4-methoxyphenoxy)methyl]-N-[(1-methylindol-5-yl)methyl]azetidine-1-carboxamide
Show/Hide
|
C22H25N3O3
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0573222
|
N-(1-methylindol-5-yl)-2-[4-(4-methylphenoxy)phenyl]-2-oxoacetamide
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|
C24H20N2O3
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0553137
|
N-[(1-methylindol-5-yl)methyl]-3-[[4-(trifluoromethyl)phenoxy]methyl]azetidine-1-carboxamide
Show/Hide
|
C22H22F3N3O2
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0423348
|
N-(3-fluoro-1-methylindol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H25FN4O2
|
1
|
| 1 |
EC50 = 85 nM
|
|
|
|
CP0003551
|
N-(1-methylindol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H26N4O2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0423350
|
N-(7-fluoro-1H-indol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C22H23FN4O2
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0520783
|
N-(1-methylindol-5-yl)-2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H25N3O3
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0553131
|
N-(1-methylindol-5-yl)-2-[6-(4-methylphenoxy)pyridin-3-yl]-2-oxoacetamide
Show/Hide
|
C23H19N3O3
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0531395
|
N-(1H-indol-5-ylmethyl)-3-[[4-(trifluoromethyl)phenoxy]methyl]azetidine-1-carboxamide
Show/Hide
|
C21H20F3N3O2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0562258
|
N-[(1-methylindol-5-yl)methyl]-3-(4-methylphenoxy)pyrrolidine-1-carboxamide
Show/Hide
|
C22H25N3O2
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0574828
|
N-[(1-methylindol-5-yl)methyl]-3-(phenoxymethyl)azetidine-1-carboxamide
Show/Hide
|
C21H23N3O2
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0553133
|
N-(3-fluoro-1-methylpyrrolo[2,3-b]pyridin-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C22H24FN5O2
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0561786
|
N-[(1-methylindol-5-yl)methyl]-4-(4-methylphenoxy)piperidine-1-carboxamide
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0553135
|
3-[(4-fluorophenoxy)methyl]-N-[(1-methylindol-5-yl)methyl]azetidine-1-carboxamide
Show/Hide
|
C21H22FN3O2
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0423347
|
N-(1H-indol-5-yl)-2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoacetamide
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
|
CP0561787
|
N-[(1-methylindol-5-yl)methyl]-3-[(4-methylphenoxy)methyl]pyrrolidine-1-carboxamide
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0570915
|
3-[(4-cyanophenoxy)methyl]-N-[(1-methylindol-5-yl)methyl]azetidine-1-carboxamide
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0573223
|
2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-N-(1-methylpyrrolo[2,3-b]pyridin-5-yl)-2-oxoacetamide
Show/Hide
|
C22H25N5O2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0423349
|
N-(3-chloro-1-methylindol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H25ClN4O2
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0553134
|
N-[(1-methylindol-5-yl)methyl]-4-[(4-methylphenyl)methyl]piperazine-1-carboxamide
Show/Hide
|
C23H28N4O
|
1
|
| 1 |
EC50 = 490 nM
|
|
|
|
CP0485193
|
N-(1-methylindol-5-yl)-2-[1-[(4-methylphenyl)methyl]piperidin-4-yl]-2-oxoacetamide
Show/Hide
|
C24H27N3O2
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0423351
|
N-[(1-methylindol-5-yl)methyl]-3-(4-methylphenoxy)azetidine-1-carboxamide
Show/Hide
|
C21H23N3O2
|
1
|
| 1 |
EC50 = 620 nM
|
|
|
|
CP0423406
|
N-(1-methylindol-5-yl)-2-[5-(4-methylphenoxy)pyrazin-2-yl]-2-oxoacetamide
Show/Hide
|
C22H18N4O3
|
1
|
| 1 |
EC50 = 650 nM
|
|
|
|
CP0471405
|
[5-(1-methylindol-4-yl)-1,3,4-oxadiazol-2-yl]-[4-[(4-methylphenyl)methyl]piperazin-1-yl]methanone
Show/Hide
|
C24H25N5O2
|
1
|
| 1 |
EC50 = 660 nM
|
|
|
|
CP0480132
|
N-(1-methylindol-5-yl)-2-[4-(6-methylpyridin-3-yl)oxycyclohexyl]-2-oxoacetamide
Show/Hide
|
C23H25N3O3
|
1
|
| 1 |
EC50 = 670 nM
|
|
|
|
CP0561784
|
N-(1-methyl-2,3-dihydroindol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H28N4O2
|
1
|
| 1 |
EC50 = 820 nM
|
|
|
|
CP0561783
|
N-(6-fluoro-1-methylindol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H25FN4O2
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0423357
|
N-(1H-indol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperidin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
EC50 = 910 nM
|
|
|
|
CP0553132
|
N-(1,3-dimethylindol-5-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C24H28N4O2
|
1
|
| 1 |
EC50 = 920 nM
|
|
|
|
CP0552986
|
N-(3-fluoro-1-methylindol-6-yl)-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C23H25FN4O2
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0423407
|
[4-[(4-chlorophenyl)methyl]piperazin-1-yl]-[2-methyl-5-(1-methylindol-5-yl)pyrazol-3-yl]methanone
Show/Hide
|
C25H26ClN5O
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
|
CP0548442
|
N-(1-methylindol-5-yl)-2-[3-[(4-methylphenoxy)methyl]azetidin-1-yl]-2-oxoacetamide
Show/Hide
|
C22H23N3O3
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0520784
|
N-indolizin-7-yl-2-[4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-oxoacetamide
Show/Hide
|
C22H24N4O2
|
1
|
| 1 |
EC50 = 3300 nM
|
|
|
