Brief Information of the Cell Line and Protein
Cell Line ID: CL000088 , Flp-In-293
Synonyms
Flp-In 293
293 Flp-In
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_U421
Protein ID: PT01494 , Beta-2 adrenergic receptor
Gene Name ADRB2
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P07550
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000088  Protein ID: PT01494
 
Compound ID Compound Name Compound Formula
CP0244206
7-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]thieno[2,3-c]pyridine
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C21H12F3N3OS
 1
1
Ki = 5900 nM
   TI
   LI
   LO
   TS
CP0369306
4-[4-imidazo[1,2-a]pyridin-5-yl-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
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C21H12F3N3O2
 1
1
Ki = 8600 nM
   TI
   LI
   LO
   TS
CP0064183
4-[3-methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy]furo[3,2-c]pyridine
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C21H16N4O2
 1
1
Ki = 9300 nM
   TI
   LI
   LO
   TS
CP0002070
1-(1H-Indol-3-yl)-2-propanamine
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C11H14N2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0002071
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N-prop-2-enylprop-2-en-1-amine
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C17H22N2O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0054519
(1R,12R,13S,17R,21S)-12-ethyl-18-propyl-7-(trifluoromethyl)-10,18-diazapentacyclo[11.7.1.02,11.04,9.017,21]henicosa-2(11),3,5,7,9-pentaene
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C25H31F3N2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0085414
(3aS,6R,6aS,9aR,9bR)-6-benzyl-1-methyl-3,3a,4,6,6a,7,8,9,9a,9b-decahydro-2H-benzo[de]quinolin-5-one
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C20H27NO
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0064188
4-[4-(6-methylimidazo[1,2-a]pyrazin-5-yl)-3-(trifluoromethyl)phenoxy]furo[3,2-c]pyridine
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C21H13F3N4O2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0127400
(-)-Pramipexole
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C10H17N3S
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS