Brief Information of the Cell Line and Protein
Cell Line ID: CL000077 , Ba/F3
Synonyms
BA/F3
BaF3
BAF3
Baf3
Category Factor-dependent cell line
Organism
Mus musculus (Mouse)
Cellosaurus ID
CVCL_0161
Protein ID: PT01664 , Tyrosine-protein kinase Fer
Gene Name FER
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P16591
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000077  Protein ID: PT01664
 
Compound ID Compound Name Compound Formula
CP0508321
7-[[(1R,2S)-2-aminocyclohexyl]amino]-5-(3-methylanilino)-4-oxo-3H-pyrido[3,4-d]pyridazine-8-carbonitrile
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C21H23N7O
 1
1
GI50 = 1.9 nM
   TI
   LI
   LO
   TS
CP0427066
7-[[(1R,2S)-2-aminocyclohexyl]amino]-5-(3-methylanilino)-3H-pyrido[3,4-d]pyridazin-4-one
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C20H24N6O
 1
1
GI50 = 69 nM
   TI
   LI
   LO
   TS
CP0482287
7-[(2-aminocyclohexyl)amino]-5-(3-methylanilino)-3H-pyrido[3,4-d]pyridazin-4-one
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C20H24N6O
 1
1
GI50 = 83 nM
   TI
   LI
   LO
   TS
CP0458204
7-[(2-aminocyclohexyl)amino]-8-chloro-5-(3-methylanilino)-3H-pyrido[3,4-d]pyridazin-4-one
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C20H23ClN6O
 1
1
GI50 = 120 nM
   TI
   LI
   LO
   TS
CP0420693
7-[[(1R,2S)-2-aminocyclohexyl]amino]-8-bromo-5-(3-methylanilino)-3H-pyrido[3,4-d]pyridazin-4-one
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C20H23BrN6O
 1
1
GI50 = 140 nM
   TI
   LI
   LO
   TS
CP0534495
6-[(2-aminocyclohexyl)amino]-8-(3-methylanilino)-2H-2,7-naphthyridin-1-one
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C21H25N5O
 1
1
GI50 = 460 nM
   TI
   LI
   LO
   TS
CP0531980
6-[(2-aminocyclohexyl)amino]-8-(3-methylanilino)-3,4-dihydro-2H-2,7-naphthyridin-1-one
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C21H27N5O
 1
1
GI50 = 480 nM
   TI
   LI
   LO
   TS
CP0427064
3-amino-6-[(2-aminocyclohexyl)amino]-1-benzylpyrrolo[2,3-b]pyridine-5-carbonitrile
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C21H24N6
 1
1
GI50 > 4000 nM
   TI
   LI
   LO
   TS