| Compound ID |
Compound Name |
Compound Formula |
|
CP0084905
|
(2S)-N-[4-[3-cyano-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]indazol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C25H24N6O3
|
1
|
| 1 |
IC50 = 67 nM
|
|
|
|
CP0072063
|
(2S)-N-[4-[3-cyano-1-(2-methyl-1-oxo-3H-isoindol-5-yl)indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C29H25N5O3
|
2
|
| 1 |
IC50 = 140 nM
|
|
|
| 2 |
IC50 = 2180 nM
|
|
|
|
CP0084903
|
(2S)-N-[4-[3-cyano-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C26H25N5O3
|
2
|
| 1 |
IC50 = 281 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0084899
|
(2S)-N-[4-[3-cyano-1-(2-methylpropyl)indazol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C23H25N5O2
|
2
|
| 1 |
IC50 = 297 nM
|
|
|
| 2 |
IC50 = 15400 nM
|
|
|
|
CP0084901
|
(2S)-N-[4-[3-cyano-1-(2-methylpropyl)indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C24H26N4O2
|
2
|
| 1 |
IC50 = 343 nM
|
|
|
| 2 |
IC50 = 5770 nM
|
|
|
|
CP0259656
|
(2S)-N-[4-[3-cyano-1-(oxan-4-ylmethyl)indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C26H28N4O3
|
2
|
| 1 |
IC50 = 633 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0072065
|
(2S)-N-[4-[1-methyl-3-(1-methylpyrazol-4-yl)indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C24H25N5O2
|
2
|
| 1 |
IC50 = 979 nM
|
|
|
| 2 |
IC50 = 9710 nM
|
|
|
|
CP0246772
|
(2S)-N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C22H22N4O2
|
2
|
| 1 |
IC50 = 3050 nM
|
|
|
| 2 |
IC50 = 12000 nM
|
|
|
|
CP0119441
|
(2S)-N-[4-(1-benzyl-3-cyanoindol-5-yl)oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C27H24N4O2
|
1
|
| 1 |
IC50 = 6950 nM
|
|
|
|
CP0524302
|
(2S)-N-[4-[3-cyano-1-[2-(dimethylamino)ethyl]indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C24H27N5O2
|
2
|
| 1 |
IC50 = 7480 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0282315
|
(2S)-N-[4-(3-cyano-1-phenylindol-5-yl)oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C26H22N4O2
|
1
|
| 1 |
IC50 = 8710 nM
|
|
|
|
CP0111468
|
2-amino-N-[4-(2-amino-1-benzyl-3-cyanoindol-5-yl)oxyphenyl]acetamide
Show/Hide
|
C24H21N5O2
|
2
|
| 1 |
IC50 = 12600 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0072066
|
(2S)-N-[4-[[3-cyano-1-(2-methylpropyl)indol-5-yl]-methylamino]phenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C25H29N5O
|
2
|
| 1 |
IC50 = 13700 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0172548
|
(2S)-N-[4-[3-cyano-1-(2-methylpropyl)indol-5-yl]sulfanylphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C24H26N4OS
|
1
|
| 1 |
IC50 = 14000 nM
|
|
|
|
CP0051690
|
(2S)-N-[4-[3-cyano-1-[2-(methylamino)-2-oxoethyl]indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C23H23N5O3
|
2
|
| 1 |
IC50 = 14000 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0172543
|
2-amino-N-[4-[2-amino-3-cyano-1-(2-methylpropyl)indol-5-yl]oxyphenyl]acetamide
Show/Hide
|
C21H23N5O2
|
2
|
| 1 |
IC50 = 16400 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0084898
|
(2S)-N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]azetidine-2-carboxamide
Show/Hide
|
C21H20N4O2
|
1
|
| 1 |
IC50 = 19600 nM
|
|
|
|
CP0282316
|
(2S)-N-[4-[3-cyano-1-(2-methylpropyl)indol-5-yl]sulfonylphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C24H26N4O3S
|
2
|
| 1 |
IC50 = 24700 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
|
CP0051689
|
(2S)-N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]-N-methylpyrrolidine-2-carboxamide
Show/Hide
|
C23H24N4O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0051691
|
(2S)-N-[4-[[3-cyano-1-(2-methylpropyl)indol-5-yl]amino]phenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C24H27N5O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0072062
|
N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]-2-(methylamino)acetamide
Show/Hide
|
C20H20N4O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0072899
|
2-amino-N-[4-(2-amino-3-cyano-1-methylindol-5-yl)oxyphenyl]acetamide
Show/Hide
|
C18H17N5O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0117230
|
2-amino-N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]acetamide
Show/Hide
|
C19H18N4O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0154584
|
2-amino-N-[4-[2-amino-3-cyano-1-[2-(dimethylamino)-2-oxoethyl]indol-5-yl]oxyphenyl]acetamide
Show/Hide
|
C21H22N6O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0170151
|
N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]-2-(dimethylamino)acetamide
Show/Hide
|
C21H22N4O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0171547
|
2-amino-N-[4-[[3-(1-methylpyrazol-4-yl)-1H-indazol-5-yl]oxy]phenyl]acetamide
Show/Hide
|
C19H18N6O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0172545
|
(2R)-N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0317360
|
(2S)-N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]-N-methyl-5-oxopyrrolidine-2-carboxamide
Show/Hide
|
C23H22N4O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0488237
|
(2S)-N-[4-(3-cyano-1-ethylindol-5-yl)oxyphenyl]piperidine-2-carboxamide
Show/Hide
|
C23H24N4O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0780865
|
(2S)-N-[4-[[3-(1-Methylpyrazol-4-yl)-1H-indol-5-yl]oxy]-phenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C23H23N5O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0051697
|
(2S)-N-[4-[[3-cyano-1-(2-methylpropyl)indol-5-yl]methyl]phenyl]pyrrolidine-2-carboxamide
Show/Hide
|
C25H28N4O
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0157996
|
2-amino-N-[4-(2-amino-3-cyano-1-ethylindol-5-yl)oxyphenyl]acetamide
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0709800
|
(2S)-2-Amino-N-[4-[(2-amino-3-cyano-1H-indol-5-yl)oxy]phenyl]-3-hydroxy-propanamide
Show/Hide
|
C18H17N5O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
