Compound ID |
Compound Name |
Compound Formula |
CP0049593
|
2-(4-chloro-N-[4-[2-(2-methoxyethoxy)ethoxy]phenyl]sulfonylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
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|
C27H27ClN4O7S
|
2
|
1 |
IC50 = 7 nM
|
|
|
2 |
Ki = 3 nM
|
|
|
CP0377968
|
CHEMBL2113185
Show/Hide
|
C28H28ClN5O6S
|
2
|
1 |
IC50 = 7 nM
|
|
|
2 |
Ki = 0.9 nM
|
|
|
CP0176028
|
CHEMBL2113211
Show/Hide
|
C25H23ClN4O6S
|
2
|
1 |
IC50 = 8 nM
|
|
|
2 |
Ki = 7 nM
|
|
|
CP0198143
|
CHEMBL2113201
Show/Hide
|
C27H28ClN5O5S
|
2
|
1 |
IC50 = 14 nM
|
|
|
2 |
Ki = 1.1 nM
|
|
|
CP0302223
|
(Z)-3-(4-(N-(4-chlorophenyl)-N-(2-oxo-2-(2-(2-oxoindolin-3-ylidene)hydrazinyl)ethyl)sulfamoyl)phenyl)-N-(3-(dimethylamino)propyl)propanamide
Show/Hide
|
C30H33ClN6O5S
|
2
|
1 |
IC50 = 14 nM
|
|
|
2 |
Ki = 0.65 nM
|
|
|
CP0485778
|
2-(4-chloro-N-[4-[3-(dimethylamino)propoxy]phenyl]sulfonylanilino)-N-[(1-hydroxy-3-oxo-2H-isoquinolin-4-yl)imino]acetamide
Show/Hide
|
C28H28ClN5O6S
|
2
|
1 |
IC50 = 15 nM
|
|
|
2 |
Ki = 1.6 nM
|
|
|
CP0070065
|
4-ethoxy-N-(2-oxo-2-(2-(2-oxoindolin-3-ylidene)hydrazinyl)ethyl)-N-p-tolylbenzenesulfonamide
Show/Hide
|
C25H24N4O5S
|
2
|
1 |
IC50 = 30 nM
|
|
|
2 |
Ki = 14 nM
|
|
|
CP0250764
|
2-(4-chloro-N-[4-(3-hydroxypropyl)phenyl]sulfonylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C25H23ClN4O5S
|
2
|
1 |
IC50 = 32 nM
|
|
|
2 |
Ki = 4.1 nM
|
|
|
CP0250765
|
CHEMBL2113177
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|
C28H29ClN6O5S
|
2
|
1 |
IC50 = 49 nM
|
|
|
2 |
Ki = 7 nM
|
|
|
CP0177122
|
(2S)-5-amino-2-{[(2S)-1-{[(4R,7S,10S,13S,16R)-13-[(2S)-butan-2-yl]-7-(carbamoylmethyl)-16-[(4-ethoxyphenyl)methyl]-10-[(1R)-1-hydroxyethyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosan-4-yl]carbonyl}pyrrolidin-2-yl]formamido}-N-(carbamoylmethyl)pentanamide
Show/Hide
|
C43H67N11O12S2
|
2
|
1 |
IC50 = 59 nM
|
|
|
2 |
Ki = 27 nM
|
|
|
CP0198144
|
2-(4-chloro-N-[4-[2-(dimethylamino)ethoxy]phenyl]sulfonylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C26H26ClN5O5S
|
2
|
1 |
IC50 = 59 nM
|
|
|
2 |
Ki = 2.1 nM
|
|
|
CP0446409
|
2-(4-chloro-N-[4-[3-(dimethylamino)propoxy]phenyl]sulfonylanilino)-N-[(2-hydroxy-1H-pyrrolo[3,2-c]pyridin-3-yl)imino]acetamide
Show/Hide
|
C26H27ClN6O5S
|
2
|
1 |
IC50 = 840 nM
|
|
|
2 |
Ki = 115 nM
|
|
|
CP0483645
|
3-[4-[(4-chlorophenyl)-[2-[(2-hydroxy-1H-indol-3-yl)diazenyl]-2-oxoethyl]sulfamoyl]phenyl]-N-(3-hydroxypropyl)propanamide
Show/Hide
|
C28H28ClN5O6S
|
1
|
1 |
Ki = 0.9 nM
|
|
|
CP0303775
|
CHEMBL2113198
Show/Hide
|
C24H21ClN4O5S
|
1
|
1 |
Ki = 3.9 nM
|
|
|
CP0292348
|
2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin-3-yl)-5-methyl-4H-1,2,4-triazol-3-yl)pyrazine
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|
C20H17FN6O
|
1
|
1 |
Ki = 6 nM
|
|
|
CP0439005
|
2-[N-(benzenesulfonyl)-4-chloroanilino]-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C22H17ClN4O4S
|
1
|
1 |
Ki = 8.7 nM
|
|
|
CP0194007
|
5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5-(methoxymethyl)-4H-1,2,4-triazol-4-yl)-2-methoxypyridine
Show/Hide
|
C19H19ClFN5O3
|
1
|
1 |
Ki = 9.5 nM
|
|
|
CP0480330
|
2-(4-chloro-N-(4-propoxyphenyl)sulfonylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C25H23ClN4O5S
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0718296
|
N-(4-chlorophenyl)-4-ethoxy-N-(2-(2-(2-hydroxybenzylidene)hydrazinyl)-2-oxoethyl)benzenesulfonamide
Show/Hide
|
C23H22ClN3O5S
|
1
|
1 |
Ki = 15 nM
|
|
|
CP0198146
|
2-(N-(4-butoxyphenyl)sulfonyl-4-chloroanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C26H25ClN4O5S
|
1
|
1 |
Ki = 18 nM
|
|
|
CP0889531
|
N-(4-chlorophenyl)-3,4-dimethoxy-N-{2-oxo-2-[(2E)-2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}benzenesulfonamide
Show/Hide
|
C24H21ClN4O6S
|
1
|
1 |
Ki = 18 nM
|
|
|
CP0467144
|
CHEMBL2113215
Show/Hide
|
C24H22N4O5S
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0515591
|
N-[(2-hydroxy-1H-indol-3-yl)imino]-2-(4-methyl-N-(4-propoxyphenyl)sulfonylanilino)acetamide
Show/Hide
|
C26H26N4O5S
|
1
|
1 |
Ki = 21 nM
|
|
|
CP0331982
|
5-(3-(4-ethoxy-3-methylphenyl)-5-(ethoxymethyl)-4H-1,2,4-triazol-4-yl)-2-methoxypyridine
Show/Hide
|
C20H24N4O3
|
1
|
1 |
Ki = 28 nM
|
|
|
CP0483731
|
2-(4-chloro-N-(4-propylphenyl)sulfonylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C25H23ClN4O4S
|
1
|
1 |
Ki = 36 nM
|
|
|
CP0910329
|
4-ethoxy-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-N-phenylbenzenesulfonamide
Show/Hide
|
C24H22N4O5S
|
1
|
1 |
Ki = 36 nM
|
|
|
CP0464488
|
2-(4-chloro-N-thiophen-2-ylsulfonylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C20H15ClN4O4S2
|
1
|
1 |
Ki = 37 nM
|
|
|
CP0415346
|
(R)-(4-(methoxyimino)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl)(2'-methylbiphenyl-4-yl)methanone
Show/Hide
|
C22H22N4O3
|
1
|
1 |
Ki = 50 nM
|
|
|
CP0415340
|
2-methoxy-5-(3-(2'-methoxybiphenyl-4-yl)-5-methyl-4H-1,2,4-triazol-4-yl)pyridine
Show/Hide
|
C22H20N4O2
|
1
|
1 |
Ki = 56 nM
|
|
|
CP0910343
|
4-ethoxy-N-{2-[2-(2-hydroxybenzylidene)hydrazino]-2-oxoethyl}-N-(4-methylphenyl)benzenesulfonamide
Show/Hide
|
C24H25N3O5S
|
1
|
1 |
Ki = 60 nM
|
|
|
CP0453756
|
2-(N-(4-tert-butylphenyl)sulfonyl-4-chloroanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C26H25ClN4O4S
|
1
|
1 |
Ki = 61 nM
|
|
|
CP0321565
|
2-(4-chloro-N-(4-ethoxyphenyl)sulfonylanilino)-N-[(2-hydroxy-1H-pyrrolo[3,2-c]pyridin-3-yl)imino]acetamide
Show/Hide
|
C23H20ClN5O5S
|
1
|
1 |
Ki = 64 nM
|
|
|
CP0341519
|
2-[N-(benzenesulfonyl)-4-methylanilino]-N-[(E)-(2-hydroxyphenyl)methylideneamino]acetamide
Show/Hide
|
C22H21N3O4S
|
1
|
1 |
Ki = 67 nM
|
|
|
CP0377965
|
2-[N-(benzenesulfonyl)-4-chloroanilino]-N-[(E)-(2-hydroxyphenyl)methylideneamino]acetamide
Show/Hide
|
C21H18ClN3O4S
|
1
|
1 |
Ki = 67 nM
|
|
|
CP0393452
|
2-[N-(benzenesulfonyl)anilino]-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C22H18N4O4S
|
1
|
1 |
Ki = 90 nM
|
|
|
CP0441895
|
2-[N-(benzenesulfonyl)-4-methylanilino]-N-(3-chloro-2-methylphenyl)acetamide
Show/Hide
|
C22H21ClN2O3S
|
1
|
1 |
Ki = 93 nM
|
|
|
CP0107768
|
2-[Benzenesulfonyl-(4-methoxy-phenyl)-amino]-N-(3-chloro-2-methyl-phenyl)-acetamide
Show/Hide
|
C22H21ClN2O4S
|
1
|
1 |
Ki = 100 nM
|
|
|
CP0907489
|
N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}[1,1'-biphenyl]-4-sulfonamide
Show/Hide
|
C29H24N4O4S
|
1
|
1 |
Ki = 104 nM
|
|
|
CP0453758
|
methyl 3-[[2-(4-chloro-N-[4-[3-(dimethylamino)propoxy]phenyl]sulfonylanilino)acetyl]diazenyl]-2-hydroxy-1H-indole-7-carboxylate
Show/Hide
|
C29H30ClN5O7S
|
1
|
1 |
Ki = 109 nM
|
|
|
CP0498457
|
CHEMBL2113205
Show/Hide
|
C24H19N5O4S
|
1
|
1 |
Ki = 111 nM
|
|
|
CP0224226
|
N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-N-(4-methoxyphenyl)benzenesulfonamide
Show/Hide
|
C24H24N2O4S
|
1
|
1 |
Ki = 160 nM
|
|
|
CP0480329
|
2-[N-(benzenesulfonyl)-4-chloroanilino]-N-(3-chloro-2-methylphenyl)acetamide
Show/Hide
|
C21H18Cl2N2O3S
|
1
|
1 |
Ki = 160 nM
|
|
|
CP0453759
|
N-[(2-hydroxy-1H-indol-3-yl)imino]-2-(4-methyl-N-naphthalen-1-ylsulfonylanilino)acetamide
Show/Hide
|
C27H22N4O4S
|
1
|
1 |
Ki = 174 nM
|
|
|
CP0916890
|
N'-(1-(2-hydroxyphenyl)ethylidene)-2-(N-phenylphenylsulfonamido)acetohydrazide
Show/Hide
|
C22H21N3O4S
|
1
|
1 |
Ki = 237 nM
|
|
|
CP0847573
|
N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}-2-naphthalenesulfonamide
Show/Hide
|
C27H22N4O4S
|
1
|
1 |
Ki = 239 nM
|
|
|
CP0493159
|
4-{2-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4-yl)-phenoxy]-ethyl}-morpholine
Show/Hide
|
C27H28N4O2
|
1
|
1 |
Ki = 304 nM
|
|
|
CP0441813
|
2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
Show/Hide
|
C27H29N3O6S
|
1
|
1 |
Ki = 320 nM
|
|
|
CP0485597
|
2-[3-[[2-(4-chloro-N-[4-[3-(dimethylamino)propoxy]phenyl]sulfonylanilino)acetyl]diazenyl]-2-hydroxyindol-1-yl]acetamide
Show/Hide
|
C29H31ClN6O6S
|
1
|
1 |
Ki = 322 nM
|
|
|
CP0480327
|
2-(N-(4-ethoxyphenyl)sulfonyl-4-methylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]propanamide
Show/Hide
|
C26H26N4O5S
|
1
|
1 |
Ki = 448 nM
|
|
|
CP0480328
|
N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-N-(4-methylphenyl)benzenesulfonamide
Show/Hide
|
C24H24N2O3S
|
1
|
1 |
Ki = 470 nM
|
|
|
CP0391566
|
2-(2-(2-(4-ethoxy-N-p-tolylphenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)acetamide
Show/Hide
|
C28H31N3O5S
|
1
|
1 |
Ki = 500 nM
|
|
|
CP0391575
|
2-(2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)acetamide
Show/Hide
|
C28H31N3O6S
|
1
|
1 |
Ki = 510 nM
|
|
|
CP0453757
|
N-(3-chloro-2-methylphenyl)-2-(N-(3,4-dimethoxyphenyl)sulfonyl-4-methylanilino)acetamide
Show/Hide
|
C24H25ClN2O5S
|
1
|
1 |
Ki = 620 nM
|
|
|
CP0467145
|
2-(2-(4-ethoxy-N-(4-methoxyphenyl)phenylsulfonamido)acetyl)isoindoline-1-carboxamide
Show/Hide
|
C26H27N3O6S
|
1
|
1 |
Ki = 770 nM
|
|
|
CP0393401
|
2-[N-(benzenesulfonyl)-4-methoxyanilino]-N-(4-chloro-2-methylphenyl)acetamide
Show/Hide
|
C22H21ClN2O4S
|
1
|
1 |
Ki = 800 nM
|
|
|
CP0377964
|
2-(N-(4-ethoxyphenyl)sulfonyl-4-methylanilino)-3-hydroxy-N-[(2-hydroxy-1H-indol-3-yl)imino]propanamide
Show/Hide
|
C26H26N4O6S
|
1
|
1 |
Ki = 1376 nM
|
|
|
CP0391565
|
2-(4-chloro-N-[4-(2-methylbutan-2-yl)phenyl]sulfonylanilino)-N-[(2-hydroxy-1H-indol-3-yl)imino]acetamide
Show/Hide
|
C27H27ClN4O4S
|
1
|
1 |
Ki = 1750 nM
|
|
|
CP0684505
|
N-(4-chlorophenyl)-4-ethoxy-N-(2-oxo-2-(2-(pyridin-2-ylmethylene)hydrazinyl)ethyl)benzenesulfonamide
Show/Hide
|
C22H21ClN4O4S
|
1
|
1 |
Ki = 2750 nM
|
|
|
CP0854598
|
2-(N-(3-chlorophenyl)phenylsulfonamido)-N'-(1-(2-hydroxyphenyl)ethylidene)acetohydrazide
Show/Hide
|
C22H20ClN3O4S
|
1
|
1 |
Ki = 4900 nM
|
|
|
CP0393402
|
2-[N-(benzenesulfonyl)-4-ethoxyanilino]-N-(3-chloro-2-methylphenyl)acetamide
Show/Hide
|
C23H23ClN2O4S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0847574
|
4-ethoxy-N-(2-{(2E)-2-[1-(1-hydroxy-2-naphthyl)ethylidene]hydrazino}-2-oxoethyl}-N-(4-methylphenyl)benzenesulfonamide
Show/Hide
|
C29H29N3O5S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0853634
|
N-(2-{2-[4-(diethylamino)-2-hydroxybenzylidene]hydrazino}-2-oxoethyl)-4-ethoxy-N-(4-methylphenyl)benzenesulfonamide
Show/Hide
|
C28H34N4O5S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0854609
|
N-{2-{(E)-[2-(2-{[(4-ethoxyphenyl)sulfonyl]-4-methylanilino}acetyl)hydrazono]methyl}phenyl)acetamide
Show/Hide
|
C26H28N4O5S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0879679
|
N-{2-[(2E)-2-(2-aminobenzylidene)hydrazino]-2-oxoethyl}-4-ethoxy-N-(4-methylphenyl)benzenesulfonamide
Show/Hide
|
C24H26N4O4S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0889528
|
3-({[4-chloro({4-[3-(dimethylamino)propoxy]phenyl}sulfonyl)anilino]acetyl}hydrazono)-2-oxo-2,3-dihydro-1H-indole-7-carboxylic acid
Show/Hide
|
C28H28ClN5O7S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0889529
|
N-(4-chlorophenyl)-4-ethoxy-N-{2-[(2E)-2-(1H-imidazol-2-ylmethylene)hydrazino]-2-oxoethyl}benzenesulfonamide
Show/Hide
|
C20H20ClN5O4S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0889532
|
4-ethoxy-N-(2-{2-[(2-hydroxy-1-naphthyl)methylene]hydrazino}-2-oxoethyl}-N-(4-methylphenyl)benzenesulfonamide
Show/Hide
|
C29H29N3O5S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0889533
|
3-[({[(4-ethoxyphenyl)sulfonyl]-4-methylanilino}-acetyl)hydrazono]-2-oxo-2,3-dihydro-1H-indole-5-sulfonic acid
Show/Hide
|
C25H24N4O8S2
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0889534
|
4-ethoxy-N-(4-methylphenyl)-N-{3-oxo-3-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]propyl}benzenesulfonamide
Show/Hide
|
C26H26N4O5S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0904928
|
4-ethoxy-N-{2-[2-(5-nitro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]-2-oxoethyl}-N-phenylbenzenesulfonamide
Show/Hide
|
C24H21N5O7S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0910289
|
4-ethoxy-N-{2-[2-(5-iodo-2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]-2-oxoethyl}-N-phenylbenzenesulfonamide
Show/Hide
|
C24H21IN4O5S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0926723
|
N-(2-{2-[1-(2,4-dihydroxyphenyl)ethylidene]hydrazino}-2-oxoethyl)-4-ethoxy-N-(4-methylphenyl)benzenesulfonamide
Show/Hide
|
C25H27N3O6S
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0911081
|
4'-methoxy-N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1,2-dihydro-3H-indol-3-ylidene)hydrazino]ethyl}[1,1'-biphenyl]-4-sulfonamide
Show/Hide
|
C30H26N4O5S
|
1
|
1 |
Ki > 214 nM
|
|
|