Brief Information of the Cell Line and Protein
Cell Line ID: CL000064 , Chem-1
 Cell Line Info 
Synonyms
ChemiSCREEN Chem-1
Wild-type control Chem-1 cell line
ChemiSCREEN Chem-1 parental cell line
Category Undefined cell line type
Organism
Rattus norvegicus (Rat)
Cellosaurus ID
CVCL_L474
Protein ID: PT01298 , Cannabinoid receptor 1
 Protein Info 
Gene Name CNR1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P21554
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000064
 Cell Line Info 
 Protein ID: PT01298
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0000753
 Compound Info 
(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-[[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]-1-[(2S)-2-[[(2S,3R)-2-[[(2S)-2-(hexadecanoylamino)-3-methylbutanoyl]amino]-3-hydroxybutanoyl]amino]-4-methylpentanoyl]pyrrolidine-2-carboxamide
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C88H137N17O18
  2
1
EC50 > 30000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
IC50 > 30000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0050487
 Compound Info 
(11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphthalen-1-ylcarbonyl)-9-oxa-1-azatricyclo[6.3.1.0^{4,12}]dodeca-2,4(12),5,7-tetraene
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C27H26N2O3
  2
1
IC50 = 200 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
Ki = 150 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS