Compound ID |
Compound Name |
Compound Formula |
CP0036082
|
N-(3-chloro-4-fluorophenyl)-7-methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4-amine
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|
C22H24ClFN4O3
|
1
|
1 |
IC50 = 12.5 nM
|
|
|
CP0404829
|
2-cyano-N-[(2-hydroxy-5-morpholin-4-ylsulfonyl-1H-indol-3-yl)imino]acetamide
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|
C15H15N5O5S
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0007142
|
N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[(2-methylsulfonylethylamino)methyl]furan-2-yl]quinazolin-4-amine
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|
C29H26ClFN4O4S
|
1
|
1 |
IC50 = 27.1 nM
|
|
|
CP0471157
|
5-morpholin-4-ylsulfonyl-3-phenyldiazenyl-1H-indol-2-ol
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|
C18H18N4O4S
|
1
|
1 |
IC50 = 46 nM
|
|
|
CP0553866
|
3-(4-methoxyphenyl)-9-morpholin-4-ylsulfonyl-1-oxo-6,11a-dihydroindolo[3,2-b]quinoxaline-2,4-dicarbonitrile
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|
C27H20N6O5S
|
1
|
1 |
IC50 = 108 nM
|
|
|
CP0533473
|
N-[(2-hydroxy-5-morpholin-4-ylsulfonyl-1H-indol-3-yl)imino]-2-iminochromene-3-carboxamide
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|
C22H19N5O6S
|
1
|
1 |
IC50 = 205 nM
|
|
|
CP0565279
|
3-(4-hydroxyphenyl)imino-5-morpholin-4-ylsulfonyl-1H-indol-2-one
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|
C18H17N3O5S
|
1
|
1 |
IC50 = 751 nM
|
|
|
CP0519137
|
5-morpholin-4-ylsulfonyl-3-[4-[(5-morpholin-4-ylsulfonyl-2-oxo-1H-indol-3-ylidene)amino]phenyl]imino-1H-indol-2-one
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|
C30H28N6O8S2
|
1
|
1 |
IC50 = 1182 nM
|
|
|
CP0457718
|
2-amino-4-(4-methoxyphenyl)-1-[(Z)-(5-morpholin-4-ylsulfonyl-2-oxo-1H-indol-3-ylidene)amino]-6-oxopyridine-3,5-dicarbonitrile
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|
C26H21N7O6S
|
1
|
1 |
IC50 = 1931 nM
|
|
|
CP0033646
|
AZD-9291
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|
C28H33N7O2
|
1
|
1 |
IC50 = 2239 nM
|
|
|
CP0486473
|
3-[4-(3-bromoanilino)-6-methoxyquinazolin-7-yl]oxypropyl 3-(prop-2-enyldisulfanyl)propanoate
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|
C24H26BrN3O4S2
|
1
|
1 |
IC50 > 10000 nM
|
|
|