Compound ID |
Compound Name |
Compound Formula |
CP0060236
|
Balicatib
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|
C23H33N5O2
|
1
|
1 |
IC50 = 48 nM
|
|
|
CP0146153
|
(2S)-N-(cyanomethyl)-3-cyclohexyl-2-(phenylformamido)propanamide
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|
C18H23N3O2
|
1
|
1 |
IC50 = 230 nM
|
|
|
CP0041940
|
(2R)-N-(cyanomethyl)-4-methyl-2-{3-[4-(piperazin-1-yl)phenyl]phenyl}pentanamide
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|
C24H30N4O
|
1
|
1 |
IC50 = 320 nM
|
|
|
CP0134851
|
N-[1-(cyanomethylcarbamoyl)cyclohexyl]-4-[2-(4-methylpiperazin-1-yl)-1,3-thiazol-4-yl]benzamide
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|
C24H30N6O2S
|
1
|
1 |
IC50 = 340 nM
|
|
|
CP0077258
|
N-{1-[(cyanomethyl)carbamoyl]cyclohexyl}-4-[2-(morpholin-4-yl)-1,3-thiazol-4-yl]benzamide
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|
C23H27N5O3S
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0077259
|
N-{1-[(cyanomethyl)carbamoyl]cyclohexyl}-4-(morpholin-4-yl)benzamide
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|
C20H26N4O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|