| Compound ID |
Compound Name |
Compound Formula |
|
CP0556950
|
N-[(1S)-1-[3-(2-cyclopropylpyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C18H17F3N6O2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0444680
|
N-[(1S)-1-[3-(2-methoxypyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C16H15F3N6O3
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0537139
|
2-methyl-5-(trifluoromethyl)-N-[(1S)-1-[3-[2-(trifluoromethyl)pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-3-carboxamide
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|
C16H12F6N6O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0565077
|
N-[(1S)-1-[3-[2-(difluoromethyl)pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C16H13F5N6O2
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0451216
|
N-[(1S)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C16H13F4N5O2
|
1
|
| 1 |
IC50 = 136 nM
|
|
|
|
CP0563812
|
2-methyl-N-[(1S)-1-[3-(2-methylpyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C16H15F3N6O2
|
1
|
| 1 |
IC50 = 165 nM
|
|
|
|
CP0572892
|
5-cyclopropyl-2-methyl-N-[(1S)-1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-3-carboxamide
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|
C19H21N5O2
|
1
|
| 1 |
IC50 = 167 nM
|
|
|
|
CP0451217
|
2-methyl-N-[(1S)-1-[3-[2-(methylamino)pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C16H16F3N7O2
|
1
|
| 1 |
IC50 = 195 nM
|
|
|
|
CP0551767
|
N-[(1S)-1-[3-[2-(methoxymethyl)pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C17H17F3N6O3
|
1
|
| 1 |
IC50 = 322 nM
|
|
|
|
CP0537137
|
5-ethyl-2-methyl-N-[(1S)-1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-3-carboxamide
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|
C18H21N5O2
|
1
|
| 1 |
IC50 = 335 nM
|
|
|
|
CP0568334
|
N-[(1S)-1-[3-[2-(dimethylamino)pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C17H18F3N7O2
|
1
|
| 1 |
IC50 = 454 nM
|
|
|
|
CP0520861
|
N-[(1S)-1-[3-(2-methoxy-6-methylpyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C17H17F3N6O3
|
1
|
| 1 |
IC50 = 505 nM
|
|
|
|
CP0520860
|
2-methyl-N-[(1S)-1-[3-(2-pyrrolidin-1-ylpyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C19H20F3N7O2
|
1
|
| 1 |
IC50 = 573 nM
|
|
|
|
CP0444682
|
N-[(1S)-1-[3-[2-[(1S)-1-methoxyethyl]pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C18H19F3N6O3
|
1
|
| 1 |
IC50 = 744 nM
|
|
|
|
CP0572077
|
N-[(1S)-1-[3-[2-[(1R)-1-methoxyethyl]pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C18H19F3N6O3
|
1
|
| 1 |
IC50 = 778 nM
|
|
|
|
CP0549602
|
2-methyl-N-[1-[5-(3-methylphenyl)-1,2,4-oxadiazol-3-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C17H16F3N5O2
|
1
|
| 1 |
IC50 = 977 nM
|
|
|
|
CP0560235
|
2-methyl-N-[(1S)-1-[3-(5-methylpyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C16H15F3N6O2
|
1
|
| 1 |
IC50 = 1373 nM
|
|
|
|
CP0553346
|
2-methyl-N-[(1S)-1-[3-(6-methylpyrimidin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
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|
C15H14F3N7O2
|
1
|
| 1 |
IC50 = 1410 nM
|
|
|
|
CP0560109
|
2-methyl-N-[1-[1-(3-methylphenyl)pyrazol-4-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C18H18F3N5O
|
1
|
| 1 |
IC50 = 1597 nM
|
|
|
|
CP0572893
|
5-cyclopropyl-2-methyl-N-[1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-3-carboxamide
Show/Hide
|
C19H21N5O2
|
1
|
| 1 |
IC50 = 1876 nM
|
|
|
|
CP0520859
|
2-methyl-N-[(1S)-1-[3-(1-methylpyrazol-4-yl)-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C14H14F3N7O2
|
1
|
| 1 |
IC50 = 2642 nM
|
|
|
|
CP0572076
|
5-cyclopropyl-2-methyl-N-[(1R)-1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-3-carboxamide
Show/Hide
|
C19H21N5O2
|
1
|
| 1 |
IC50 = 3314 nM
|
|
|
|
CP0556187
|
2-methyl-N-[(1S)-1-[3-(4-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C16H15F3N6O2
|
1
|
| 1 |
IC50 = 4466 nM
|
|
|
|
CP0557790
|
2-methyl-N-[(1S)-1-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C15H13F3N6O2
|
1
|
| 1 |
IC50 = 5245 nM
|
|
|
|
CP0556188
|
N-[(1S)-1-[3-[2-(2-methoxypropan-2-yl)pyridin-4-yl]-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C19H21F3N6O3
|
1
|
| 1 |
IC50 = 6282 nM
|
|
|
|
CP0557789
|
N-[(1S)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N,2-dimethyl-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C17H15F4N5O2
|
1
|
| 1 |
IC50 = 6489 nM
|
|
|
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CP0558142
|
N-[1-(2,3-dihydro-1H-inden-5-yl)ethyl]-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
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|
C23H25N3O2
|
1
|
| 1 |
IC50 = 9285 nM
|
|
|
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CP0549601
|
5-cyclopropyl-2-methyl-N-[(1S)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]pyrazole-3-carboxamide
Show/Hide
|
C18H19N5O2
|
1
|
| 1 |
IC50 = 11430 nM
|
|
|
|
CP0557791
|
2-methyl-N-[(1S)-1-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C15H13F3N6O2
|
1
|
| 1 |
IC50 = 11800 nM
|
|
|
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CP0537138
|
N-[(1S)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-methyl-5-(trifluoromethyl)pyrazole-3-sulfonamide
Show/Hide
|
C15H13F4N5O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0551765
|
5-cyclopropyl-1-methyl-N-[(1S)-1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]pyrazole-3-carboxamide
Show/Hide
|
C19H21N5O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
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CP0556949
|
2-methyl-N-[(1S)-1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C15H13F3N6O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0557275
|
2-methyl-N-[(1S)-1-[3-(6-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl]-5-(trifluoromethyl)pyrazole-3-carboxamide
Show/Hide
|
C16H15F3N6O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
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CP0560234
|
5-cyclopropyl-2-methyl-N-[(1S)-1-[5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]ethyl]pyrazole-3-carboxamide
Show/Hide
|
C19H21N5O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
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