| Compound ID |
Compound Name |
Compound Formula |
|
CP0434249
|
N-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
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|
C32H49N5O8
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0077025
|
N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)-4-[3-methyl-4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C32H49N5O8
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0440114
|
N-(1-hydroxy-2-methylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C27H41N3O8
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0484236
|
N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C31H47N5O8
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0425738
|
N-[2-(dimethylamino)ethyl]-2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C31H49N5O8
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0499323
|
N-(2-methyl-1-oxo-1-piperidin-1-ylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C32H48N4O8
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0481389
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-phenylmethoxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C24H25F3N2O7
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0447943
|
2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C27H40N4O8
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0185802
|
N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C31H47N5O8
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0479534
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-phenylmethoxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C26H32N2O7
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0465285
|
N-(2-hydroxyethyl)-2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C29H44N4O9
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0377483
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C20H28N2O6
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0447941
|
N-(2-amino-2-oxoethyl)-2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C29H43N5O9
|
1
|
| 1 |
IC50 = 103 nM
|
|
|
|
CP0950546
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-methylthiophenyl)methyl]-5-trifluoromethyl-1H-pyrazole
Show/Hide
|
C18H21F3N2O6S
|
1
|
| 1 |
IC50 = 109 nM
|
|
|
|
CP0447934
|
N-(2-methyl-1-morpholin-4-yl-1-oxopropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C31H46N4O9
|
1
|
| 1 |
IC50 = 124 nM
|
|
|
|
CP0957420
|
4-(2-Phenylethyl)-1H-indazol-3-yl beta-D-glucopyranoside
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|
C21H24N2O6
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0440115
|
N-(3-hydroxypropyl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C26H39N3O8
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0529938
|
(1S,3'R,4'S,5'S,6'R)-5-chloro-6'-(hydroxymethyl)-6-(4-methoxybenzyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
|
C21H23ClO7
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0452237
|
(2S,3R,4S,5S,6R)-2-[[5-tert-butyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C27H34N2O7
|
1
|
| 1 |
IC50 = 203 nM
|
|
|
|
CP0488186
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-hydroxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C19H26N2O7
|
1
|
| 1 |
IC50 = 207 nM
|
|
|
|
CP0440113
|
N-(2-hydroxyethyl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C25H37N3O8
|
1
|
| 1 |
IC50 = 217 nM
|
|
|
|
CP0479535
|
(2S,3R,4S,5S,6R)-2-[[4-[(4-ethylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H30N2O6
|
1
|
| 1 |
IC50 = 223 nM
|
|
|
|
CP0962676
|
4-[(4-Ethylphenyl)methyl]-3-(beta-D-glucopyranosyloxy)-5-methyl-1H-pyrazole
Show/Hide
|
C19H26N2O6
|
1
|
| 1 |
IC50 = 233 nM
|
|
|
|
CP0481383
|
(2S,3R,4S,5S,6R)-2-[[4-[(2,4-dimethylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H30N2O6
|
1
|
| 1 |
IC50 = 246 nM
|
|
|
|
CP0500320
|
(2S,3R,4S,5S,6R)-2-[[5-cyclopropyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C26H30N2O7
|
1
|
| 1 |
IC50 = 278 nM
|
|
|
|
CP0515875
|
(2S,3R,4S,5S,6R)-2-[[4-[(2-fluorophenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C19H25FN2O6
|
1
|
| 1 |
IC50 = 298 nM
|
|
|
|
CP0452239
|
(2S,3R,4S,5S,6R)-2-[[5-ethyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C25H30N2O7
|
1
|
| 1 |
IC50 = 306 nM
|
|
|
|
CP0207318
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-hydroxy-2-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C20H28N2O7
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0899365
|
3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-methylphenyl)methyl]-1H-pyrazole
Show/Hide
|
C18H24N2O6
|
1
|
| 1 |
IC50 = 321 nM
|
|
|
|
CP0848374
|
3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-propylphenyl)methyl]-1H-pyrazole
Show/Hide
|
C20H28N2O6
|
1
|
| 1 |
IC50 = 345 nM
|
|
|
|
CP0447937
|
4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C23H33N3O7
|
1
|
| 1 |
IC50 = 351 nM
|
|
|
|
CP0864400
|
5-Ethyl-3-(beta-D-glucopyranosyloxy)-4-[(4-methylthiophenyl)methyl]-1H-pyrazole
Show/Hide
|
C19H26N2O6S
|
1
|
| 1 |
IC50 = 378 nM
|
|
|
|
CP0447939
|
N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]acetamide
Show/Hide
|
C21H29N3O7
|
1
|
| 1 |
IC50 = 392 nM
|
|
|
|
CP0848373
|
3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-methylthiophenyl)methyl]-1H-pyrazole
Show/Hide
|
C18H24N2O6S
|
1
|
| 1 |
IC50 = 405 nM
|
|
|
|
CP0428005
|
(2S,3R,4S,5S,6R)-2-[[4-[(4-aminophenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C19H27N3O6
|
1
|
| 1 |
IC50 = 422 nM
|
|
|
|
CP0513434
|
(2S,3R,4S,5S,6R)-2-[[4-benzyl-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C17H19F3N2O6
|
1
|
| 1 |
IC50 = 442 nM
|
|
|
|
CP0465287
|
3-amino-N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]propanamide
Show/Hide
|
C22H32N4O7
|
1
|
| 1 |
IC50 = 446 nM
|
|
|
|
CP0957463
|
5-Isopropyl-4-[4-(methylsulfanyl)benzyl]-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
|
C20H28N2O6S
|
1
|
| 1 |
IC50 = 468 nM
|
|
|
|
CP0499948
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-hydroxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C17H19F3N2O7
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0511296
|
N-(2-hydroxyethyl)-N-methyl-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C26H39N3O8
|
1
|
| 1 |
IC50 = 517 nM
|
|
|
|
CP0050531
|
1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)-3-(4-hydroxyphenyl)propan-1-one
Show/Hide
|
C21H24O10
|
1
|
| 1 |
IC50 = 536 nM
|
|
|
|
CP0404716
|
(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(4-ethylbenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
|
C22H25ClO6
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0944866
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-methoxyphenyl)methyl]-5-methyl-1H-pyrazole
Show/Hide
|
C18H24N2O7
|
1
|
| 1 |
IC50 = 626 nM
|
|
|
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CP0479533
|
(2S,3R,4S,5S,6R)-2-[[4-[(2-ethylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H30N2O6
|
1
|
| 1 |
IC50 = 675 nM
|
|
|
|
CP0493998
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-methoxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C20H28N2O7
|
1
|
| 1 |
IC50 = 689 nM
|
|
|
|
CP0414954
|
(1S,3'R,4'S,5'S,6'S)-5-chloro-4-(4-ethylbenzyl)-6'-(fluoromethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
|
C22H24ClFO5
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0417976
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H25ClO5
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0428006
|
N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]propanamide
Show/Hide
|
C22H31N3O7
|
1
|
| 1 |
IC50 = 724 nM
|
|
|
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CP0558118
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C20H28N2O6
|
1
|
| 1 |
IC50 = 725 nM
|
|
|
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CP0440118
|
(2S,3R,4S,5S,6R)-2-[(4-benzyl-5-propan-2-yl-1H-pyrazol-3-yl)oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C19H26N2O6
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1
|
| 1 |
IC50 = 738 nM
|
|
|
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CP0523450
|
N-(2-amino-2-oxoethyl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C25H36N4O8
|
1
|
| 1 |
IC50 = 772 nM
|
|
|
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CP0450417
|
2-amino-N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]acetamide
Show/Hide
|
C21H30N4O7
|
1
|
| 1 |
IC50 = 831 nM
|
|
|
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CP0377484
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[5-methyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C24H28N2O7
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1
|
| 1 |
IC50 = 871 nM
|
|
|
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CP0198642
|
(2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl}-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H25ClO6
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
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CP0484241
|
N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]methanesulfonamide
Show/Hide
|
C20H29N3O8S
|
1
|
| 1 |
IC50 = 931 nM
|
|
|
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CP0414956
|
(1S,3'R,4'S,5'S,6'R)-5-chloro-6'-(hydroxymethyl)-6-(2-methoxy-3-methylbenzyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H25ClO7
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
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CP0475152
|
(1S,3'R,4'S,5'S,6'R)-6'-(azidomethyl)-5-chloro-4-(4-ethylbenzyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H24ClN3O5
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
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CP0490705
|
(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(4-ethoxy-2-methylbenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
|
C23H27ClO7
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
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CP0531172
|
(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(4-fluoro-2-methylbenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
|
C21H22ClFO6
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
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CP0447942
|
5-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]pentanamide
Show/Hide
|
C24H35N3O7
|
1
|
| 1 |
IC50 = 1030 nM
|
|
|
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CP0920794
|
4-[(4-Ethoxyphenyl)methyl]-3-(beta-D-glucopyranosyloxy)-5-methyl-1H-pyrazole
Show/Hide
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C19H26N2O7
|
1
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| 1 |
IC50 = 1030 nM
|
|
|
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CP0500318
|
(2S,3R,4S,5S,6R)-2-[[4-[(4-fluorophenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C19H25FN2O6
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1
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| 1 |
IC50 = 1190 nM
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CP0481384
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-hydroxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C19H26N2O7
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1
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| 1 |
IC50 = 1230 nM
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CP0475790
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(4-ethoxybenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H25ClO7
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1
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| 1 |
IC50 = 1300 nM
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CP0955979
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4-Benzyl-5-methyl-1H-pyrazol-3-yl beta-D-glucopyranoside
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C17H22N2O6
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1
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| 1 |
IC50 = 1320 nM
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CP0452235
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C20H28N2O6
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1
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| 1 |
IC50 = 1330 nM
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CP0465286
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4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]benzamide
Show/Hide
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C20H27N3O7
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1
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| 1 |
IC50 = 1470 nM
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CP0414953
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(2-fluoro-3-methylbenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C21H22ClFO6
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1
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| 1 |
IC50 = 1500 nM
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CP0450418
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N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
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C23H33N3O7
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1
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| 1 |
IC50 = 1500 nM
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CP0496930
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(1S,3'R,4'S,5'S,6'R)-5-chloro-4-((4-ethylphenyl)difluoromethyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H23ClF2O6
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1
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| 1 |
IC50 = 1600 nM
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CP0899366
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3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-propoxyphenyl)methyl]-1H-pyrazole
Show/Hide
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C20H28N2O7
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1
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| 1 |
IC50 = 1630 nM
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CP0944581
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5-Methyl-4-(2-methylbenzyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
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C18H24N2O6
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1
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| 1 |
IC50 = 1630 nM
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CP0888453
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3-(beta-D-Glucopyranosyloxy)-4-[(4-isopropylphenyl)methyl]-5-methyl-1H-pyrazole
Show/Hide
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C20H28N2O6
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1
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| 1 |
IC50 = 1690 nM
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CP0452238
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-phenylmethoxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C24H25F3N2O7
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1
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| 1 |
IC50 = 1720 nM
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CP0499949
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-hydroxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C17H19F3N2O7
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1
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| 1 |
IC50 = 1940 nM
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CP0505498
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3-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]propanamide
Show/Hide
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C22H31N3O7
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1
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| 1 |
IC50 = 1990 nM
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CP0545208
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[5-propan-2-yl-4-[[2-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C20H25F3N2O6
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1
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| 1 |
IC50 = 2430 nM
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CP0495712
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6'-(hydroxymethyl)-6-(4-isopropylbenzyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C23H27ClO6
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1
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| 1 |
IC50 = 2500 nM
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CP0414957
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(1S,3'R,4'S,5'S,6'R)-5-chloro-4-(4-ethylbenzyl)-6'-(methoxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C23H27ClO6
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1
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| 1 |
IC50 = 2700 nM
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CP0952348
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3-(beta-D-Glucopyranosyloxy)-4-[(4-isopropoxyphenyl)methyl]-5-methyl-1H-pyrazole
Show/Hide
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C20H28N2O7
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1
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| 1 |
IC50 = 2780 nM
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CP0398265
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6'-(hydroxymethyl)-6-(4-(trifluoromethoxy)benzyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C21H20ClF3O7
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1
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| 1 |
IC50 = 3100 nM
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CP0473813
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((1S,3'R,4'S,5'S,6'R)-5-chloro-4-(4-ethylbenzyl)-3',4',5'-trihydroxy-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-6'-yl)methyl acetate
Show/Hide
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C24H27ClO7
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1
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| 1 |
IC50 = 3500 nM
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CP0398959
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-hydroxyethoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H31ClO7
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1
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| 1 |
IC50 = 4200 nM
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CP0507251
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-hydroxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C17H19F3N2O7
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1
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| 1 |
IC50 = 4310 nM
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CP0507775
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4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]benzonitrile
Show/Hide
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C20H25N3O6
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1
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| 1 |
IC50 = 4310 nM
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CP0498027
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(1S,3'R,4'S,5'S,6'R)-6-(4-ethylbenzyl)-5-fluoro-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H25FO6
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1
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| 1 |
IC50 = 5300 nM
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CP0513991
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(1S,3'R,4'S,5'S,6'R)-5-chloro-4-(1-(4-ethylphenyl)cyclopropyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C24H27ClO6
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1
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| 1 |
IC50 = 6000 nM
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CP0417996
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2-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]acetamide
Show/Hide
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C21H29N3O7
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1
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| 1 |
IC50 = 6170 nM
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CP0452236
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2-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]benzonitrile
Show/Hide
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C20H25N3O6
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1
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| 1 |
IC50 = 7170 nM
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CP0494000
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-methoxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C20H28N2O7
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1
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| 1 |
IC50 = 7280 nM
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CP0943911
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5-Methyl-4-(3-methylbenzyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
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C18H24N2O6
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1
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| 1 |
IC50 = 8710 nM
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CP0507776
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-phenylmethoxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C24H25F3N2O7
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1
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| 1 |
IC50 = 8930 nM
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CP0493999
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-hydroxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
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C19H26N2O7
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1
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| 1 |
IC50 = 9520 nM
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CP0529939
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(1S,3'R,4'S,5'S,6'R)-6-(4-tert-butylbenzyl)-5-chloro-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C24H29ClO6
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1
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| 1 |
IC50 = 9700 nM
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CP0414952
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(1S,3'R,4'S,5'S,6'R)-6-(4-ethoxybenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H26O7
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1
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| 1 |
IC50 = 10000 nM
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CP0414955
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(2-chloro-4-ethoxybenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H24Cl2O7
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1
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| 1 |
IC50 = 10000 nM
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CP0475151
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(2-ethoxy-4-fluorobenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H24ClFO7
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1
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| 1 |
IC50 = 10000 nM
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CP0502733
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6'-(hydroxymethyl)-6-(4-methoxy-2-methylbenzyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H25ClO7
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1
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| 1 |
IC50 = 10000 nM
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CP0400661
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1-(5-chloro-4-(4-ethylbenzyl)-2-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2Hpyran-2-yl)benzyloxy)propan-2-one
Show/Hide
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C25H31ClO7
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1
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| 1 |
IC50 > 10000 nM
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CP0417974
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-methoxyethoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H33ClO7
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1
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| 1 |
IC50 > 10000 nM
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CP0501978
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(2S,3R,4R,5S,6R)-2-(4-chloro-2-((2,2-difluoroethoxy)methyl)-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H29ClF2O6
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1
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| 1 |
IC50 > 10000 nM
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CP0556609
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[5-methyl-4-[(4-propan-2-yloxyphenyl)methyl]-1-propylpyrazol-3-yl]oxyoxane-3,4,5-triol
Show/Hide
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C23H34N2O7
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1
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| 1 |
IC50 = 10300 nM
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CP0496932
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(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(3-chloro-4-ethoxybenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H24Cl2O7
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1
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| 1 |
IC50 = 10500 nM
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CP0527638
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(2S,3R,4S,5S,6R)-2-[1-ethyl-5-methyl-4-[(4-propan-2-yloxyphenyl)methyl]pyrazol-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C22H32N2O7
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1
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| 1 |
IC50 = 13300 nM
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CP0507630
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(2S,3R,4S,5S,6R)-2-[1,5-dimethyl-4-[(4-propan-2-yloxyphenyl)methyl]pyrazol-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H30N2O7
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1
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| 1 |
IC50 = 13600 nM
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CP0498873
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(1S,3'R,4'S,5'S,6'R)-5-chloro-4-(4-ethylbenzyl)-6'-((2,2,2-trifluoroethoxy)methyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C24H26ClF3O6
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1
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| 1 |
IC50 = 14000 nM
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CP0424638
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Remogliflozin
Show/Hide
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C23H34N2O7
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1
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| 1 |
IC50 = 16600 nM
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CP0421707
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-(2-(prop-2-ynyloxy)ethyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C26H31ClO6
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1
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| 1 |
IC50 > 20000 nM
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CP0960359
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5-Methyl-4-(3-phenylpropyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
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C19H26N2O6
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1
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| 1 |
IC50 = 23700 nM
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CP0514559
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(2S,3R,4R,5S,6R)-2-(2-(2-(allyloxy)ethyl)-4-chloro-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C26H33ClO6
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1
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| 1 |
IC50 = 31000 nM
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CP0956003
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5-Methyl-4-(2-phenylethyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
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C18H24N2O6
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1
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| 1 |
IC50 = 31500 nM
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CP0414958
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((1S,3'R,4'S,5'S,6'R)-5-chloro-3',4',5'-trihydroxy-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-4-yl)(4-ethylphenyl)methanone
Show/Hide
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C22H23ClO7
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1
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| 1 |
IC50 = 43000 nM
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CP0467478
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-hydroxypropoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H33ClO7
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1
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| 1 |
IC50 = 60000 nM
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CP0421706
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(2S,3R,4R,5S,6R)-2-(2-(allyloxymethyl)-4-chloro-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H31ClO6
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1
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| 1 |
IC50 = 91000 nM
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CP0537586
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(1S,3'R,4'S,5'S,6'R)-6'-(aminomethyl)-5-chloro-4-(4-ethylbenzyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
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C22H26ClNO5
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1
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| 1 |
IC50 > 100000 nM
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CP0550335
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GSK-189075
Show/Hide
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C26H38N2O9
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1
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| 1 |
IC50 > 100000 nM
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CP0556610
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(2S,3R,4S,5S,6R)-2-[2,5-dimethyl-4-[(4-propan-2-yloxyphenyl)methyl]pyrazol-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H30N2O7
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1
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| 1 |
IC50 > 100000 nM
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CP0400662
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((prop-2-ynyloxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H29ClO6
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1
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| 1 |
IC50 > 1000 nM
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CP0238397
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-(methoxymethyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H29ClO6
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1
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| 1 |
IC50 > 2000 nM
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CP0482964
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethoxybenzyl)-2-(2-methoxyethyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H31ClO7
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1
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| 1 |
IC50 > 2000 nM
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CP0438889
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-fluoroethoxy)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H30ClFO6
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1
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| 1 |
IC50 > 5000 nM
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