| Compound ID |
Compound Name |
Compound Formula |
|
CP0490304
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-cyclopropylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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|
C22H25ClO5
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0490306
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclopropyloxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C24H29ClO7
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0397286
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclobutyloxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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|
C25H31ClO7
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0508471
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(1-hydroxycyclopropyl)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H25ClO6
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0198642
|
(2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl}-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H25ClO6
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0962676
|
4-[(4-Ethylphenyl)methyl]-3-(beta-D-glucopyranosyloxy)-5-methyl-1H-pyrazole
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|
C19H26N2O6
|
2
|
| 1 |
IC50 = 3.9 nM
|
|
|
| 2 |
IC50 = 190 nM
|
|
|
|
CP0499421
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclopentyloxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C26H33ClO7
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0526691
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethenylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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|
C21H23ClO5
|
1
|
| 1 |
IC50 = 4.4 nM
|
|
|
|
CP0848373
|
3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-methylthiophenyl)methyl]-1H-pyrazole
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|
C18H24N2O6S
|
2
|
| 1 |
IC50 = 4.9 nM
|
|
|
| 2 |
IC50 = 84 nM
|
|
|
|
CP0499392
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-prop-2-enoxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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|
C24H29ClO7
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0452238
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-phenylmethoxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C24H25F3N2O7
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0526692
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-prop-2-ynoxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C24H27ClO7
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0440114
|
N-(1-hydroxy-2-methylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C27H41N3O8
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0848374
|
3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-propylphenyl)methyl]-1H-pyrazole
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|
C20H28N2O6
|
2
|
| 1 |
IC50 = 8.8 nM
|
|
|
| 2 |
IC50 = 441 nM
|
|
|
|
CP0499419
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-hydroxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C19H21ClO6
|
1
|
| 1 |
IC50 = 9.4 nM
|
|
|
|
CP0375566
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(3-cyclopropylprop-2-ynoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C25H27ClO6
|
1
|
| 1 |
IC50 = 9.6 nM
|
|
|
|
CP0473989
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethynylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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|
C21H21ClO5
|
1
|
| 1 |
IC50 = 9.6 nM
|
|
|
|
CP0388468
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-[2-(1-methylcyclopropyl)oxyethoxy]phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C25H31ClO7
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0512496
|
4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]benzonitrile
Show/Hide
|
C20H20ClNO5
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0952348
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-isopropoxyphenyl)methyl]-5-methyl-1H-pyrazole
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|
C20H28N2O7
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
IC50 = 181 nM
|
|
|
|
CP0920794
|
4-[(4-Ethoxyphenyl)methyl]-3-(beta-D-glucopyranosyloxy)-5-methyl-1H-pyrazole
Show/Hide
|
C19H26N2O7
|
2
|
| 1 |
IC50 = 10.8 nM
|
|
|
| 2 |
IC50 = 185 nM
|
|
|
|
CP0899365
|
3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-methylphenyl)methyl]-1H-pyrazole
Show/Hide
|
C18H24N2O6
|
2
|
| 1 |
IC50 = 12.2 nM
|
|
|
| 2 |
IC50 = 280 nM
|
|
|
|
CP0944866
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-methoxyphenyl)methyl]-5-methyl-1H-pyrazole
Show/Hide
|
C18H24N2O7
|
2
|
| 1 |
IC50 = 12.3 nM
|
|
|
| 2 |
IC50 = 383 nM
|
|
|
|
CP0899366
|
3-(beta-D-Glucopyranosyloxy)-5-methyl-4-[(4-propoxyphenyl)methyl]-1H-pyrazole
Show/Hide
|
C20H28N2O7
|
2
|
| 1 |
IC50 = 15.4 nM
|
|
|
| 2 |
IC50 = 702 nM
|
|
|
|
CP0888453
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-isopropylphenyl)methyl]-5-methyl-1H-pyrazole
Show/Hide
|
C20H28N2O6
|
2
|
| 1 |
IC50 = 16.2 nM
|
|
|
| 2 |
IC50 = 441 nM
|
|
|
|
CP0950546
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-methylthiophenyl)methyl]-5-trifluoromethyl-1H-pyrazole
Show/Hide
|
C18H21F3N2O6S
|
2
|
| 1 |
IC50 = 16.3 nM
|
|
|
| 2 |
IC50 = 679 nM
|
|
|
|
CP0434249
|
N-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C32H49N5O8
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0424638
|
Remogliflozin
Show/Hide
|
C23H34N2O7
|
2
|
| 1 |
IC50 = 18.4 nM
|
|
|
| 2 |
IC50 = 369 nM
|
|
|
|
CP0484236
|
N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C31H47N5O8
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0050531
|
1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)-3-(4-hydroxyphenyl)propan-1-one
Show/Hide
|
C21H24O10
|
1
|
| 1 |
IC50 = 38 nM
|
|
|
|
CP0499323
|
N-(2-methyl-1-oxo-1-piperidin-1-ylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C32H48N4O8
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0527638
|
(2S,3R,4S,5S,6R)-2-[1-ethyl-5-methyl-4-[(4-propan-2-yloxyphenyl)methyl]pyrazol-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H32N2O7
|
1
|
| 1 |
IC50 = 43.4 nM
|
|
|
|
CP0425738
|
N-[2-(dimethylamino)ethyl]-2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C31H49N5O8
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0864400
|
5-Ethyl-3-(beta-D-glucopyranosyloxy)-4-[(4-methylthiophenyl)methyl]-1H-pyrazole
Show/Hide
|
C19H26N2O6S
|
2
|
| 1 |
IC50 = 51.2 nM
|
|
|
| 2 |
IC50 = 509 nM
|
|
|
|
CP0556609
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[5-methyl-4-[(4-propan-2-yloxyphenyl)methyl]-1-propylpyrazol-3-yl]oxyoxane-3,4,5-triol
Show/Hide
|
C23H34N2O7
|
1
|
| 1 |
IC50 = 66.1 nM
|
|
|
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CP0479535
|
(2S,3R,4S,5S,6R)-2-[[4-[(4-ethylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H30N2O6
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0447943
|
2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C27H40N4O8
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0957420
|
4-(2-Phenylethyl)-1H-indazol-3-yl beta-D-glucopyranoside
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|
C21H24N2O6
|
1
|
| 1 |
IC50 = 86 nM
|
|
|
|
CP0490305
|
2-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenoxy]acetic acid
Show/Hide
|
C21H23ClO8
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0447934
|
N-(2-methyl-1-morpholin-4-yl-1-oxopropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C31H46N4O9
|
1
|
| 1 |
IC50 = 98 nM
|
|
|
|
CP0507630
|
(2S,3R,4S,5S,6R)-2-[1,5-dimethyl-4-[(4-propan-2-yloxyphenyl)methyl]pyrazol-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H30N2O7
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0465285
|
N-(2-hydroxyethyl)-2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C29H44N4O9
|
1
|
| 1 |
IC50 = 151 nM
|
|
|
|
CP0499948
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-hydroxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C17H19F3N2O7
|
1
|
| 1 |
IC50 = 154 nM
|
|
|
|
CP0957463
|
5-Isopropyl-4-[4-(methylsulfanyl)benzyl]-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
|
C20H28N2O6S
|
1
|
| 1 |
IC50 = 154 nM
|
|
|
|
CP0955979
|
4-Benzyl-5-methyl-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
|
C17H22N2O6
|
1
|
| 1 |
IC50 = 181 nM
|
|
|
|
CP0447941
|
N-(2-amino-2-oxoethyl)-2-methyl-2-[4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanoylamino]propanamide
Show/Hide
|
C29H43N5O9
|
1
|
| 1 |
IC50 = 209 nM
|
|
|
|
CP0377483
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C20H28N2O6
|
1
|
| 1 |
IC50 = 231 nM
|
|
|
|
CP0488186
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-hydroxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C19H26N2O7
|
1
|
| 1 |
IC50 = 285 nM
|
|
|
|
CP0440115
|
N-(3-hydroxypropyl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C26H39N3O8
|
1
|
| 1 |
IC50 = 319 nM
|
|
|
|
CP0513434
|
(2S,3R,4S,5S,6R)-2-[[4-benzyl-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C17H19F3N2O6
|
1
|
| 1 |
IC50 = 342 nM
|
|
|
|
CP0875197
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-isobutylphenyl)methyl]-5-methyl-1H-pyrazole
Show/Hide
|
C21H30N2O6
|
1
|
| 1 |
IC50 = 346 nM
|
|
|
|
CP0511296
|
N-(2-hydroxyethyl)-N-methyl-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C26H39N3O8
|
1
|
| 1 |
IC50 = 358 nM
|
|
|
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CP0077025
|
N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)-4-[3-methyl-4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C32H49N5O8
|
1
|
| 1 |
IC50 = 371 nM
|
|
|
|
CP0493998
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-methoxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
Show/Hide
|
C20H28N2O7
|
1
|
| 1 |
IC50 = 377 nM
|
|
|
|
CP0942271
|
3-(beta-D-Glucopyranosyloxy)-4-[(4-methoxyphenyl)methyl]-5-trifluoromethyl-1H-pyrazole
Show/Hide
|
C18H21F3N2O7
|
1
|
| 1 |
IC50 = 415 nM
|
|
|
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CP0526693
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-hydroxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H25ClO7
|
1
|
| 1 |
IC50 = 428 nM
|
|
|
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CP0447942
|
5-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]pentanamide
Show/Hide
|
C24H35N3O7
|
1
|
| 1 |
IC50 = 457 nM
|
|
|
|
CP0440113
|
N-(2-hydroxyethyl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C25H37N3O8
|
1
|
| 1 |
IC50 = 608 nM
|
|
|
|
CP0963840
|
(2S,3R,4S,5S,6R)-2-[4-(4-Ethyl-benzyl)-5-trifluoromethyl-1H-pyrazol-3-yloxy]-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C19H23F3N2O6
|
1
|
| 1 |
IC50 = 634 nM
|
|
|
|
CP0943911
|
5-Methyl-4-(3-methylbenzyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
|
C18H24N2O6
|
1
|
| 1 |
IC50 = 757 nM
|
|
|
|
CP0864399
|
3-(beta-D-Glucopyranosyloxy)-1-methyl-4-[(4-methylthiophenyl)methyl]-5-trifluoromethylpyrazole
Show/Hide
|
C19H23F3N2O6S
|
1
|
| 1 |
IC50 = 835 nM
|
|
|
|
CP0944581
|
5-Methyl-4-(2-methylbenzyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
Show/Hide
|
C18H24N2O6
|
1
|
| 1 |
IC50 = 914 nM
|
|
|
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CP0484241
|
N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]methanesulfonamide
Show/Hide
|
C20H29N3O8S
|
1
|
| 1 |
IC50 = 936 nM
|
|
|
|
CP0523450
|
N-(2-amino-2-oxoethyl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
Show/Hide
|
C25H36N4O8
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
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CP0447937
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4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
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C23H33N3O7
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1
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| 1 |
IC50 = 1070 nM
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CP0515875
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(2S,3R,4S,5S,6R)-2-[[4-[(2-fluorophenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C19H25FN2O6
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1
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| 1 |
IC50 = 1390 nM
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CP0428005
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(2S,3R,4S,5S,6R)-2-[[4-[(4-aminophenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C19H27N3O6
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1
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| 1 |
IC50 = 1590 nM
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CP0185802
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N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)-4-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
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C31H47N5O8
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1
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| 1 |
IC50 = 1730 nM
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CP0440118
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(2S,3R,4S,5S,6R)-2-[(4-benzyl-5-propan-2-yl-1H-pyrazol-3-yl)oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C19H26N2O6
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1
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| 1 |
IC50 = 2020 nM
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CP0465286
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4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]benzamide
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C20H27N3O7
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1
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| 1 |
IC50 = 2470 nM
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CP0550335
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GSK-189075
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C26H38N2O9
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1
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| 1 |
IC50 = 2530 nM
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CP0505498
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3-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]propanamide
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C22H31N3O7
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1
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| 1 |
IC50 = 2540 nM
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CP0499949
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-hydroxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C17H19F3N2O7
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1
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| 1 |
IC50 = 2790 nM
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CP0447939
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N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]acetamide
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C21H29N3O7
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1
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| 1 |
IC50 = 3090 nM
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CP0507775
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4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]benzonitrile
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C20H25N3O6
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1
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| 1 |
IC50 = 3580 nM
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CP0960359
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5-Methyl-4-(3-phenylpropyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
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C19H26N2O6
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1
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| 1 |
IC50 = 3950 nM
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CP0450418
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N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]butanamide
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C23H33N3O7
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1
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| 1 |
IC50 = 3980 nM
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CP0500318
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(2S,3R,4S,5S,6R)-2-[[4-[(4-fluorophenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C19H25FN2O6
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1
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| 1 |
IC50 = 4140 nM
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CP0450417
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2-amino-N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]acetamide
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C21H30N4O7
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1
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| 1 |
IC50 = 4700 nM
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CP0377484
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[5-methyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C24H28N2O7
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1
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| 1 |
IC50 = 5010 nM
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CP0428006
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N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]propanamide
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C22H31N3O7
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1
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| 1 |
IC50 = 5100 nM
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CP0956003
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5-Methyl-4-(2-phenylethyl)-1H-pyrazol-3-yl beta-D-glucopyranoside
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C18H24N2O6
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1
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| 1 |
IC50 = 5290 nM
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CP0465287
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3-amino-N-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]propanamide
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C22H32N4O7
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1
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| 1 |
IC50 = 5620 nM
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CP0507776
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-phenylmethoxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C24H25F3N2O7
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1
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| 1 |
IC50 = 5680 nM
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CP0452235
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C20H28N2O6
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1
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| 1 |
IC50 = 5980 nM
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CP0481383
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(2S,3R,4S,5S,6R)-2-[[4-[(2,4-dimethylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H30N2O6
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1
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| 1 |
IC50 = 6010 nM
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CP0207318
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(4-hydroxy-2-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C20H28N2O7
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1
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| 1 |
IC50 = 6890 nM
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CP0417996
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2-[4-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]phenyl]acetamide
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C21H29N3O7
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1
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| 1 |
IC50 = 9950 nM
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CP0481384
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(3-hydroxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C19H26N2O7
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1
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| 1 |
IC50 = 13300 nM
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CP0452239
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(2S,3R,4S,5S,6R)-2-[[5-ethyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C25H30N2O7
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1
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| 1 |
IC50 = 13900 nM
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CP0481389
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-phenylmethoxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C24H25F3N2O7
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1
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| 1 |
IC50 = 14000 nM
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CP0479533
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(2S,3R,4S,5S,6R)-2-[[4-[(2-ethylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H30N2O6
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1
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| 1 |
IC50 = 14100 nM
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CP0507251
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-hydroxyphenyl)methyl]-5-(trifluoromethyl)-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C17H19F3N2O7
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1
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| 1 |
IC50 = 14900 nM
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CP0558118
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-methylphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C20H28N2O6
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1
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| 1 |
IC50 = 18500 nM
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CP0545208
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[5-propan-2-yl-4-[[2-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C20H25F3N2O6
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1
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| 1 |
IC50 = 60500 nM
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CP0452237
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(2S,3R,4S,5S,6R)-2-[[5-tert-butyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
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C27H34N2O7
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1
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| 1 |
IC50 = 64700 nM
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CP0452236
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2-[[5-propan-2-yl-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-1H-pyrazol-4-yl]methyl]benzonitrile
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C20H25N3O6
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1
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| 1 |
IC50 = 65700 nM
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CP0479534
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-phenylmethoxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C26H32N2O7
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1
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| 1 |
IC50 = 74000 nM
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CP0493999
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-hydroxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol
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C19H26N2O7
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1
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| 1 |
IC50 = 75900 nM
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CP0944865
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1-(4-Methylsulfanyl-benzyl)-5-trifluoromethyl-1,2-dihydro-pyrazol-3-one
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C12H11F3N2OS
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1
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| 1 |
IC50 > 100000 nM
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CP0556610
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(2S,3R,4S,5S,6R)-2-[2,5-dimethyl-4-[(4-propan-2-yloxyphenyl)methyl]pyrazol-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H30N2O7
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1
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| 1 |
IC50 > 1000 nM
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