| Compound ID |
Compound Name |
Compound Formula |
|
CP0390921
|
2-[5-(diethylsulfamoylamino)pentylamino]-4-pyridin-2-yl-1,3-thiazole
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|
C17H27N5O2S2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0393035
|
2-methoxy-5-methyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]benzenesulfonamide
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|
C21H26N4O3S2
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0452383
|
N-[5-(4,5-dihydro-[1]benzothiepino[5,4-d][1,3]thiazol-2-ylamino)pentyl]propane-2-sulfonamide
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|
C19H27N3O2S3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0391227
|
2,4-dimethyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]-1,3-thiazole-5-sulfonamide
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|
C18H23N5O2S3
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0452382
|
N-[5-[(4-thiophen-3-yl-1,3-thiazol-2-yl)amino]pentyl]propane-2-sulfonamide
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|
C15H23N3O2S3
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0085089
|
2-[5-(dimethylsulfamoylamino)pentylamino]-4-pyridin-2-yl-1,3-thiazole
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|
C15H23N5O2S2
|
1
|
| 1 |
Ki = 7.6 nM
|
|
|
|
CP0041441
|
2-Nitro-N-(4-{[(1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-amino]-methyl}-cyclohexylmethyl)-benzenesulfonamide
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|
C25H33N3O4S
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0488658
|
2-fluoro-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]benzenesulfonamide
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|
C19H21FN4O2S2
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0393872
|
N-[[4-[(naphthalen-2-ylmethylamino)methyl]cyclohexyl]methyl]-2-(trifluoromethyl)benzenesulfonamide
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|
C26H29F3N2O2S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0461105
|
2-amino-N-[[4-[(1,2,3,4-tetrahydronaphthalen-2-ylmethylamino)methyl]cyclohexyl]methyl]benzenesulfonamide
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|
C25H35N3O2S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0454764
|
N-[[4-[(1,2,3,4-tetrahydronaphthalen-2-ylmethylamino)methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide
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|
C29H36N2O2S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0494335
|
N-[[4-[(2,3-dihydro-1,4-benzodioxin-6-ylmethylamino)methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide
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|
C27H32N2O4S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0440253
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]propane-2-sulfonamide
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|
C16H24N4O2S2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0383458
|
2-Nitro-N-(4-{[(quinolin-2-ylmethyl)-amino]-methyl}-cyclohexylmethyl)-benzenesulfonamide
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|
C24H28N4O4S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0460756
|
N-[[4-[(1,2,3,4-tetrahydronaphthalen-2-ylmethylamino)methyl]cyclohexyl]methyl]naphthalene-2-sulfonamide
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|
C29H36N2O2S
|
2
|
| 1 |
Ki = 14 nM
|
|
|
| 2 |
Ki = 32 nM
|
|
|
|
CP0463643
|
N-[[4-[[[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]amino]methyl]cyclohexyl]methyl]naphthalene-1-sulfonamide
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|
C27H33ClN2O3S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0496113
|
3,5-dimethyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]-1,2-oxazole-4-sulfonamide
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|
C18H23N5O3S2
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0463724
|
N-[[4-[(naphthalen-1-ylmethylamino)methyl]cyclohexyl]methyl]-2-(trifluoromethyl)benzenesulfonamide
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|
C26H29F3N2O2S
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0438595
|
2-Nitro-N-(4-{[(quinolin-4-ylmethyl)-amino]-methyl}-cyclohexylmethyl)-benzenesulfonamide
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|
C24H28N4O4S
|
1
|
| 1 |
Ki = 28 nM
|
|
|
|
CP0393036
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]thiophene-2-sulfonamide
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|
C17H20N4O2S3
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0388726
|
N-[5-[[4-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3-thiazol-2-yl]amino]pentyl]propane-2-sulfonamide
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|
C16H26N4O2S3
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0440248
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]morpholine-4-sulfonamide
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|
C17H25N5O3S2
|
1
|
| 1 |
Ki = 38 nM
|
|
|
|
CP0390898
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]cyclopropanesulfonamide
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|
C16H22N4O2S2
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0437300
|
1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid [6-(2-nitro-benzenesulfonylamino)-hexyl]-amide
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|
C23H29N3O5S
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0488657
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]butane-2-sulfonamide
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|
C17H26N4O2S2
|
1
|
| 1 |
Ki = 49 nM
|
|
|
|
CP0388717
|
2-[5-[bis(2-methoxyethyl)sulfamoylamino]pentylamino]-4-pyridin-2-yl-1,3-thiazole
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|
C19H31N5O4S2
|
1
|
| 1 |
Ki = 60 nM
|
|
|
|
CP0388716
|
2,6-dimethyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]morpholine-4-sulfonamide
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|
C19H29N5O3S2
|
1
|
| 1 |
Ki = 75 nM
|
|
|
|
CP0496109
|
N-[5-[(4-thiophen-3-yl-1,3-thiazol-2-yl)amino]pentyl]methanesulfonamide
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|
C13H19N3O2S3
|
1
|
| 1 |
Ki = 80 nM
|
|
|
|
CP0377714
|
1-(3,4-dichlorophenyl)-3-[[4-[(naphthalen-1-ylsulfonylamino)methyl]cyclohexyl]methyl]urea
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|
C25H27Cl2N3O3S
|
1
|
| 1 |
Ki = 95 nM
|
|
|
|
CP0409650
|
1-naphthalen-1-yl-3-[[4-[[(2-nitrophenyl)sulfonylamino]methyl]cyclohexyl]methyl]urea
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|
C25H28N4O5S
|
1
|
| 1 |
Ki = 103 nM
|
|
|
|
CP0440252
|
1,1,1-trifluoro-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]methanesulfonamide
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|
C14H17F3N4O2S2
|
1
|
| 1 |
Ki = 109 nM
|
|
|
|
CP0393034
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]cyclohexanesulfonamide
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|
C19H28N4O2S2
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0528870
|
N-[6-(naphthalen-2-ylmethylamino)hexyl]naphthalene-2-sulfonamide
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|
C27H30N2O2S
|
1
|
| 1 |
Ki = 123 nM
|
|
|
|
CP0475166
|
N-[5-[[4-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3-thiazol-2-yl]amino]pentyl]methanesulfonamide
Show/Hide
|
C14H22N4O2S3
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0496110
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]ethanesulfonamide
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|
C15H22N4O2S2
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0432446
|
1-naphthalen-1-yl-3-[6-[(2-nitrophenyl)sulfonylamino]hexyl]urea
Show/Hide
|
C23H26N4O5S
|
1
|
| 1 |
Ki = 151 nM
|
|
|
|
CP0440254
|
1,3,5-trimethyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]pyrazole-4-sulfonamide
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|
C19H26N6O2S2
|
1
|
| 1 |
Ki = 159 nM
|
|
|
|
CP0393032
|
N-[5-[(4-thiophen-2-yl-1,3-thiazol-2-yl)amino]pentyl]methanesulfonamide
Show/Hide
|
C13H19N3O2S3
|
1
|
| 1 |
Ki = 170 nM
|
|
|
|
CP0463496
|
4-methyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]piperazine-1-sulfonamide
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|
C18H28N6O2S2
|
1
|
| 1 |
Ki = 170 nM
|
|
|
|
CP0535486
|
2-[(4-methylphenyl)sulfonylamino]-N-[[4-[(naphthalen-2-ylsulfonylamino)methyl]cyclohexyl]methyl]-3-phenylpropanamide
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|
C34H39N3O5S2
|
1
|
| 1 |
Ki = 199 nM
|
|
|
|
CP0488204
|
1-naphthalen-1-yl-3-[6-(naphthalen-1-ylsulfonylamino)hexyl]urea
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|
C27H29N3O3S
|
1
|
| 1 |
Ki = 231 nM
|
|
|
|
CP0452380
|
benzyl 4-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentylsulfamoyl]piperidine-1-carboxylate
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|
C26H33N5O4S2
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0388719
|
1-cyclopentyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]methanesulfonamide
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|
C19H28N4O2S2
|
1
|
| 1 |
Ki = 250 nM
|
|
|
|
CP0391225
|
N-[2-[2-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]ethoxy]ethyl]propane-2-sulfonamide
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|
C15H22N4O3S2
|
1
|
| 1 |
Ki = 290 nM
|
|
|
|
CP0440251
|
N-[5-[[4-(5-chloro-3-methyl-1-benzothiophen-2-yl)-1,3-thiazol-2-yl]amino]pentyl]methanesulfonamide
Show/Hide
|
C18H22ClN3O2S3
|
1
|
| 1 |
Ki = 360 nM
|
|
|
|
CP0466567
|
N-[6-[(2-nitrophenyl)sulfonylamino]hexyl]naphthalene-2-carboxamide
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|
C23H25N3O5S
|
1
|
| 1 |
Ki = 412 nM
|
|
|
|
CP0498097
|
2-[(4-methylphenyl)sulfonylamino]-N-[6-(naphthalen-1-ylsulfonylamino)hexyl]-3-phenylpropanamide
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|
C32H37N3O5S2
|
1
|
| 1 |
Ki = 426 nM
|
|
|
|
CP0482922
|
N-[5-[(4-pyridin-3-yl-1,3-thiazol-2-yl)amino]pentyl]propane-2-sulfonamide
Show/Hide
|
C16H24N4O2S2
|
1
|
| 1 |
Ki = 515 nM
|
|
|
|
CP0496347
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]methanesulfonamide
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|
C14H20N4O2S2
|
1
|
| 1 |
Ki = 530 nM
|
|
|
|
CP0498092
|
1-naphthalen-1-yl-3-[4-[(2-nitrophenyl)sulfonylamino]butyl]urea
Show/Hide
|
C21H22N4O5S
|
1
|
| 1 |
Ki = 724 nM
|
|
|
|
CP0535477
|
1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid [6-(naphthalene-1-sulfonylamino)-hexyl]-amide
Show/Hide
|
C27H32N2O3S
|
1
|
| 1 |
Ki = 724 nM
|
|
|
|
CP0535986
|
1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid {4-[(8-nitro-naphthalene-2-sulfonylamino)-methyl]-cyclohexylmethyl}-amide
Show/Hide
|
C29H33N3O5S
|
1
|
| 1 |
Ki = 724 nM
|
|
|
|
CP0496348
|
N-[5-[[4-[1-(benzenesulfonyl)pyrrol-3-yl]-1,3-thiazol-2-yl]amino]pentyl]methanesulfonamide
Show/Hide
|
C19H24N4O4S3
|
1
|
| 1 |
Ki = 740 nM
|
|
|
|
CP0390919
|
4-pyridin-2-yl-2-[5-(sulfamoylamino)pentylamino]-1,3-thiazole
Show/Hide
|
C13H19N5O2S2
|
1
|
| 1 |
Ki = 803 nM
|
|
|
|
CP0393038
|
1-methyl-N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]imidazole-4-sulfonamide
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|
C17H22N6O2S2
|
1
|
| 1 |
Ki = 1122 nM
|
|
|
|
CP0482923
|
N-[5-[[4-(3-methylpyrazin-2-yl)-1,3-thiazol-2-yl]amino]pentyl]propane-2-sulfonamide
Show/Hide
|
C16H25N5O2S2
|
1
|
| 1 |
Ki = 1851 nM
|
|
|
|
CP0496111
|
N-[5-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]pentyl]piperidine-4-sulfonamide
Show/Hide
|
C18H27N5O2S2
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0464624
|
1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid {4-[(naphthalene-1-sulfonylamino)-methyl]-cyclohexylmethyl}-amide
Show/Hide
|
C29H34N2O3S
|
1
|
| 1 |
Ki = 4120 nM
|
|
|
|
CP0488656
|
N-[5-[[4-(1,3-thiazol-2-yl)-1,3-thiazol-2-yl]amino]pentyl]methanesulfonamide
Show/Hide
|
C12H18N4O2S3
|
1
|
| 1 |
Ki = 4300 nM
|
|
|
|
CP0437688
|
N-[2-(4-propan-2-ylsulfonylpiperazin-1-yl)ethyl]-4-pyridin-2-yl-1,3-thiazol-2-amine
Show/Hide
|
C17H25N5O2S2
|
1
|
| 1 |
Ki = 5000 nM
|
|
|
|
CP0497133
|
1,2,3,4-Tetrahydro-naphthalene-2-carboxylic acid {4-[(naphthalene-2-sulfonylamino)-methyl]-cyclohexylmethyl}-amide
Show/Hide
|
C29H34N2O3S
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
