Compound ID |
Compound Name |
Compound Formula |
CP0369408
|
1-phenyl-7-pyridin-3-yl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline
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|
C21H16N4
|
1
|
1 |
IC50 = 84 nM
|
|
|
CP0048211
|
3-cyclopropyl-2-(4-ethyl-5-fluoropyridin-3-yl)-6-fluoroimidazo[1,2-a]pyridine
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|
C17H15F2N3
|
1
|
1 |
IC50 = 5700 nM
|
|
|
CP0133117
|
1-cyclopropyl-5,6-difluoro-2-(5-fluoropyridin-3-yl)benzimidazole
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|
C15H10F3N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0401274
|
1-cyclopropyl-5,6-difluoro-2-(5-fluoro-4-methylpyridin-3-yl)benzimidazole
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|
C16H12F3N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0643522
|
2-(5-(1-cyclopropyl-6-fluoro-1H-benzo[d]imidazol-2-yl)pyridin-3-yl)propan-2-ol
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|
C18H18FN3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0667085
|
2-(5-(1-cyclopropyl-5,6-difluoro-1H-benzo[d]imidazol-2-yl)pyridin-3-yl)propan-2-ol
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|
C18H17F2N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0040950
|
7-[5-(2-methoxypropan-2-yl)pyridin-3-yl]-1-methyl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline
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|
C20H22N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0065022
|
(2S)-1,1,1-trifluoro-2-[5-(1-methyl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinolin-7-yl)pyridin-3-yl]propan-2-ol
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|
C19H17F3N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0252415
|
methyl 5-(1-methyl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinolin-7-yl)pyridine-3-carboxylate
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|
C18H16N4O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0091723
|
6-chloro-3-cyclopropyl-7-fluoro-2-(5-fluoropyridin-3-yl)imidazo[1,2-a]pyridine
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|
C15H10ClF2N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0190104
|
3-cyclopropyl-6-fluoro-2-(5-fluoro-4-methylpyridin-3-yl)imidazo[1,2-a]pyridine
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|
C16H13F2N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0294276
|
(2S)-2-[5-(3-cyclopropyl-6-fluoroimidazo[1,2-a]pyridin-2-yl)pyridin-3-yl]-1,1,1-trifluoropropan-2-ol
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|
C18H15F4N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0108244
|
(2R)-1,1,1-trifluoro-2-[5-(3-methylindazol-1-yl)pyridin-3-yl]propan-2-ol
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|
C16H14F3N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0180854
|
2-[5-[4-(trifluoromethyl)indazol-1-yl]pyridin-3-yl]propan-2-ol
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|
C16H14F3N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0201912
|
2-[5-(4-fluoro-3-methylindazol-1-yl)pyridin-3-yl]propan-2-ol
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|
C16H16FN3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0240397
|
(2S)-1,1,1-trifluoro-2-[5-[3-(trifluoromethyl)indazol-1-yl]pyridin-3-yl]propan-2-ol
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|
C16H11F6N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0244010
|
(2S)-1,1,1-trifluoro-2-[5-(3-methylindazol-1-yl)pyridin-3-yl]propan-2-ol
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|
C16H14F3N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|