Compound ID |
Compound Name |
Compound Formula |
CP0497145
|
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-methyl-amide} 1-[(2-nitro-phenyl)-amide]
Show/Hide
|
C34H35N5O5
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0373447
|
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
Show/Hide
|
C33H33N5O5
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0465354
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-3-phenyl-propyl]-amide
Show/Hide
|
C31H35ClN4O2S
|
1
|
1 |
IC50 = 206 nM
|
|
|
CP0495118
|
(S)-1-(2-Fluoro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C30H33FN4O2S
|
1
|
1 |
IC50 = 290 nM
|
|
|
CP0487373
|
(S)-1-(2-Methyl-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C31H36N4O2S
|
1
|
1 |
IC50 = 410 nM
|
|
|
CP0496277
|
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
Show/Hide
|
C31H32N6O5
|
1
|
1 |
IC50 = 410 nM
|
|
|
CP0408418
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide} 1-(2-chloro-benzylamide)
Show/Hide
|
C30H33ClN4O3
|
1
|
1 |
IC50 = 590 nM
|
|
|
CP0945726
|
(R)-1-(2-Nitro-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
Show/Hide
|
C33H33N5O4S
|
1
|
1 |
IC50 = 800 nM
|
|
|
CP0448249
|
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-(3,4-dichloro-phenyl)-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
Show/Hide
|
C29H29Cl2N5O5
|
1
|
1 |
IC50 = 820 nM
|
|
|
CP0536868
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(4-nitro-phenyl)-amide]
Show/Hide
|
C33H33N5O5
|
1
|
1 |
IC50 = 1000 nM
|
|
|
CP0560252
|
(R)-1-(2-Bromo-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C29H31BrN4O2S
|
1
|
1 |
IC50 = 1000 nM
|
|
|
CP0437588
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-phenethyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C31H35ClN4O2S
|
1
|
1 |
IC50 = 2500 nM
|
|
|
CP0881403
|
1-[N-cyano-N'-(2-nitro-phenyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
Show/Hide
|
C34H33N7O4
|
1
|
1 |
IC50 = 2700 nM
|
|
|
CP0429038
|
(R)-1-(2-Chloro-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C29H31ClN4O2S
|
1
|
1 |
IC50 = 3200 nM
|
|
|
CP0504122
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid {(S)-1-[2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-amide
Show/Hide
|
C32H34ClN5O2S
|
1
|
1 |
IC50 = 3700 nM
|
|
|
CP0495113
|
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
Show/Hide
|
C33H33N5O5
|
1
|
1 |
IC50 = 7100 nM
|
|
|
CP0462784
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 1-[(2-acetylamino-phenyl)-amide] 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide}
Show/Hide
|
C35H37N5O4
|
1
|
1 |
IC50 = 9600 nM
|
|
|
CP0510133
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-pyridin-4-ylmethyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C29H32ClN5O2S
|
1
|
1 |
IC50 = 10000 nM
|
|
|
CP0510135
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 1-[(2-amino-phenyl)-amide] 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide}
Show/Hide
|
C33H35N5O3
|
1
|
1 |
IC50 = 19700 nM
|
|
|
CP0537037
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-2-benzo[b]thiophen-2-yl-1-(benzyl-methyl-carbamoyl)-ethyl]-amide
Show/Hide
|
C32H33ClN4O2S2
|
1
|
1 |
IC50 = 29400 nM
|
|
|
CP0897890
|
(R)-1-[N-(2-Nitro-phenyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
Show/Hide
|
C33H34N6O4
|
1
|
1 |
IC50 = 60600 nM
|
|
|
CP0169323
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
Show/Hide
|
C33H33N5O5
|
1
|
1 |
IC50 = 82400 nM
|
|
|
CP0402190
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-phenyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C29H31ClN4O2S
|
1
|
1 |
IC50 = 100000 nM
|
|
|
CP0916651
|
(R)-1-(2-Nitro-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C29H31N5O4S
|
1
|
1 |
IC50 = 100000 nM
|
|
|
CP0432584
|
2-({(S)-2-[(S)-1-(Benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethylcarbamoyl]-pyrrolidine-1-carbonyl}-amino)-benzoic acid methyl ester
Show/Hide
|
C35H36N4O5
|
1
|
1 |
Ki = 0.3 nM
|
|
|
CP0536882
|
(S)-1-[N-(2-Chloro-benzyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
Show/Hide
|
C34H36ClN5O2
|
1
|
1 |
Ki = 0.5 nM
|
|
|
CP0380432
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-fluoro-phenyl)-amide]
Show/Hide
|
C33H33FN4O3
|
1
|
1 |
Ki = 0.7 nM
|
|
|
CP0383503
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
Show/Hide
|
C34H35ClN4O2S
|
1
|
1 |
Ki = 0.7 nM
|
|
|
CP0536875
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-carbamoyl-phenyl)-amide]
Show/Hide
|
C34H35N5O4
|
1
|
1 |
Ki = 0.8 nM
|
|
|
CP0498239
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-phenylamide
Show/Hide
|
C33H34N4O3
|
1
|
1 |
Ki = 0.88 nM
|
|
|
CP0384346
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-methoxymethyl-phenyl)-amide]
Show/Hide
|
C35H38N4O4
|
1
|
1 |
Ki = 1 nM
|
|
|
CP0374982
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(4-cyano-phenyl)-amide]
Show/Hide
|
C34H33N5O3
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0406053
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-cyano-phenyl)-amide]
Show/Hide
|
C34H33N5O3
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0384345
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-methyl-amide
Show/Hide
|
C35H37ClN4O2S
|
1
|
1 |
Ki = 1.7 nM
|
|
|
CP0428947
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-hydroxymethyl-phenyl)-amide]
Show/Hide
|
C34H36N4O4
|
1
|
1 |
Ki = 1.7 nM
|
|
|
CP0515012
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(4-fluoro-phenyl)-amide]
Show/Hide
|
C33H33FN4O3
|
1
|
1 |
Ki = 2.2 nM
|
|
|
CP0437590
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-nitro-phenyl)-amide]
Show/Hide
|
C33H33N5O5
|
1
|
1 |
Ki = 2.3 nM
|
|
|
CP0516101
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-(2-chloro-benzylamide)
Show/Hide
|
C34H35ClN4O3
|
1
|
1 |
Ki = 2.3 nM
|
|
|
CP0536891
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-hydroxy-phenyl)-amide]
Show/Hide
|
C33H34N4O4
|
1
|
1 |
Ki = 2.6 nM
|
|
|
CP0536482
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-fluoro-phenyl)-amide]
Show/Hide
|
C33H33FN4O3
|
1
|
1 |
Ki = 3.5 nM
|
|
|
CP0403568
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-methylcarbamoyl-phenyl)-amide]
Show/Hide
|
C35H37N5O4
|
1
|
1 |
Ki = 3.8 nM
|
|
|
CP0403567
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-cyano-phenyl)-amide]
Show/Hide
|
C34H33N5O3
|
1
|
1 |
Ki = 4.2 nM
|
|
|
CP0465100
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-(1-methyl-1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C33H36ClN5O2S
|
1
|
1 |
Ki = 4.7 nM
|
|
|
CP0373430
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-(3,4-dichloro-phenyl)-ethyl]-amide
Show/Hide
|
C30H31Cl3N4O2S
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0380690
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-carbamoyl-phenyl)-amide]
Show/Hide
|
C34H35N5O4
|
1
|
1 |
Ki = 5 nM
|
|
|
CP0496216
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-dimethylcarbamoyl-phenyl)-amide]
Show/Hide
|
C36H39N5O4
|
1
|
1 |
Ki = 6.1 nM
|
|
|
CP0479724
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-pyridin-3-ylamide
Show/Hide
|
C32H33N5O3
|
1
|
1 |
Ki = 6.7 nM
|
|
|
CP0374979
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-biphenyl-4-yl-ethyl]-amide
Show/Hide
|
C36H37ClN4O2S
|
1
|
1 |
Ki = 7.2 nM
|
|
|
CP0510134
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-1-yl-ethyl]-amide
Show/Hide
|
C34H35ClN4O2S
|
1
|
1 |
Ki = 13.7 nM
|
|
|
CP0537870
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide
Show/Hide
|
C32H34ClN5O2S
|
1
|
1 |
Ki = 16.7 nM
|
|
|
CP0506554
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-naphthalen-1-ylmethyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C34H35ClN4O2S
|
1
|
1 |
Ki = 17.1 nM
|
|
|
CP0373448
|
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-trifluoromethyl-phenyl)-amide]
Show/Hide
|
C34H33F3N4O3
|
1
|
1 |
Ki = 18.2 nM
|
|
|
CP0538459
|
(S)-1-[N-(2-Chloro-benzyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C30H34ClN5O2
|
1
|
1 |
Ki = 18.5 nM
|
|
|
CP0374986
|
(S)-1-(2,6-Dichloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C30H32Cl2N4O2S
|
1
|
1 |
Ki = 25.9 nM
|
|
|
CP0467590
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid {(S)-1-[(3,5-bis-trifluoromethyl-benzyl)-methyl-carbamoyl]-2-phenyl-ethyl}-amide
Show/Hide
|
C32H31ClF6N4O2S
|
1
|
1 |
Ki = 26.9 nM
|
|
|
CP0409642
|
(S)-1-(2-Trifluoromethyl-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C31H33F3N4O2S
|
1
|
1 |
Ki = 27.2 nM
|
|
|
CP0529642
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2,2-diphenyl-ethyl]-amide
Show/Hide
|
C36H37ClN4O2S
|
1
|
1 |
Ki = 29.4 nM
|
|
|
CP0504233
|
(S)-1-(2-Bromo-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C30H33BrN4O2S
|
1
|
1 |
Ki = 29.7 nM
|
|
|
CP0496276
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C30H33ClN4O2S
|
1
|
1 |
Ki = 29.9 nM
|
|
|
CP0487563
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-naphthalen-2-ylmethyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C34H35ClN4O2S
|
1
|
1 |
Ki = 36 nM
|
|
|
CP0516036
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-methyl-amide
Show/Hide
|
C31H35ClN4O2S
|
1
|
1 |
Ki = 38 nM
|
|
|
CP0464784
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid ((S)-1-{[2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-2-phenyl-ethyl)-amide
Show/Hide
|
C33H36ClN5O2S
|
1
|
1 |
Ki = 48 nM
|
|
|
CP0854641
|
(S)-1-(2-Nitro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C30H33N5O4S
|
1
|
1 |
Ki = 77.6 nM
|
|
|
CP0514141
|
(S)-1-(3,5-Bis-trifluoromethyl-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C32H32F6N4O2S
|
1
|
1 |
Ki = 78.6 nM
|
|
|
CP0376581
|
(2S)-N-[(2S)-1-[benzyl(methyl)amino]-1-oxo-3-phenylpropan-2-yl]-1-(phenylcarbamothioyl)pyrrolidine-2-carboxamide
Show/Hide
|
C29H32N4O2S
|
1
|
1 |
Ki = 80 nM
|
|
|
CP0537776
|
2-({(S)-2-[(S)-1-(Benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethylcarbamoyl]-pyrrolidine-1-carbonyl}-amino)-benzoic acid
Show/Hide
|
C34H34N4O5
|
1
|
1 |
Ki = 172 nM
|
|
|
CP0467452
|
(S)-1-Benzylthiocarbamoyl-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C30H34N4O2S
|
1
|
1 |
Ki = 1010 nM
|
|
|
CP0430325
|
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-benzyl-2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxo-ethyl]-amide
Show/Hide
|
C31H33ClN4O2S
|
1
|
1 |
Ki = 8000 nM
|
|
|