Brief Information of the Cell Line and Protein
Cell Line ID: CL000053 , COS-7
Synonyms
Cos-7
COS 7
Cos 7
COS7
Cos7
CV-1 in Origin Simian-7
Category Transformed cell line
Organism
Chlorocebus aethiops (Green monkey)
Cellosaurus ID
CVCL_0224
Protein ID: PT01410 , Substance-P receptor
Gene Name TACR1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P25103
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000053  Protein ID: PT01410
 
Compound ID Compound Name Compound Formula
CP0497145
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-methyl-amide} 1-[(2-nitro-phenyl)-amide]
   Show/Hide
C34H35N5O5
 1
1
IC50 = 140 nM
   TI
   LI
   LO
   TS
CP0373447
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
   Show/Hide
C33H33N5O5
 1
1
IC50 = 160 nM
   TI
   LI
   LO
   TS
CP0465354
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-3-phenyl-propyl]-amide
   Show/Hide
C31H35ClN4O2S
 1
1
IC50 = 206 nM
   TI
   LI
   LO
   TS
CP0495118
(S)-1-(2-Fluoro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C30H33FN4O2S
 1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS
CP0487373
(S)-1-(2-Methyl-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C31H36N4O2S
 1
1
IC50 = 410 nM
   TI
   LI
   LO
   TS
CP0496277
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
   Show/Hide
C31H32N6O5
 1
1
IC50 = 410 nM
   TI
   LI
   LO
   TS
CP0408418
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide} 1-(2-chloro-benzylamide)
   Show/Hide
C30H33ClN4O3
 1
1
IC50 = 590 nM
   TI
   LI
   LO
   TS
CP0945726
(R)-1-(2-Nitro-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
   Show/Hide
C33H33N5O4S
 1
1
IC50 = 800 nM
   TI
   LI
   LO
   TS
CP0448249
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(R)-1-(benzyl-methyl-carbamoyl)-2-(3,4-dichloro-phenyl)-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
   Show/Hide
C29H29Cl2N5O5
 1
1
IC50 = 820 nM
   TI
   LI
   LO
   TS
CP0536868
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(4-nitro-phenyl)-amide]
   Show/Hide
C33H33N5O5
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0560252
(R)-1-(2-Bromo-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C29H31BrN4O2S
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0437588
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-phenethyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C31H35ClN4O2S
 1
1
IC50 = 2500 nM
   TI
   LI
   LO
   TS
CP0881403
1-[N-cyano-N'-(2-nitro-phenyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
   Show/Hide
C34H33N7O4
 1
1
IC50 = 2700 nM
   TI
   LI
   LO
   TS
CP0429038
(R)-1-(2-Chloro-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C29H31ClN4O2S
 1
1
IC50 = 3200 nM
   TI
   LI
   LO
   TS
CP0504122
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid {(S)-1-[2-(1H-indol-3-yl)-ethylcarbamoyl]-2-phenyl-ethyl}-amide
   Show/Hide
C32H34ClN5O2S
 1
1
IC50 = 3700 nM
   TI
   LI
   LO
   TS
CP0495113
(R)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
   Show/Hide
C33H33N5O5
 1
1
IC50 = 7100 nM
   TI
   LI
   LO
   TS
CP0462784
(S)-Pyrrolidine-1,2-dicarboxylic acid 1-[(2-acetylamino-phenyl)-amide] 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide}
   Show/Hide
C35H37N5O4
 1
1
IC50 = 9600 nM
   TI
   LI
   LO
   TS
CP0510133
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-pyridin-4-ylmethyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C29H32ClN5O2S
 1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0510135
(S)-Pyrrolidine-1,2-dicarboxylic acid 1-[(2-amino-phenyl)-amide] 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide}
   Show/Hide
C33H35N5O3
 1
1
IC50 = 19700 nM
   TI
   LI
   LO
   TS
CP0537037
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-2-benzo[b]thiophen-2-yl-1-(benzyl-methyl-carbamoyl)-ethyl]-amide
   Show/Hide
C32H33ClN4O2S2
 1
1
IC50 = 29400 nM
   TI
   LI
   LO
   TS
CP0897890
(R)-1-[N-(2-Nitro-phenyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
   Show/Hide
C33H34N6O4
 1
1
IC50 = 60600 nM
   TI
   LI
   LO
   TS
CP0169323
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-nitro-phenyl)-amide]
   Show/Hide
C33H33N5O5
 1
1
IC50 = 82400 nM
   TI
   LI
   LO
   TS
CP0402190
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-phenyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C29H31ClN4O2S
 1
1
IC50 = 100000 nM
   TI
   LI
   LO
   TS
CP0916651
(R)-1-(2-Nitro-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(R)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C29H31N5O4S
 1
1
IC50 = 100000 nM
   TI
   LI
   LO
   TS
CP0432584
2-({(S)-2-[(S)-1-(Benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethylcarbamoyl]-pyrrolidine-1-carbonyl}-amino)-benzoic acid methyl ester
   Show/Hide
C35H36N4O5
 1
1
Ki = 0.3 nM
   TI
   LI
   LO
   TS
CP0536882
(S)-1-[N-(2-Chloro-benzyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
   Show/Hide
C34H36ClN5O2
 1
1
Ki = 0.5 nM
   TI
   LI
   LO
   TS
CP0380432
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-fluoro-phenyl)-amide]
   Show/Hide
C33H33FN4O3
 1
1
Ki = 0.7 nM
   TI
   LI
   LO
   TS
CP0383503
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide
   Show/Hide
C34H35ClN4O2S
 1
1
Ki = 0.7 nM
   TI
   LI
   LO
   TS
CP0536875
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-carbamoyl-phenyl)-amide]
   Show/Hide
C34H35N5O4
 1
1
Ki = 0.8 nM
   TI
   LI
   LO
   TS
CP0498239
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-phenylamide
   Show/Hide
C33H34N4O3
 1
1
Ki = 0.88 nM
   TI
   LI
   LO
   TS
CP0384346
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-methoxymethyl-phenyl)-amide]
   Show/Hide
C35H38N4O4
 1
1
Ki = 1 nM
   TI
   LI
   LO
   TS
CP0374982
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(4-cyano-phenyl)-amide]
   Show/Hide
C34H33N5O3
 1
1
Ki = 1.1 nM
   TI
   LI
   LO
   TS
CP0406053
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-cyano-phenyl)-amide]
   Show/Hide
C34H33N5O3
 1
1
Ki = 1.1 nM
   TI
   LI
   LO
   TS
CP0384345
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-methyl-amide
   Show/Hide
C35H37ClN4O2S
 1
1
Ki = 1.7 nM
   TI
   LI
   LO
   TS
CP0428947
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-hydroxymethyl-phenyl)-amide]
   Show/Hide
C34H36N4O4
 1
1
Ki = 1.7 nM
   TI
   LI
   LO
   TS
CP0515012
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(4-fluoro-phenyl)-amide]
   Show/Hide
C33H33FN4O3
 1
1
Ki = 2.2 nM
   TI
   LI
   LO
   TS
CP0437590
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-nitro-phenyl)-amide]
   Show/Hide
C33H33N5O5
 1
1
Ki = 2.3 nM
   TI
   LI
   LO
   TS
CP0516101
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-(2-chloro-benzylamide)
   Show/Hide
C34H35ClN4O3
 1
1
Ki = 2.3 nM
   TI
   LI
   LO
   TS
CP0536891
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-hydroxy-phenyl)-amide]
   Show/Hide
C33H34N4O4
 1
1
Ki = 2.6 nM
   TI
   LI
   LO
   TS
CP0536482
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-fluoro-phenyl)-amide]
   Show/Hide
C33H33FN4O3
 1
1
Ki = 3.5 nM
   TI
   LI
   LO
   TS
CP0403568
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-methylcarbamoyl-phenyl)-amide]
   Show/Hide
C35H37N5O4
 1
1
Ki = 3.8 nM
   TI
   LI
   LO
   TS
CP0403567
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-cyano-phenyl)-amide]
   Show/Hide
C34H33N5O3
 1
1
Ki = 4.2 nM
   TI
   LI
   LO
   TS
CP0465100
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-(1-methyl-1H-indol-3-yl)-ethyl]-amide
   Show/Hide
C33H36ClN5O2S
 1
1
Ki = 4.7 nM
   TI
   LI
   LO
   TS
CP0373430
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-(3,4-dichloro-phenyl)-ethyl]-amide
   Show/Hide
C30H31Cl3N4O2S
 1
1
Ki = 5 nM
   TI
   LI
   LO
   TS
CP0380690
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(3-carbamoyl-phenyl)-amide]
   Show/Hide
C34H35N5O4
 1
1
Ki = 5 nM
   TI
   LI
   LO
   TS
CP0496216
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-dimethylcarbamoyl-phenyl)-amide]
   Show/Hide
C36H39N5O4
 1
1
Ki = 6.1 nM
   TI
   LI
   LO
   TS
CP0479724
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-pyridin-3-ylamide
   Show/Hide
C32H33N5O3
 1
1
Ki = 6.7 nM
   TI
   LI
   LO
   TS
CP0374979
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-biphenyl-4-yl-ethyl]-amide
   Show/Hide
C36H37ClN4O2S
 1
1
Ki = 7.2 nM
   TI
   LI
   LO
   TS
CP0510134
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-1-yl-ethyl]-amide
   Show/Hide
C34H35ClN4O2S
 1
1
Ki = 13.7 nM
   TI
   LI
   LO
   TS
CP0537870
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide
   Show/Hide
C32H34ClN5O2S
 1
1
Ki = 16.7 nM
   TI
   LI
   LO
   TS
CP0506554
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-naphthalen-1-ylmethyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C34H35ClN4O2S
 1
1
Ki = 17.1 nM
   TI
   LI
   LO
   TS
CP0373448
(S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethyl]-amide} 1-[(2-trifluoromethyl-phenyl)-amide]
   Show/Hide
C34H33F3N4O3
 1
1
Ki = 18.2 nM
   TI
   LI
   LO
   TS
CP0538459
(S)-1-[N-(2-Chloro-benzyl)-carbamimidoyl]-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C30H34ClN5O2
 1
1
Ki = 18.5 nM
   TI
   LI
   LO
   TS
CP0374986
(S)-1-(2,6-Dichloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C30H32Cl2N4O2S
 1
1
Ki = 25.9 nM
   TI
   LI
   LO
   TS
CP0467590
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid {(S)-1-[(3,5-bis-trifluoromethyl-benzyl)-methyl-carbamoyl]-2-phenyl-ethyl}-amide
   Show/Hide
C32H31ClF6N4O2S
 1
1
Ki = 26.9 nM
   TI
   LI
   LO
   TS
CP0409642
(S)-1-(2-Trifluoromethyl-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C31H33F3N4O2S
 1
1
Ki = 27.2 nM
   TI
   LI
   LO
   TS
CP0529642
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2,2-diphenyl-ethyl]-amide
   Show/Hide
C36H37ClN4O2S
 1
1
Ki = 29.4 nM
   TI
   LI
   LO
   TS
CP0504233
(S)-1-(2-Bromo-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C30H33BrN4O2S
 1
1
Ki = 29.7 nM
   TI
   LI
   LO
   TS
CP0496276
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C30H33ClN4O2S
 1
1
Ki = 29.9 nM
   TI
   LI
   LO
   TS
CP0487563
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(methyl-naphthalen-2-ylmethyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C34H35ClN4O2S
 1
1
Ki = 36 nM
   TI
   LI
   LO
   TS
CP0516036
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-methyl-amide
   Show/Hide
C31H35ClN4O2S
 1
1
Ki = 38 nM
   TI
   LI
   LO
   TS
CP0464784
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid ((S)-1-{[2-(1H-indol-3-yl)-ethyl]-methyl-carbamoyl}-2-phenyl-ethyl)-amide
   Show/Hide
C33H36ClN5O2S
 1
1
Ki = 48 nM
   TI
   LI
   LO
   TS
CP0854641
(S)-1-(2-Nitro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C30H33N5O4S
 1
1
Ki = 77.6 nM
   TI
   LI
   LO
   TS
CP0514141
(S)-1-(3,5-Bis-trifluoromethyl-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C32H32F6N4O2S
 1
1
Ki = 78.6 nM
   TI
   LI
   LO
   TS
CP0376581
(2S)-N-[(2S)-1-[benzyl(methyl)amino]-1-oxo-3-phenylpropan-2-yl]-1-(phenylcarbamothioyl)pyrrolidine-2-carboxamide
   Show/Hide
C29H32N4O2S
 1
1
Ki = 80 nM
   TI
   LI
   LO
   TS
CP0537776
2-({(S)-2-[(S)-1-(Benzyl-methyl-carbamoyl)-2-naphthalen-2-yl-ethylcarbamoyl]-pyrrolidine-1-carbonyl}-amino)-benzoic acid
   Show/Hide
C34H34N4O5
 1
1
Ki = 172 nM
   TI
   LI
   LO
   TS
CP0467452
(S)-1-Benzylthiocarbamoyl-pyrrolidine-2-carboxylic acid [(S)-1-(benzyl-methyl-carbamoyl)-2-phenyl-ethyl]-amide
   Show/Hide
C30H34N4O2S
 1
1
Ki = 1010 nM
   TI
   LI
   LO
   TS
CP0430325
(S)-1-(2-Chloro-benzylthiocarbamoyl)-pyrrolidine-2-carboxylic acid [(S)-1-benzyl-2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxo-ethyl]-amide
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C31H33ClN4O2S
 1
1
Ki = 8000 nM
   TI
   LI
   LO
   TS