| Compound ID |
Compound Name |
Compound Formula |
|
CP0426334
|
methyl N-[1-[[(1R,2S)-2-[benzyl(methyl)carbamoyl]-2-(3,4-dichlorophenyl)cyclopropyl]methyl]-4-phenylpiperidin-4-yl]carbamate
Show/Hide
|
C32H35Cl2N3O3
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0512756
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methyl-2-((4-(2-oxo-2-(pyrrolidin-1-yl)ethyl)piperazin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C29H35Cl2FN4O2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0489233
|
(1S,2R)-1-(3,4-dichlorophenyl)-2-((3-(4-(N,N-dimethylsulfamoyl)piperazin-1-yl)azetidin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C28H36Cl2FN5O3S
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0426335
|
(1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-2-((4-(3,3-dimethylureido)-4-phenylpiperidin-1-yl)methyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C33H38Cl2N4O2
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0516565
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methyl-2-((4-(2-morpholinoacetyl)piperazin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C29H35Cl2FN4O3
|
1
|
| 1 |
Ki = 3.3 nM
|
|
|
|
CP0513054
|
N'-[1-[[(1R,2S)-2-[benzyl(methyl)carbamoyl]-2-(3,4-dichlorophenyl)cyclopropyl]methyl]-4-phenylpiperidin-4-yl]-N'-methyloxamide
Show/Hide
|
C33H36Cl2N4O3
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0426336
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methyl-2-((4-(2-morpholinoethyl)piperazin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C29H37Cl2FN4O2
|
1
|
| 1 |
Ki = 3.7 nM
|
|
|
|
CP0498917
|
(1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2-((4-(N-methylacetamido)-4-phenylpiperidin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C33H37Cl2N3O2
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0489226
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-methyl-N-[[4-(trifluoromethyl)phenyl]methyl]cyclopropane-1-carboxamide
Show/Hide
|
C33H34Cl2F3N3O2
|
1
|
| 1 |
Ki = 4.6 nM
|
|
|
|
CP0489224
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-methyl-N-[(2-methylphenyl)methyl]cyclopropane-1-carboxamide
Show/Hide
|
C33H37Cl2N3O2
|
1
|
| 1 |
Ki = 5.3 nM
|
|
|
|
CP0399281
|
(1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2-((4-(3-methylureido)-4-phenylpiperidin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C32H36Cl2N4O2
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
|
CP0378685
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methyl-2-((4-(pyrrolidin-1-ylsulfonyl)piperazin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C27H33Cl2FN4O3S
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0513051
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H34Cl2FN3O2
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0057704
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-benzyl-1-(3,4-dichlorophenyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H35Cl2N3O2
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0498914
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(2,4-dimethoxyphenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C34H39Cl2N3O4
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0409511
|
(1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2-((4-phenyl-4-(piperidine-1-carbonyl)piperidin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C36H41Cl2N3O2
|
1
|
| 1 |
Ki = 6.1 nM
|
|
|
|
CP0409512
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methyl-2-((4-(2-(piperidin-1-yl)acetyl)piperazin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C30H37Cl2FN4O2
|
1
|
| 1 |
Ki = 7.3 nM
|
|
|
|
CP0498916
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(3,4-dimethylphenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C34H40FN3O2
|
1
|
| 1 |
Ki = 7.3 nM
|
|
|
|
CP0513052
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-methyl-N-[(4-methylphenyl)methyl]cyclopropane-1-carboxamide
Show/Hide
|
C33H37Cl2N3O2
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0051744
|
(1S,2R)-1-(3,4-dichlorophenyl)-2-((4-(N,N-dimethylsulfamoyl)piperazin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C25H31Cl2FN4O3S
|
1
|
| 1 |
Ki = 7.6 nM
|
|
|
|
CP0489232
|
(1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2-((4-(methylsulfonamido)-4-phenylpiperidin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C31H35Cl2N3O3S
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0381520
|
(1S,2R)-2-((4-(2-(azepan-1-yl)acetyl)piperazin-1-yl)methyl)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C31H39Cl2FN4O2
|
1
|
| 1 |
Ki = 8.7 nM
|
|
|
|
CP0543425
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-N-[(4-chlorophenyl)methyl]-1-(3,4-dichlorophenyl)-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H34Cl3N3O2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0381516
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(3-fluorophenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H34Cl2FN3O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0477713
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methyl-2-((4-(2-(pyrrolidin-1-yl)acetyl)piperazin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C29H35Cl2FN4O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0512755
|
(1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2-((4-phenyl-4-ureidopiperidin-1-yl)methyl)cyclopropanecarboxamide
Show/Hide
|
C31H34Cl2N4O2
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0498913
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H33Cl4N3O2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0543424
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(2-methoxyphenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C33H37Cl2N3O3
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0543427
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-methyl-N-(thiophen-3-ylmethyl)cyclopropane-1-carboxamide
Show/Hide
|
C30H33Cl2N3O2S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0487295
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(4-methoxyphenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C33H37Cl2N3O3
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0512722
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(2,4-dichlorophenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H33Cl4N3O2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0469075
|
(1S,2R)-1-(3,4-dichlorophenyl)-2-((4-(3-(dimethylamino)-3-oxopropyl)piperazin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C28H35Cl2FN4O2
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0465489
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(2-fluorophenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H34Cl2FN3O2
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0487294
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-N-[(2-chlorophenyl)methyl]-1-(3,4-dichlorophenyl)-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H34Cl3N3O2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0438299
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(3,5-dichlorophenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H33Cl4N3O2
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0426333
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-N-[(3-chlorophenyl)methyl]-1-(3,4-dichlorophenyl)-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H34Cl3N3O2
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0489227
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(2,3-dichlorophenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C32H33Cl4N3O2
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0487296
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-methyl-N-[(4-methylsulfanylphenyl)methyl]cyclopropane-1-carboxamide
Show/Hide
|
C33H37Cl2N3O2S
|
1
|
| 1 |
Ki = 28 nM
|
|
|
|
CP0378058
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(3-chlorophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H35ClFN3O2
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0543426
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(3,5-dimethoxyphenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C34H39Cl2N3O4
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0505785
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(3-methoxyphenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C33H37Cl2N3O3
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0377247
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(4-chlorophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H35ClFN3O2
|
1
|
| 1 |
Ki = 36 nM
|
|
|
|
CP0509374
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methyl-1-p-tolylcyclopropanecarboxamide
Show/Hide
|
C33H38FN3O2
|
1
|
| 1 |
Ki = 37 nM
|
|
|
|
CP0381518
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methyl-1-m-tolylcyclopropanecarboxamide
Show/Hide
|
C33H38FN3O2
|
1
|
| 1 |
Ki = 40 nM
|
|
|
|
CP0489229
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(3,4-difluorophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H34F3N3O2
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0489225
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-methyl-N-[[3-(trifluoromethyl)phenyl]methyl]cyclopropane-1-carboxamide
Show/Hide
|
C33H34Cl2F3N3O2
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0404959
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-1-(3-methoxyphenyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C33H38FN3O3
|
1
|
| 1 |
Ki = 56 nM
|
|
|
|
CP0487297
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-1-(4-fluorophenyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H35F2N3O2
|
1
|
| 1 |
Ki = 67 nM
|
|
|
|
CP0512723
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-[(3,4-dimethoxyphenyl)methyl]-N-methylcyclopropane-1-carboxamide
Show/Hide
|
C34H39Cl2N3O4
|
1
|
| 1 |
Ki = 67 nM
|
|
|
|
CP0498915
|
2-[(4-acetamido-4-phenylpiperidin-1-yl)methyl]-1-(3,4-dichlorophenyl)-N-methyl-N-(thiophen-2-ylmethyl)cyclopropane-1-carboxamide
Show/Hide
|
C30H33Cl2N3O2S
|
1
|
| 1 |
Ki = 70 nM
|
|
|
|
CP0505784
|
(1R,2S)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-benzyl-1-(3,4-dichlorophenyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H35Cl2N3O2
|
1
|
| 1 |
Ki = 83 nM
|
|
|
|
CP0489231
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(3,5-dichlorophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H34Cl2FN3O2
|
1
|
| 1 |
Ki = 90 nM
|
|
|
|
CP0409510
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methyl-1-(thiophen-2-yl)cyclopropanecarboxamide
Show/Hide
|
C30H34FN3O2S
|
1
|
| 1 |
Ki = 93 nM
|
|
|
|
CP0477712
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methyl-1-(thiophen-3-yl)cyclopropanecarboxamide
Show/Hide
|
C30H34FN3O2S
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0377248
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-1-(3-fluorophenyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C32H35F2N3O2
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0438302
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(benzo[d][1,3]dioxol-5-yl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C33H36FN3O4
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0509349
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-2-((isopropylamino)methyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C22H25Cl2FN2O
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0498919
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-N-methyl-2-((propylamino)methyl)cyclopropanecarboxamide
Show/Hide
|
C22H25Cl2FN2O
|
1
|
| 1 |
Ki = 150 nM
|
|
|
|
CP0469074
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methyl-1-(3-(trifluoromethyl)phenyl)cyclopropanecarboxamide
Show/Hide
|
C33H35F4N3O2
|
1
|
| 1 |
Ki = 210 nM
|
|
|
|
CP0489228
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(4-cyanophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C33H35FN4O2
|
1
|
| 1 |
Ki = 270 nM
|
|
|
|
CP0438301
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-1-(4-methoxyphenyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C33H38FN3O3
|
1
|
| 1 |
Ki = 350 nM
|
|
|
|
CP0513053
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methyl-1-(4-(trifluoromethyl)phenyl)cyclopropanecarboxamide
Show/Hide
|
C33H35F4N3O2
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0409508
|
(1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)methyl)-1-(3-cyanophenyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Show/Hide
|
C33H35FN4O2
|
1
|
| 1 |
Ki = 1900 nM
|
|
|
