| Compound ID |
Compound Name |
Compound Formula |
|
CP0203139
|
(2R)-7-cyclopropylsulfonyl-4,17,20-trimethyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6,8,10(21),16(20),17-hexaene-3,12-dione
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|
C33H34N4O6S
|
1
|
| 1 |
Ki = 4.2 nM
|
|
|
|
CP0534211
|
2-[(2R,5R)-17,20-dimethyl-3,12-dioxo-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6(21),7,9,16(20),17-hexaen-5-yl]acetic acid
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|
C31H30N4O6
|
1
|
| 1 |
Ki = 9.6 nM
|
|
|
|
CP0476604
|
(2R)-7-ethylsulfonyl-4-methyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6,8,10(21),16(20),17-hexaene-3,12-dione
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|
C30H30N4O6S
|
1
|
| 1 |
Ki = 61 nM
|
|
|
|
CP0534552
|
3-[[(2R)-17-ethyl-4-methyl-3,12-dioxo-7-propan-2-ylsulfanyl-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaen-2-yl]amino]benzamide
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|
C31H36N4O4S
|
1
|
| 1 |
Ki = 91 nM
|
|
|
|
CP0558573
|
ethyl 2-[(2R,5R)-17,20-dimethyl-3,12-dioxo-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6(21),7,9,16(20),17-hexaen-5-yl]acetate
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|
C33H34N4O6
|
1
|
| 1 |
Ki = 360 nM
|
|
|
|
CP0476605
|
(2R,8R)-20,23-dimethyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-16-oxa-4,14-diazatetracyclo[17.2.2.19,13.04,8]tetracosa-1(22),9(24),10,12,19(23),20-hexaene-3,15-dione
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|
C32H32N4O4
|
1
|
| 1 |
Ki = 840 nM
|
|
|
|
CP0454480
|
3-[[(2R)-4-methyl-3,12-dioxo-7-propan-2-ylsulfonyl-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6,8,10(21),16(20),17-hexaen-2-yl]amino]benzamide
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|
C29H32N4O6S
|
1
|
| 1 |
Ki = 940 nM
|
|
|
|
CP0465819
|
4,17,20-trimethyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6(21),7,9,16(20),17-hexaene-3,12-dione
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|
C30H30N4O4
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
|
CP0541571
|
3-[(17,20-diethyl-3,12-dioxo-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6(21),7,9,16,19-hexaen-2-yl)amino]benzamide
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|
C29H32N4O4
|
1
|
| 1 |
Ki = 2100 nM
|
|
|
|
CP0548151
|
3-[(17-ethyl-3,12-dioxo-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6(21),7,9,16,19-hexaen-2-yl)amino]benzamide
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|
C27H28N4O4
|
1
|
| 1 |
Ki = 9200 nM
|
|
|
|
CP0454481
|
3-[(3,12-dioxo-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6(21),7,9,16(20),17-hexaen-2-yl)amino]benzamide
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|
C25H24N4O4
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
